HUP0401273A3 - Naphtothiazine positive allosteric ampa receptor modulators, their use and pharmaceutical compositions containing them - Google Patents
Naphtothiazine positive allosteric ampa receptor modulators, their use and pharmaceutical compositions containing themInfo
- Publication number
- HUP0401273A3 HUP0401273A3 HU0401273A HUP0401273A HUP0401273A3 HU P0401273 A3 HUP0401273 A3 HU P0401273A3 HU 0401273 A HU0401273 A HU 0401273A HU P0401273 A HUP0401273 A HU P0401273A HU P0401273 A3 HUP0401273 A3 HU P0401273A3
- Authority
- HU
- Hungary
- Prior art keywords
- naphtothiazine
- pharmaceutical compositions
- compositions containing
- receptor modulators
- positive allosteric
- Prior art date
Links
- 102000003678 AMPA Receptors Human genes 0.000 title 1
- 108090000078 AMPA Receptors Proteins 0.000 title 1
- 230000003281 allosteric effect Effects 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10123952A DE10123952A1 (de) | 2001-05-17 | 2001-05-17 | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
| PCT/EP2002/005338 WO2002100411A1 (en) | 2001-05-17 | 2002-05-15 | Naphtothiazine positive allosteric ampa receptor modulators (paarm) |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| HUP0401273A2 HUP0401273A2 (hu) | 2004-10-28 |
| HUP0401273A3 true HUP0401273A3 (en) | 2006-11-28 |
Family
ID=7685080
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU0401273A HUP0401273A3 (en) | 2001-05-17 | 2002-05-15 | Naphtothiazine positive allosteric ampa receptor modulators, their use and pharmaceutical compositions containing them |
Country Status (26)
| Country | Link |
|---|---|
| EP (1) | EP1404340A1 (xx) |
| JP (1) | JP2004529980A (xx) |
| KR (1) | KR20040007572A (xx) |
| CN (1) | CN1533278A (xx) |
| AR (1) | AR036332A1 (xx) |
| BG (1) | BG108324A (xx) |
| BR (1) | BR0209796A (xx) |
| CA (1) | CA2449189A1 (xx) |
| CO (1) | CO5550460A2 (xx) |
| CZ (1) | CZ20033112A3 (xx) |
| DE (1) | DE10123952A1 (xx) |
| EA (1) | EA006608B1 (xx) |
| EC (1) | ECSP034852A (xx) |
| EE (1) | EE200300566A (xx) |
| HR (1) | HRP20030933A2 (xx) |
| HU (1) | HUP0401273A3 (xx) |
| IL (1) | IL158642A0 (xx) |
| MX (1) | MXPA03010373A (xx) |
| NO (1) | NO20035088D0 (xx) |
| NZ (1) | NZ530154A (xx) |
| PL (1) | PL364053A1 (xx) |
| SK (1) | SK14222003A3 (xx) |
| UY (1) | UY27290A1 (xx) |
| WO (1) | WO2002100411A1 (xx) |
| YU (1) | YU90403A (xx) |
| ZA (1) | ZA200308466B (xx) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2660431C (en) * | 2006-08-31 | 2015-03-17 | The Governors Of The University Of Alberta | Method of inhibition of respiratory depression using positive allosteric ampa receptor modulators |
| CN111518058B (zh) * | 2020-05-29 | 2021-03-09 | 四川大学华西医院 | 一种噁噻嗪类化合物及其用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1998012185A1 (en) * | 1996-09-17 | 1998-03-26 | The Regents Of The University Of California | Benzothiadiazide derivatives and their use as allosteric up-modulators of the ampa receptor |
| CA2335510A1 (en) * | 1998-06-25 | 1999-12-29 | Merck & Co., Inc. | Naphtho[1,8-de]thiasin-2-yl methyl carbapenem antibacterials |
