HUP0100163A2 - Szerves szintézisekben alkalmazható védő- és kötőcsoportok - Google Patents
Szerves szintézisekben alkalmazható védő- és kötőcsoportokInfo
- Publication number
- HUP0100163A2 HUP0100163A2 HU0100163A HUP0100163A HUP0100163A2 HU P0100163 A2 HUP0100163 A2 HU P0100163A2 HU 0100163 A HU0100163 A HU 0100163A HU P0100163 A HUP0100163 A HU P0100163A HU P0100163 A2 HUP0100163 A2 HU P0100163A2
- Authority
- HU
- Hungary
- Prior art keywords
- substituted
- unsaturated
- saturated
- imino
- group
- Prior art date
Links
- 238000003786 synthesis reaction Methods 0.000 title abstract 2
- 125000005647 linker group Chemical group 0.000 title 1
- 125000006239 protecting group Chemical group 0.000 title 1
- 125000001841 imino group Chemical group [H]N=* 0.000 abstract 4
- 229920006395 saturated elastomer Polymers 0.000 abstract 4
- -1 cycloheteroaryl Chemical group 0.000 abstract 2
- 229930186217 Glycolipid Natural products 0.000 abstract 1
- 102000002068 Glycopeptides Human genes 0.000 abstract 1
- 108010015899 Glycopeptides Proteins 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 125000005035 acylthio group Chemical group 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000003282 alkyl amino group Chemical group 0.000 abstract 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- 125000001769 aryl amino group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 125000004391 aryl sulfonyl group Chemical group 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 150000001732 carboxylic acid derivatives Chemical class 0.000 abstract 1
- 150000001767 cationic compounds Chemical class 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004122 cyclic group Chemical group 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000004663 dialkyl amino group Chemical group 0.000 abstract 1
- 125000004986 diarylamino group Chemical group 0.000 abstract 1
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 1
- 125000002795 guanidino group Chemical group C(N)(=N)N* 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000004404 heteroalkyl group Chemical group 0.000 abstract 1
- 125000001072 heteroaryl group Chemical group 0.000 abstract 1
- 125000000592 heterocycloalkyl group Chemical group 0.000 abstract 1
- 125000000717 hydrazino group Chemical group [H]N([*])N([H])[H] 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 229910001411 inorganic cation Inorganic materials 0.000 abstract 1
- 229910021645 metal ion Inorganic materials 0.000 abstract 1
- 125000000896 monocarboxylic acid group Chemical group 0.000 abstract 1
- 229920001542 oligosaccharide Polymers 0.000 abstract 1
- 150000002482 oligosaccharides Chemical class 0.000 abstract 1
- 150000002892 organic cations Chemical class 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 102000004196 processed proteins & peptides Human genes 0.000 abstract 1
- 108090000765 processed proteins & peptides Proteins 0.000 abstract 1
- 125000001453 quaternary ammonium group Chemical group 0.000 abstract 1
- 125000001439 semicarbazido group Chemical group [H]N([H])C(=O)N([H])N([H])* 0.000 abstract 1
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 1
- 125000005346 substituted cycloalkyl group Chemical group 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 239000011593 sulfur Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/12—Acyclic radicals, not substituted by cyclic structures attached to a nitrogen atom of the saccharide radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/60—Three or more oxygen or sulfur atoms
- C07D239/62—Barbituric acids
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Biotechnology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Crystallography & Structural Chemistry (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Treatments Of Macromolecular Shaped Articles (AREA)
Abstract
