IE36907B1 - Stereoisomers of 1-(1'-(o-chlorobenzyl)-2'-pyrryl)-2-disec.butylamino-ethanol - Google Patents
Stereoisomers of 1-(1'-(o-chlorobenzyl)-2'-pyrryl)-2-disec.butylamino-ethanolInfo
- Publication number
- IE36907B1 IE36907B1 IE1460/72A IE146072A IE36907B1 IE 36907 B1 IE36907 B1 IE 36907B1 IE 1460/72 A IE1460/72 A IE 1460/72A IE 146072 A IE146072 A IE 146072A IE 36907 B1 IE36907 B1 IE 36907B1
- Authority
- IE
- Ireland
- Prior art keywords
- disec
- pyrryl
- chlorobenzyl
- butylamino
- optically active
- Prior art date
Links
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N EtOH Substances CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 title abstract 4
- OKKJLVBELUTLKV-UHFFFAOYSA-N Methanol Chemical compound OC OKKJLVBELUTLKV-UHFFFAOYSA-N 0.000 abstract 3
- -1 butylamino ethanol Chemical compound 0.000 abstract 2
- 238000002360 preparation method Methods 0.000 abstract 2
- BHRZNVHARXXAHW-UHFFFAOYSA-N sec-butylamine Chemical compound CCC(C)N BHRZNVHARXXAHW-UHFFFAOYSA-N 0.000 abstract 2
- FJKROLUGYXJWQN-UHFFFAOYSA-M 4-hydroxybenzoate Chemical compound OC1=CC=C(C([O-])=O)C=C1 FJKROLUGYXJWQN-UHFFFAOYSA-M 0.000 abstract 1
- FJKROLUGYXJWQN-UHFFFAOYSA-N 4-hydroxybenzoic acid Chemical class OC(=O)C1=CC=C(O)C=C1 FJKROLUGYXJWQN-UHFFFAOYSA-N 0.000 abstract 1
- HQABUPZFAYXKJW-UHFFFAOYSA-N N-butylamine Natural products CCCCN HQABUPZFAYXKJW-UHFFFAOYSA-N 0.000 abstract 1
- 230000000202 analgesic effect Effects 0.000 abstract 1
- 125000006309 butyl amino group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000001640 fractional crystallisation Methods 0.000 abstract 1
- 150000004820 halides Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000003287 optical effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/335—Radicals substituted by nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/337—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT3058871 | 1971-10-30 | ||
| IT3058671 | 1971-10-30 | ||
| IT3058771 | 1971-10-30 | ||
| IT3058571 | 1971-10-30 | ||
| IT2656472A IT1044847B (it) | 1972-07-04 | 1972-07-04 | Benzil pirril aminoetanolo dotato di attivita antagonista nei con fronti della capacita ad indurre dipendenza fisica di composti dotati di attivita analgesica |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE36907L IE36907L (en) | 1973-04-30 |
| IE36907B1 true IE36907B1 (en) | 1977-03-16 |
Family
ID=27517845
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE1460/72A IE36907B1 (en) | 1971-10-30 | 1972-10-30 | Stereoisomers of 1-(1'-(o-chlorobenzyl)-2'-pyrryl)-2-disec.butylamino-ethanol |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US3857857A (enExample) |
| JP (1) | JPS5418247B2 (enExample) |
| AR (1) | AR194281A1 (enExample) |
| AU (1) | AU475877B2 (enExample) |
| BE (1) | BE790747A (enExample) |
| CA (1) | CA974245A (enExample) |
| CH (1) | CH583194A5 (enExample) |
| CS (1) | CS174859B2 (enExample) |
| DE (1) | DE2253150C3 (enExample) |
| DK (1) | DK138642B (enExample) |
| FI (1) | FI54105C (enExample) |
| FR (1) | FR2158056B1 (enExample) |
| GB (1) | GB1405148A (enExample) |
| IE (1) | IE36907B1 (enExample) |
| IL (1) | IL40665A (enExample) |
| NL (1) | NL178073C (enExample) |
| NO (1) | NO137784C (enExample) |
| SE (1) | SE387940B (enExample) |
| SU (1) | SU533334A3 (enExample) |
