IE33494L - Cycloalkano-quinolones - Google Patents
Cycloalkano-quinolonesInfo
- Publication number
- IE33494L IE33494L IE100369A IE100369A IE33494L IE 33494 L IE33494 L IE 33494L IE 100369 A IE100369 A IE 100369A IE 100369 A IE100369 A IE 100369A IE 33494 L IE33494 L IE 33494L
- Authority
- IE
- Ireland
- Prior art keywords
- ethoxycarbonyl
- acrylate
- ethyl
- amino
- cycloalkano
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/04—Ortho- or peri-condensed ring systems
- C07D221/06—Ring systems of three rings
- C07D221/16—Ring systems of three rings containing carbocyclic rings other than six-membered
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/04—Ortho- or peri-condensed ring systems
- C07D221/06—Ring systems of three rings
- C07D221/08—Aza-anthracenes
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/04—Ortho- or peri-condensed ring systems
- C07D221/06—Ring systems of three rings
- C07D221/10—Aza-phenanthrenes
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
1,210,638. Cycloalkano-quinoline derivatives. BOEHRINGER MANNHEIM G.m.b.H. [21 July, 1969 [23 July, 1968; 14 March, 1969], No. 36601/69. Heading C2C. Novel cycloalkano-quinoline derivatives of the Formula I wherein one of the symbols R 1 and R 2 represents H halogen, NO 2 , NH 2 , OH, acylamino, acyloxy, alkoxy or aryloxy, while the other one, together with R 3 , forms an aliphatic bridge containing 2-6 carbon atoms, X is H, C 1-4 alkyl or C 2-4 alkenyl, and Y is OH, NH 2 or C 1-4 alkoxy and pharmacologically compatible salts thereof are prepared by cyclising a cycloalkano-benzene derivative of Formula II above, in which Y<SP>1</SP> is alkoxy or NH 2 , whereafter, if desired, the products obtained are saponified, esterified, transesterified or converted into amides, and/or the substituents R 1 or R 2 are introduced or chemically changed and/or, when X is H, the product is N-alkylated. Ethyl α - ethoxycarbonyl- # - (4 - indanylamino)-acrylate, ethyl α-ethoxycarbonyl-#-(5- indanylamino)acrylate, ethyl α - ethoxycarbonyl- # - (1,2,3,4 - tetrahydronaphthyl - 6 - amino) acrylate and ethyl α-ethoxycarbonyl-#- (1,2,3,4- tetrahydronaphthyl-5-amino) acrylate are obtained by reacting diethyl. ethoxymethylenemalonate with 4-aminoindane, 5-aminoindane, 6 - amino - 1,2,3,4 - tetrahydronaphthalene and 5 - -amino - 1,2,3,4 - tetrahydronaphthalene respectively. Pharmaceutical compositions, having antimicrobial activity, contain at least one of the above novel compounds in admixture with solid or liquid pharmaceutical diluents or carriers.
[GB1210638A]
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19681770951 DE1770951A1 (en) | 1968-07-23 | 1968-07-23 | Cyclopentanoquinolone derivatives and processes for their preparation |
DE19691912944 DE1912944A1 (en) | 1969-03-14 | 1969-03-14 | Cycloalkanoquinolone derivatives and processes for their preparation |
Publications (2)
Publication Number | Publication Date |
---|---|
IE33494L true IE33494L (en) | 1970-01-23 |
IE33494B1 IE33494B1 (en) | 1974-07-24 |
Family
ID=25755585
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IE100369A IE33494B1 (en) | 1968-07-23 | 1969-07-21 | Cycloalkano-quinolone derivatives |
Country Status (9)
Country | Link |
---|---|
AT (1) | AT294094B (en) |
CA (1) | CA944354A (en) |
CH (1) | CH529135A (en) |
FI (1) | FI49499C (en) |
FR (1) | FR2013519A1 (en) |
GB (1) | GB1210638A (en) |
IE (1) | IE33494B1 (en) |
NL (1) | NL6911270A (en) |
SE (1) | SE343059B (en) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2207856A1 (en) * | 1972-02-19 | 1973-08-23 | Boehringer Mannheim Gmbh | CYCLOALKANOCHINOLONE CARBONIC ACID ESTERS AND PROCESS FOR THEIR PRODUCTION |
US3966743A (en) | 1968-07-23 | 1976-06-29 | Boehringer Mannheim G.M.B.H. | Ortho fused cycloalkano-4-quinolone-3-carboxylic acid derivatives |
DE2011885C3 (en) * | 1970-03-13 | 1981-05-21 | Boehringer Mannheim Gmbh, 6800 Mannheim | 1,4-Dihydro-3-carboxy-cyclopentano (h) -quinolone- (4) -derivatives, process for the preparation thereof and their use |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3324135A (en) * | 1963-04-19 | 1967-06-06 | Sterling Drug Inc | 4-alkyl-1-benzo[f]quinolone-2-carboxylic acids |
-
1969
- 1969-07-10 CA CA056,733A patent/CA944354A/en not_active Expired
- 1969-07-21 GB GB3660169A patent/GB1210638A/en not_active Expired
- 1969-07-21 IE IE100369A patent/IE33494B1/en unknown
- 1969-07-21 CH CH1115569A patent/CH529135A/en not_active IP Right Cessation
- 1969-07-21 FI FI216069A patent/FI49499C/en active
- 1969-07-22 AT AT704869A patent/AT294094B/en not_active IP Right Cessation
- 1969-07-22 FR FR6924872A patent/FR2013519A1/fr not_active Withdrawn
- 1969-07-22 SE SE1030669A patent/SE343059B/xx unknown
- 1969-07-23 NL NL6911270A patent/NL6911270A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
GB1210638A (en) | 1970-10-28 |
FI49499B (en) | 1975-04-01 |
SE343059B (en) | 1972-02-28 |
IE33494B1 (en) | 1974-07-24 |
AT294094B (en) | 1971-11-10 |
FR2013519A1 (en) | 1970-04-03 |
FI49499C (en) | 1975-07-10 |
NL6911270A (en) | 1970-01-27 |
CH529135A (en) | 1972-10-15 |
CA944354A (en) | 1974-03-26 |
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