HUP0402401A2 - Rák kezelésére szolgáló eljárások egy FPT inhibitor és daganatellenes szerek felhasználásával - Google Patents
Rák kezelésére szolgáló eljárások egy FPT inhibitor és daganatellenes szerek felhasználásával Download PDFInfo
- Publication number
- HUP0402401A2 HUP0402401A2 HU0402401A HUP0402401A HUP0402401A2 HU P0402401 A2 HUP0402401 A2 HU P0402401A2 HU 0402401 A HU0402401 A HU 0402401A HU P0402401 A HUP0402401 A HU P0402401A HU P0402401 A2 HUP0402401 A2 HU P0402401A2
- Authority
- HU
- Hungary
- Prior art keywords
- administered
- amount
- fpt inhibitor
- twice daily
- per cycle
- Prior art date
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
- A61K33/24—Heavy metals; Compounds thereof
- A61K33/243—Platinum; Compounds thereof
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
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- Chemical Kinetics & Catalysis (AREA)
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- Inorganic Chemistry (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
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|---|---|---|---|
| US33441101P | 2001-11-30 | 2001-11-30 | |
| PCT/US2002/037954 WO2003047697A2 (en) | 2001-11-30 | 2002-11-25 | Use of an farsenyl protein tranferase inhibitor in combination with other antineoplastic agents for the manufacture of a medicament against cancer |
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| HUP0402401A2 true HUP0402401A2 (hu) | 2005-03-29 |
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|---|---|
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| EP (1) | EP1448268A2 (enExample) |
| JP (1) | JP2005511663A (enExample) |
| CN (2) | CN1617755A (enExample) |
| AU (1) | AU2002352941A1 (enExample) |
| BR (1) | BR0214564A (enExample) |
| CA (1) | CA2468839A1 (enExample) |
| HU (1) | HUP0402401A2 (enExample) |
| MX (1) | MXPA04005207A (enExample) |
| NO (1) | NO20042730L (enExample) |
| NZ (1) | NZ532562A (enExample) |
| WO (1) | WO2003047697A2 (enExample) |
| ZA (1) | ZA200403737B (enExample) |
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| CA2439440A1 (en) * | 2002-09-05 | 2004-03-05 | Emory University | Treatment of tuberous sclerosis associated neoplasms |
| AU2004289256A1 (en) * | 2003-11-06 | 2005-05-26 | Schering Corporation | Combination of a farnesyl tranferase inhibitor with an antihormonal agent for the treatment of breast cancer |
| AU2005216898A1 (en) * | 2004-02-26 | 2005-09-09 | The Penn State Research Foundation | Combinatorial therapies for the treatment of neoplasias using the opioid growth factor receptor |
| US20060205810A1 (en) * | 2004-11-24 | 2006-09-14 | Schering Corporation | Platinum therapeutic combinations |
| WO2007042465A2 (en) * | 2005-10-07 | 2007-04-19 | Novartis Ag | Combinati0n of nilotinib with farnesyl transferase inhibitors |
| JP2010507662A (ja) * | 2006-10-25 | 2010-03-11 | シェーリング コーポレイション | 癌の処置のための不連続方法 |
| EP2088862A4 (en) * | 2006-11-28 | 2009-12-02 | Smithkline Beecham Cork Ltd | METHOD OF TREATING CANCER |
| EP4615842A1 (en) | 2022-11-09 | 2025-09-17 | Merck Patent GmbH | Toll-like receptor 7 agonists as immune-stimulators to elicit the innate antitumor immunity |
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| US5874442A (en) * | 1995-12-22 | 1999-02-23 | Schering-Plough Corporation | Tricyclic amides useful for inhibition of G-protein function and for treatment of proliferative disease |
| CZ298511B6 (cs) * | 1997-12-22 | 2007-10-24 | Schering Corporation | Použití benzocykloheptapyridinových sloucenin proprípravu farmaceutického prípravku pro použití v kombinaci s antineoplastickým lécivem a/nebo radioterapií k lécení proliferacních onemocnení |
| US6096757A (en) * | 1998-12-21 | 2000-08-01 | Schering Corporation | Method for treating proliferative diseases |
| US6316462B1 (en) * | 1999-04-09 | 2001-11-13 | Schering Corporation | Methods of inducing cancer cell death and tumor regression |
| JP5491681B2 (ja) * | 2000-02-04 | 2014-05-14 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | 乳ガンの治療のためのファルネシルタンパク質トランスフェラーゼ阻害剤 |
| EP1267848B1 (en) * | 2000-02-24 | 2007-10-17 | Janssen Pharmaceutica N.V. | Dosing regimen comprising a farnesyl protein transferase inhibitor for the treatment of cancer |
| WO2001064252A2 (en) * | 2000-02-29 | 2001-09-07 | Janssen Pharmaceutica N.V. | Farnesyl protein transferase inhibitor combinations with further anti-cancer agents |
| WO2001064199A2 (en) * | 2000-02-29 | 2001-09-07 | Janssen Pharmaceutica N.V. | Farnesyl protein transferase inhibitor combinations with taxane compounds |
| AR033680A1 (es) * | 2000-08-30 | 2004-01-07 | Schering Corp | Compuestos triciclicos utiles como inhibidores de la farnesil proteino transferasa y su uso para la manufactura de medicamentos como agentes antitumorales |
| BR0114430A (pt) * | 2000-10-05 | 2004-01-06 | George Q Daley | Processos para a indução da morte de células cancerìgenas e para a regressão de tumor |
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2002
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- 2002-11-25 BR BR0214564-2A patent/BR0214564A/pt not_active IP Right Cessation
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- 2002-11-25 NZ NZ532562A patent/NZ532562A/en unknown
- 2002-11-25 CN CNA2007101860344A patent/CN101181269A/zh active Pending
- 2002-11-25 JP JP2003548949A patent/JP2005511663A/ja not_active Withdrawn
- 2002-11-25 AU AU2002352941A patent/AU2002352941A1/en not_active Abandoned
-
2004
- 2004-05-14 ZA ZA200403737A patent/ZA200403737B/en unknown
- 2004-06-29 NO NO20042730A patent/NO20042730L/no not_active Application Discontinuation
-
2006
- 2006-04-03 US US11/396,892 patent/US20060183765A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN101181269A (zh) | 2008-05-21 |
| NO20042730L (no) | 2004-06-29 |
| WO2003047697A3 (en) | 2003-10-30 |
| ZA200403737B (en) | 2005-05-23 |
| BR0214564A (pt) | 2004-11-09 |
| MXPA04005207A (es) | 2004-08-19 |
| US20030185831A1 (en) | 2003-10-02 |
| CN1617755A (zh) | 2005-05-18 |
| EP1448268A2 (en) | 2004-08-25 |
| JP2005511663A (ja) | 2005-04-28 |
| NZ532562A (en) | 2007-02-23 |
| CA2468839A1 (en) | 2003-06-12 |
| AU2002352941A1 (en) | 2003-06-17 |
| WO2003047697A2 (en) | 2003-06-12 |
| US20060183765A1 (en) | 2006-08-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD9A | Lapse of provisional protection due to non-payment of fees |