| YU (1) | YU267272A (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE848465A (fr) * | 1976-11-18 | 1977-03-16 | Stereo-isomeres de 1-(1'-benzyl-2' pyrryl)-2-disec.butylaminoethanols a activite analgesique et preparations pharmaceutiques qui les contiennent | |
| EP0342613B1 (en) * | 1988-05-20 | 1992-11-11 | ZAMBON GROUP S.p.A. | Compounds with central analgesic activity, process for their preparation and pharmaceutical compositions containing them |
| AU2009239778B2 (en) * | 2008-04-24 | 2014-03-13 | F2G Ltd | Pyrrole antifungal agents |
| MX2017006447A (es) | 2014-11-21 | 2018-01-30 | F2G Ltd | Agentes antifungicos. |
| GB201609222D0 (en) | 2016-05-25 | 2016-07-06 | F2G Ltd | Pharmaceutical formulation |
| US11819503B2 (en) | 2019-04-23 | 2023-11-21 | F2G Ltd | Method of treating coccidioides infection |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1544722A (fr) * | 1966-05-17 | 1968-11-08 | Whitefin Holding Sa | Dérivés du pyrrole et leur procédé de fabrication |
| GB1154745A (en) * | 1966-05-17 | 1969-06-11 | Whitefin Holding Sa | Haloketones |
-
0
- BE BE790747D patent/BE790747A/xx not_active IP Right Cessation
-
1972
- 1972-10-23 GB GB4878172A patent/GB1405148A/en not_active Expired
- 1972-10-24 US US00299726A patent/US3857857A/en not_active Expired - Lifetime
- 1972-10-25 IL IL40665A patent/IL40665A/xx unknown
- 1972-10-27 AR AR244847A patent/AR194281A1/es active
- 1972-10-27 NL NLAANVRAGE7214580,A patent/NL178073C/xx not_active IP Right Cessation
- 1972-10-27 YU YU02672/72A patent/YU267272A/xx unknown
- 1972-10-27 CA CA155,097A patent/CA974245A/en not_active Expired
- 1972-10-27 NO NO3880/72A patent/NO137784C/no unknown
- 1972-10-27 SE SE7213899A patent/SE387940B/xx unknown
- 1972-10-27 DK DK533472AA patent/DK138642B/da not_active IP Right Cessation
- 1972-10-30 FI FI3006/72A patent/FI54105C/fi active
- 1972-10-30 CH CH1582572A patent/CH583194A5/xx not_active IP Right Cessation
- 1972-10-30 FR FR7238462A patent/FR2158056B1/fr not_active Expired
- 1972-10-30 CS CS7290A patent/CS174859B2/cs unknown
- 1972-10-30 AU AU48321/72A patent/AU475877B2/en not_active Expired
- 1972-10-30 IE IE1460/72A patent/IE36907B1/xx unknown
- 1972-10-30 SU SU1848312A patent/SU533334A3/ru active
- 1972-10-30 DE DE2253150A patent/DE2253150C3/de not_active Expired
- 1972-10-30 JP JP10808572A patent/JPS5418247B2/ja not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| BE790747A (fr) | 1973-02-15 |
| NL7214580A (enExample) | 1973-05-02 |
| CA974245A (en) | 1975-09-09 |
| JPS5418247B2 (enExample) | 1979-07-06 |
| NO137784B (no) | 1978-01-16 |
| FI54105C (fi) | 1978-10-10 |
| CH583194A5 (enExample) | 1976-12-31 |
| JPS4852764A (enExample) | 1973-07-24 |
| US3857857A (en) | 1974-12-31 |
| FR2158056B1 (enExample) | 1976-04-23 |
| SE387940B (sv) | 1976-09-20 |
| IE36907L (en) | 1973-04-30 |
| FR2158056A1 (enExample) | 1973-06-08 |
| DE2253150B2 (de) | 1981-03-19 |
| FI54105B (fi) | 1978-06-30 |
| NL178073B (nl) | 1985-08-16 |
| AU475877B2 (en) | 1976-09-09 |
| AU4832172A (en) | 1974-05-02 |
| NO137784C (no) | 1978-04-26 |
| DK138642C (enExample) | 1979-03-12 |
| AR194281A1 (es) | 1973-06-29 |
| YU267272A (en) | 1982-02-28 |
| SU533334A3 (ru) | 1976-10-25 |
| DE2253150A1 (de) | 1973-05-10 |
| CS174859B2 (enExample) | 1977-04-29 |
| NL178073C (nl) | 1986-01-16 |
| IL40665A (en) | 1975-06-25 |
| GB1405148A (en) | 1975-09-03 |
| DE2253150C3 (de) | 1982-02-11 |
| DK138642B (da) | 1978-10-09 |
| IL40665A0 (en) | 1972-12-29 |
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