A találmány peptidek, oligoszacharidok, glikopeptidekés glikolipidek szintézisében védő- és kötőcsoportként alkalmazhatóvegyületekre vonatkozik, amelyek (I) általános képletében a gyűrű egyadott esetben szubsztituált cikloalkil-, ciklohetero-alkil-, telítettbiciklo[p,q,r]-, telített heterobiciklo-[p,q,r]-, telítetlenbiciklo[p,q,r]-, telítetlen heterobiciklo[p,q,r]-, telítetttriciklo[p,q,r,s]-, telítetlen tricikloalkil[p,q,r,s]-, telítettheterotriciklo[p,q,r,s]- vagy telítetlen heterotriciklo[p,q,r,s]-gyűrűrendszert jelent; ahol p, q, r és s jelentése azonos vagy eltérő,és egész számot jelent, amelynek értéke 0-5; X jelentése oxigén-,kénatom, iminocsoport vagy szubsztituált iminocsoport; R1 jelentésehidrogénatom; adott esetben szubsztituált alkil-, alkenil-, alkinil-,heteroalkil-, aril-, heteroaril-, cikloheteroaril-, cikloalkil-,heterocikloalkil-, alkanal- vagy tioalkanol-csoport; NH2, guanidino-,CN-, szubsztituált amino-, kvaterner ammónium-, O-, formil-, imino-vagy szubsztituált iminocsoport, COOH vagy karbonsav-származék; R2jelentése O-szubsztituált hidroxilamino-csoport, adott esetbenszubsztituált alkilamino-, dialkilamino-, arilamino-, diarilamino-,hidrazino-, hidrazido-, tiohidrazido-csoport; szemikarbazido-csoport,tioszemikarbazido-csoport, OH, O M, NH2, NHOH, SH, S-M+, halogénatom,O-alkil-, O-acil-, O-aril-, alkiltio-, S-aril-, aciltio-,alkilszulfonil- vagy arilszulfonil-csoport, amelyek bármelyikeszubsztituált vagy szubsztituálatlan; és M jelentése fémion, vagyszerves vagy szervetlen kation. Ó
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AUPO9375A AUPO937597A0 (en) | 1997-09-24 | 1997-09-24 | Protecting and linking groups for organic synthesis |
| US6198797P | 1997-10-14 | 1997-10-14 | |
| PCT/AU1998/000808 WO1999015510A1 (en) | 1997-09-24 | 1998-09-24 | Protecting and linking groups for organic synthesis |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HUP0100163A2 true HUP0100163A2 (hu) | 2001-05-28 |
Family
ID=25645622
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU0100163A HUP0100163A2 (hu) | 1997-09-24 | 1998-09-24 | Szerves szintézisekben alkalmazható védő- és kötőcsoportok |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP1017683A4 (hu) |
| JP (1) | JP2001517660A (hu) |
| CN (1) | CN1276788A (hu) |
| CA (1) | CA2304061A1 (hu) |
| HU (1) | HUP0100163A2 (hu) |
| WO (1) | WO1999015510A1 (hu) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AUPO190596A0 (en) | 1996-08-26 | 1996-09-19 | Alchemia Pty Ltd | Oligosaccharide synthesis |
| AUPO937597A0 (en) | 1997-09-24 | 1997-10-16 | Alchemia Pty Ltd | Protecting and linking groups for organic synthesis |
| AUPP823099A0 (en) | 1999-01-18 | 1999-02-11 | Alchemia Pty Ltd | Protecting groups for carbohydrate synthesis |
| EP1175427B1 (en) | 1999-03-05 | 2010-08-18 | Massachusetts Institute Of Technology | Linkers for synthesis of oligosaccharides on solid supports |
| WO2006056443A2 (en) * | 2004-11-24 | 2006-06-01 | Aplagen Gmbh | Method for solid-phase peptide synthesis and purification |
| US20120258891A1 (en) * | 2011-04-07 | 2012-10-11 | Nimblegen Systems Gmbh | Diarylsulfide backbone containing photolabile protecting groups |
| FR3035787B1 (fr) * | 2015-05-07 | 2018-08-24 | L'oreal | Procede de traitement des matieres keratiniques a partir de derives de c-glycosides amides, acides ou ester, et la composition cosmetique les contenant |
| CN108530368B (zh) * | 2018-05-18 | 2020-01-17 | 青岛市妇女儿童医院（青岛市妇幼保健院、青岛市残疾儿童医疗康复中心、青岛市新生儿疾病筛查中心） | 有机碱催化巴比妥酸与二烯二腈加成反应的方法 |
| CN111208284B (zh) * | 2018-11-22 | 2021-08-24 | 北京大学 | 糖代谢标记探针、包含其的试剂盒及其应用 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5959109A (en) * | 1996-05-15 | 1999-09-28 | Neurocrine Biosciences, Inc. | Compounds and methods for increasing endogenous levels of corticotropin-releasing factor |
| AU728149B2 (en) * | 1996-08-26 | 2001-01-04 | Alchemia Pty Ltd | Oligosaccharide synthesis |
| KR20000048925A (ko) * | 1996-10-04 | 2000-07-25 | 후쿠오카 나오히코 | 아미노메틸렌 유도체 및 이것을 함유한 자외선 흡수제 |
| AUPO536797A0 (en) * | 1997-02-28 | 1997-03-20 | Alchemia Pty Ltd | Protected aminosugars |
-
1998
- 1998-09-24 WO PCT/AU1998/000808 patent/WO1999015510A1/en not_active Application Discontinuation
- 1998-09-24 EP EP98946145A patent/EP1017683A4/en not_active Withdrawn
- 1998-09-24 CA CA002304061A patent/CA2304061A1/en not_active Abandoned
- 1998-09-24 HU HU0100163A patent/HUP0100163A2/hu unknown
- 1998-09-24 CN CN98809501A patent/CN1276788A/zh active Pending
- 1998-09-24 JP JP2000512818A patent/JP2001517660A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| CA2304061A1 (en) | 1999-04-01 |
| CN1276788A (zh) | 2000-12-13 |
| EP1017683A1 (en) | 2000-07-12 |
| EP1017683A4 (en) | 2002-03-06 |
| JP2001517660A (ja) | 2001-10-09 |
| WO1999015510A1 (en) | 1999-04-01 |
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