IE40588B1 - 3-acylamino-6-amino-3,4-dihydro-2-pyridones and their use as medicaments - Google Patents
3-acylamino-6-amino-3,4-dihydro-2-pyridones and their use as medicamentsInfo
- Publication number
- IE40588B1 IE40588B1 IE246/75A IE24675A IE40588B1 IE 40588 B1 IE40588 B1 IE 40588B1 IE 246/75 A IE246/75 A IE 246/75A IE 24675 A IE24675 A IE 24675A IE 40588 B1 IE40588 B1 IE 40588B1
- Authority
- IE
- Ireland
- Prior art keywords
- sub
- alkyl
- straight
- formula
- branched chain
- Prior art date
Links
- 239000003814 drug Substances 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 6
- 125000003342 alkenyl group Chemical group 0.000 abstract 3
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 125000003118 aryl group Chemical group 0.000 abstract 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 2
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 2
- IYFFBKXNBQQSAA-UHFFFAOYSA-N 3,6-diamino-3,4-dihydro-1h-pyridin-2-one Chemical class NC1CC=C(N)NC1=O IYFFBKXNBQQSAA-UHFFFAOYSA-N 0.000 abstract 1
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 1
- 102100035233 Furin Human genes 0.000 abstract 1
- 101001022148 Homo sapiens Furin Proteins 0.000 abstract 1
- 101000601394 Homo sapiens Neuroendocrine convertase 2 Proteins 0.000 abstract 1
- 101000701936 Homo sapiens Signal peptidase complex subunit 1 Proteins 0.000 abstract 1
- 102100037732 Neuroendocrine convertase 2 Human genes 0.000 abstract 1
- 239000003513 alkali Substances 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- -1 amidinoacetic acid ester Chemical class 0.000 abstract 1
- 230000003197 catalytic effect Effects 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 125000000392 cycloalkenyl group Chemical group 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000002541 furyl group Chemical group 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 150000002367 halogens Chemical group 0.000 abstract 1
- 239000003049 inorganic solvent Substances 0.000 abstract 1
- 229910001867 inorganic solvent Inorganic materials 0.000 abstract 1
- 125000005956 isoquinolyl group Chemical group 0.000 abstract 1
- 125000001624 naphthyl group Chemical group 0.000 abstract 1
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 1
- 125000004076 pyridyl group Chemical group 0.000 abstract 1
- 125000000714 pyrimidinyl group Chemical group 0.000 abstract 1
- 125000005493 quinolyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
- 125000001544 thienyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
- C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Stabilization Of Oscillater, Synchronisation, Frequency Synthesizers (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19742406200 DE2406200A1 (de) | 1974-02-09 | 1974-02-09 | Verfahren zur herstellung von neuen 3,6-diamino-3,4-dihydropyridonen-2 und ihre verwendung als arzneimittel |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE40588L IE40588L (en) | 1975-08-09 |
| IE40588B1 true IE40588B1 (en) | 1979-07-04 |
Family
ID=5906985
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE246/75A IE40588B1 (en) | 1974-02-09 | 1975-02-07 | 3-acylamino-6-amino-3,4-dihydro-2-pyridones and their use as medicaments |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US4001259A (en:Method) |
| JP (1) | JPS50108269A (en:Method) |
| AT (1) | AT339904B (en:Method) |
| BE (1) | BE825246A (en:Method) |
| CA (1) | CA1049525A (en:Method) |
| CH (1) | CH605753A5 (en:Method) |
| DD (1) | DD118426A5 (en:Method) |
| DE (1) | DE2406200A1 (en:Method) |
| DK (1) | DK44375A (en:Method) |
| ES (1) | ES434547A1 (en:Method) |