| DE10004572A1 (de) * | 2000-02-02 | 2001-08-09 | Boehringer Ingelheim Pharma | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
-
2001
- 2001-05-17 DE DE10123952A patent/DE10123952A1/de not_active Withdrawn
-
2002
- 2002-05-15 CA CA002449189A patent/CA2449189A1/en not_active Abandoned
- 2002-05-15 YU YU90403A patent/YU90403A/sh unknown
- 2002-05-15 PL PL02364053A patent/PL364053A1/xx not_active Application Discontinuation
- 2002-05-15 WO PCT/EP2002/005338 patent/WO2002100411A1/en not_active Application Discontinuation
- 2002-05-15 CN CNA028100832A patent/CN1533278A/zh active Pending
- 2002-05-15 SK SK1422-2003A patent/SK14222003A3/sk unknown
- 2002-05-15 EA EA200301167A patent/EA006608B1/ru not_active IP Right Cessation
- 2002-05-15 EE EEP200300566A patent/EE200300566A/xx unknown
- 2002-05-15 UY UY27290A patent/UY27290A1/es not_active Application Discontinuation
- 2002-05-15 JP JP2003503232A patent/JP2004529980A/ja not_active Abandoned
- 2002-05-15 BR BR0209796-6A patent/BR0209796A/pt not_active Expired - Fee Related
- 2002-05-15 CZ CZ20033112A patent/CZ20033112A3/cs unknown
- 2002-05-15 EP EP02750931A patent/EP1404340A1/en not_active Withdrawn
- 2002-05-15 HU HU0401273A patent/HUP0401273A3/hu unknown
- 2002-05-15 IL IL15864202A patent/IL158642A0/xx unknown
- 2002-05-15 MX MXPA03010373A patent/MXPA03010373A/es unknown
- 2002-05-15 NZ NZ530154A patent/NZ530154A/en unknown
- 2002-05-15 KR KR10-2003-7014965A patent/KR20040007572A/ko not_active Application Discontinuation
- 2002-05-17 AR ARP020101827A patent/AR036332A1/es not_active Suspension/Interruption
-
2003
- 2003-10-30 ZA ZA200308466A patent/ZA200308466B/en unknown
- 2003-11-07 BG BG108324A patent/BG108324A/bg active Pending
- 2003-11-14 HR HR20030933A patent/HRP20030933A2/xx not_active Application Discontinuation
- 2003-11-14 NO NO20035088A patent/NO20035088D0/no not_active Application Discontinuation
- 2003-11-17 EC EC2003004852A patent/ECSP034852A/es unknown
- 2003-12-01 CO CO03105591A patent/CO5550460A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| YU90403A (sh) | 2006-05-25 |
| NO20035088L (no) | 2003-11-14 |
| IL158642A0 (en) | 2004-05-12 |
| DE10123952A1 (de) | 2002-11-21 |
| WO2002100411A1 (en) | 2002-12-19 |
| BR0209796A (pt) | 2004-06-01 |
| SK14222003A3 (sk) | 2004-05-04 |
| CA2449189A1 (en) | 2002-12-19 |
| ZA200308466B (en) | 2004-05-24 |
| EE200300566A (et) | 2004-02-16 |
| NZ530154A (en) | 2005-09-30 |
| CZ20033112A3 (en) | 2004-03-17 |
| EP1404340A1 (en) | 2004-04-07 |
| ECSP034852A (es) | 2003-12-24 |
| CO5550460A2 (es) | 2005-08-31 |
| KR20040007572A (ko) | 2004-01-24 |
| BG108324A (bg) | 2004-12-30 |
| HUP0401273A2 (hu) | 2004-10-28 |
| EA200301167A1 (ru) | 2004-06-24 |
| MXPA03010373A (es) | 2004-03-16 |
| NO20035088D0 (no) | 2003-11-14 |
| UY27290A1 (es) | 2002-12-31 |
| AR036332A1 (es) | 2004-09-01 |
| JP2004529980A (ja) | 2004-09-30 |
| CN1533278A (zh) | 2004-09-29 |
| HRP20030933A2 (en) | 2004-04-30 |
| EA006608B1 (ru) | 2006-02-24 |
| PL364053A1 (en) | 2004-12-13 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD9A | Lapse of provisional protection due to non-payment of fees |