IE40003B1 - New imidazoles and processes for their production - Google Patents
New imidazoles and processes for their productionInfo
- Publication number
- IE40003B1 IE40003B1 IE1746/74A IE174674A IE40003B1 IE 40003 B1 IE40003 B1 IE 40003B1 IE 1746/74 A IE1746/74 A IE 1746/74A IE 174674 A IE174674 A IE 174674A IE 40003 B1 IE40003 B1 IE 40003B1
- Authority
- IE
- Ireland
- Prior art keywords
- lower alkyl
- alkyl
- formula
- sulphonyl
- cpd
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/91—Nitro radicals
- C07D233/92—Nitro radicals attached in position 4 or 5
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Derivs. of formula (I): (where one of R1 and R2 is H or lower alkyl and the other is NO2; R3 is lower alkyl, hydroxyalkyl, alkoxyalkyl, alkyl-sulphonyl-alkyl or aminoalkyl; R4 is O or S; X is CO and R5 is lower alkoxy, NH2 or mono- or di(lower alkyl)-amino or X is CS, SO or SO2 and R5 is lower alkyl, aryl, NH2 or mono- or di-(lower alkyl)-amino; and "alk" is lower alkylene with 2-4 C-atoms in the alkylene chain) (e. g. 1-(methyl-thiocarbamoyl)-2-oxo-3-(1-methyl-5-nitro-2-imidazolyl)-- tetrahydroimidazole) and their salts and N-oxides are new cpds. They may be prepd. e.g. by reacting a cpd. of formula (II) (where Z is a reactive esterified or etherified hydroxy gp., a free or etherified mercapto group, an ammonium gp. or a sulphonyl gp.) with a cpd. of formula (III). (I) are antimicrobial and anthelmintic agents active against bacteria (esp. gram-negative bacteria), protozoa and worms such as trichomonads, schistosomes, coccidia and, especially, amoebae. (I) may thus be used for therapeutic purposes, as animal feed additives, and for protecting organic materials against microbial degradation.
[FR2244498A1]
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH1366773A CH592653A5 (en) | 1973-09-24 | 1973-09-24 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE40003L IE40003L (en) | 1975-03-24 |
| IE40003B1 true IE40003B1 (en) | 1979-02-14 |
Family
ID=4394325
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE1746/74A IE40003B1 (en) | 1973-09-24 | 1974-08-22 | New imidazoles and processes for their production |
Country Status (26)
| Country | Link |
|---|---|
| JP (1) | JPS5910347B2 (en) |
| AR (2) | AR212578A1 (en) |
| AT (1) | AT337692B (en) |
| BE (1) | BE820206A (en) |
| BG (2) | BG22813A3 (en) |
| CH (1) | CH592653A5 (en) |
| CS (1) | CS195689B2 (en) |
| DD (1) | DD114814A5 (en) |
| DE (1) | DE2444070A1 (en) |
| DK (1) | DK447474A (en) |
| DO (1) | DOP1981002973A (en) |
| ES (1) | ES430352A1 (en) |
| FI (1) | FI62293C (en) |
| FR (1) | FR2244498A1 (en) |
| HU (1) | HU171562B (en) |
| IE (1) | IE40003B1 (en) |
| IL (1) | IL45536A (en) |
| NL (1) | NL7412482A (en) |
| NO (1) | NO141895C (en) |
| OA (1) | OA04828A (en) |
| PH (1) | PH13743A (en) |
| PL (3) | PL95691B1 (en) |
| RO (1) | RO70190A (en) |
| SE (1) | SE416300B (en) |
| SU (3) | SU542473A3 (en) |
| YU (3) | YU37337B (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5956254U (en) * | 1982-10-05 | 1984-04-12 | 住友金属鉱山株式会社 | retaining wall block |
| JPH0423998Y2 (en) * | 1985-02-01 | 1992-06-04 | ||
| DE4426757A1 (en) * | 1994-07-28 | 1996-02-01 | Bayer Ag | 2-imidazolidinone derivatives |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2944061A (en) * | 1957-09-20 | 1960-07-05 | Acyl derivatives and process | |
| IL39283A (en) * | 1971-05-03 | 1976-01-30 | Ciba Geigy Ag | Substituted 2-oxo or thioxo-3-(5-nitro-imidazol-2-yl)-tetrahydroimidazoles and their manufacture |
| BE795068A (en) * | 1972-02-08 | 1973-08-07 | Ciba Geigy | NEW 4- OR 5-NITRO-INMIDAZOLES AND METHODS FOR THEIR PREPARATION |
-
1973
- 1973-09-24 CH CH1366773A patent/CH592653A5/xx not_active IP Right Cessation
-
1974
- 1974-08-21 DK DK447474A patent/DK447474A/da not_active Application Discontinuation
- 1974-08-22 IE IE1746/74A patent/IE40003B1/en unknown
- 1974-08-26 IL IL45536A patent/IL45536A/en unknown
- 1974-09-06 SE SE7411296A patent/SE416300B/en not_active IP Right Cessation
- 1974-09-12 FI FI2669/74A patent/FI62293C/en active
- 1974-09-14 DE DE2444070A patent/DE2444070A1/en not_active Ceased
- 1974-09-18 FR FR7431471A patent/FR2244498A1/en active Granted
- 1974-09-20 NO NO743395A patent/NO141895C/en unknown
- 1974-09-20 NL NL7412482A patent/NL7412482A/en not_active Application Discontinuation
- 1974-09-21 OA OA55302A patent/OA04828A/en unknown
- 1974-09-23 AR AR255685A patent/AR212578A1/en active
- 1974-09-23 PL PL1974185103A patent/PL95691B1/en unknown
- 1974-09-23 RO RO7487513A patent/RO70190A/en unknown
- 1974-09-23 BE BE148776A patent/BE820206A/en not_active IP Right Cessation
- 1974-09-23 PH PH16324A patent/PH13743A/en unknown
- 1974-09-23 BG BG029300A patent/BG22813A3/en unknown
- 1974-09-23 PL PL1974185100A patent/PL95689B1/en unknown
- 1974-09-23 DD DD181273A patent/DD114814A5/xx unknown
- 1974-09-23 SU SU2063056A patent/SU542473A3/en active
- 1974-09-23 BG BG027754A patent/BG22823A3/en unknown
- 1974-09-23 PL PL1974174285A patent/PL96510B1/en unknown
- 1974-09-23 AT AT762174A patent/AT337692B/en not_active IP Right Cessation
- 1974-09-23 YU YU2559/74A patent/YU37337B/en unknown
- 1974-09-24 CS CS746554A patent/CS195689B2/en unknown
- 1974-09-24 HU HU74CI00001509A patent/HU171562B/en unknown
- 1974-09-24 ES ES430352A patent/ES430352A1/en not_active Expired
- 1974-09-24 JP JP49110385A patent/JPS5910347B2/en not_active Expired
-
1975
- 1975-01-01 AR AR258970A patent/AR207980A1/en active
- 1975-07-02 SU SU7502149414A patent/SU571191A3/en active
- 1975-07-02 SU SU7502149413A patent/SU564812A3/en active
-
1980
- 1980-11-24 YU YU2983/80A patent/YU37339B/en unknown
- 1980-11-24 YU YU2982/80A patent/YU37338B/en unknown
-
1981
- 1981-02-09 DO DO1981002973A patent/DOP1981002973A/en unknown
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