| FI (1) | FI750325A7 (en:Method) |
| FR (1) | FR2260346B1 (en:Method) |
| GB (1) | GB1444879A (en:Method) |
| HU (1) | HU168593B (en:Method) |
| IE (1) | IE40588B1 (en:Method) |
| IL (1) | IL46578A (en:Method) |
| LU (1) | LU71812A1 (en:Method) |
| NL (1) | NL7501499A (en:Method) |
| PL (1) | PL92432B1 (en:Method) |
| SE (1) | SE402588B (en:Method) |
| ZA (1) | ZA75789B (en:Method) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5232216A (en) * | 1975-09-05 | 1977-03-11 | Matsushita Electric Ind Co Ltd | Ghost eliminating equipment |
| DE2706977A1 (de) * | 1977-02-18 | 1978-08-24 | Hoechst Ag | Benzoesaeuren und deren derivate sowie verfahren zu ihrer herstellung |
| US5725789A (en) * | 1995-03-31 | 1998-03-10 | Minnesota Mining And Manufacturing Company | Aqueous oil and water repellent compositions |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3862161A (en) * | 1970-01-24 | 1975-01-21 | Bayer Ag | 4-pyridyl substituted 1,4-dihydropyridines |
| US3887558A (en) * | 1972-03-06 | 1975-06-03 | Bayer Ag | Process for producing 2,6-diamino -1,4- dihydro-3,5-pyridine-dicarboxylates and derivatives thereof |
-
1974
- 1974-02-09 DE DE19742406200 patent/DE2406200A1/de not_active Withdrawn
-
1975
- 1975-01-30 US US05/545,299 patent/US4001259A/en not_active Expired - Lifetime
- 1975-02-03 CA CA219,243A patent/CA1049525A/en not_active Expired
- 1975-02-06 FI FI750325A patent/FI750325A7/fi not_active Application Discontinuation
- 1975-02-06 IL IL46578A patent/IL46578A/en unknown
- 1975-02-06 BE BE153109A patent/BE825246A/xx unknown
- 1975-02-07 DK DK44375*#A patent/DK44375A/da unknown
- 1975-02-07 SE SE7501389A patent/SE402588B/xx unknown
- 1975-02-07 GB GB531375A patent/GB1444879A/en not_active Expired
- 1975-02-07 FR FR7503896A patent/FR2260346B1/fr not_active Expired
- 1975-02-07 NL NL7501499A patent/NL7501499A/xx not_active Application Discontinuation
- 1975-02-07 ZA ZA00750789A patent/ZA75789B/xx unknown
- 1975-02-07 CH CH150375A patent/CH605753A5/xx not_active IP Right Cessation
- 1975-02-07 IE IE246/75A patent/IE40588B1/xx unknown
- 1975-02-07 ES ES434547A patent/ES434547A1/es not_active Expired
- 1975-02-07 AT AT94875A patent/AT339904B/de not_active IP Right Cessation
- 1975-02-07 LU LU71812A patent/LU71812A1/xx unknown
- 1975-02-07 HU HUBA3202A patent/HU168593B/hu unknown
- 1975-02-07 JP JP50015501A patent/JPS50108269A/ja active Pending
- 1975-02-07 DD DD184074A patent/DD118426A5/xx unknown
- 1975-02-08 PL PL1975177899A patent/PL92432B1/pl unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CH605753A5 (en:Method) | 1978-10-13 |
| IL46578A (en) | 1977-11-30 |
| DK44375A (en:Method) | 1975-10-06 |
| IL46578A0 (en) | 1975-04-25 |
| SE7501389L (en:Method) | 1975-08-11 |
| US4001259A (en) | 1977-01-04 |
| BE825246A (fr) | 1975-08-06 |
| FI750325A7 (en:Method) | 1975-08-10 |
| PL92432B1 (en:Method) | 1977-04-30 |
| SE402588B (sv) | 1978-07-10 |
| ES434547A1 (es) | 1976-12-16 |
| USB545299I5 (en:Method) | 1976-02-24 |
| DE2406200A1 (de) | 1975-08-14 |
| CA1049525A (en) | 1979-02-27 |
| NL7501499A (nl) | 1975-08-12 |
| JPS50108269A (en:Method) | 1975-08-26 |
| ZA75789B (en) | 1976-03-31 |
| IE40588L (en) | 1975-08-09 |
| HU168593B (en:Method) | 1976-06-28 |
| AU7786575A (en) | 1976-08-05 |
| FR2260346B1 (en:Method) | 1980-01-11 |
| AT339904B (de) | 1977-11-10 |
| ATA94875A (de) | 1977-03-15 |
| DD118426A5 (en:Method) | 1976-03-05 |
| FR2260346A1 (en:Method) | 1975-09-05 |
| GB1444879A (en) | 1976-08-04 |
| LU71812A1 (en:Method) | 1975-12-09 |
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