HUP0001957A2 - Gombaellenes hatású, piridingyűrűben karbonsavszármazékokkal helyettesített 2-(metoxi-imino)-2-(piridinil-oxi-metil)-fenil-acetamid-származékok, intermedierjeik, előállításuk és alkalmazásuk - Google Patents

Gombaellenes hatású, piridingyűrűben karbonsavszármazékokkal helyettesített 2-(metoxi-imino)-2-(piridinil-oxi-metil)-fenil-acetamid-származékok, intermedierjeik, előállításuk és alkalmazásuk

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Publication number
HUP0001957A2
HUP0001957A2 HU0001957A HUP0001957A HUP0001957A2 HU P0001957 A2 HUP0001957 A2 HU P0001957A2 HU 0001957 A HU0001957 A HU 0001957A HU P0001957 A HUP0001957 A HU P0001957A HU P0001957 A2 HUP0001957 A2 HU P0001957A2
Authority
HU
Hungary
Prior art keywords
alkyl
pyridinyloxymethyl
methoxyimino
fungicides
intermediates
Prior art date
Application number
HU0001957A
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English (en)
Inventor
Scott J. Bis
Emily J. Canada
David H. Cooper
Christopher S. Galka
Vidyadhar B. Hegde
Neil Kirby
David G. Ouimette
Mary Pieczko
David E. Podhorez
Rebecca Rezac
Brent J. Rieder
Gary L. Sampson
John K. Swayze
Original Assignee
Dow Agrosciences Llc
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Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of HUP0001957A2 publication Critical patent/HUP0001957A2/hu
Publication of HUP0001957A3 publication Critical patent/HUP0001957A3/hu

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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61Halogen atoms or nitro radicals
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
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    • C07C251/34Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/48Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups bound to a carbon atom of a six-membered aromatic ring
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    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/83Thioacids; Thioesters; Thioamides; Thioimides

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pyridine Compounds (AREA)

Abstract

A találmány az (1) általános képletű vegyületekre, a képletben m értéke 0 és 3 közötti egész szám; Y jelentése hidrogén- vagy halogénatom, alkil-, alkoxi- vagyalkiltiocsoport; X jelentése hidrogénatom, alkil-, alkoxi-, halogén-alkil-,halogénalkoxi-csoport, halogénatom, nitro-, karbo-alkoxi-, ciano-,alkiltio- vagy halogén-alkiltio-csoport; W vagy W' jelentése egymástól függetlenül oxigén- vagy kénatom; R jelentése hidrogénatom, alkil-, vagy cikloalkil-csoport; amelyekadott esetben halogén alkil-, halogén-alkoxi-, alkenil-, halogén-alkenil-, alkinil-, ciano-, alkoxi-csoporttal, halogénatommal, aril-,helyettesített aril- vagy heteroarilcsoporttal van helyettesítve; és L jelentése -O-, -CH2-, -SOn-, -CH2O-, -OCH2-, -CH2S-, -SCH2-, -CH=CH-, -CC- vagy (c) képletű csoport, ahol n értéke 0 és 2 közöttiegész szám. vonatkozik. A találmány kiterjed a (II) általános képletűintermedierre, valamint az (a) általános képletű vegyületek - aképletekben Y jelentése klór- vagy fluoratom és m értéke 0, 1, 2 vagy3 - előállítására is. Ó
HU0001957A 1997-02-03 1998-01-29 2-methoxyimino-2-(pyridinyloxymethyl)phenyl acetamides with carboxylic acid derivatives on the pyridine ring as fungicides, intermediates, preparation and use thereof HUP0001957A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3685897P 1997-02-03 1997-02-03
PCT/US1998/001666 WO1998033772A1 (en) 1997-02-03 1998-01-29 2-methoxyimino-2-(pyridinyloxymethyl)phenyl acetamides with carboxylic acid derivatives on the pyridine ring as fungicides

Publications (2)

Publication Number Publication Date
HUP0001957A2 true HUP0001957A2 (hu) 2000-10-28
HUP0001957A3 HUP0001957A3 (en) 2000-12-28

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ID=21891047

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Application Number Title Priority Date Filing Date
HU0001957A HUP0001957A3 (en) 1997-02-03 1998-01-29 2-methoxyimino-2-(pyridinyloxymethyl)phenyl acetamides with carboxylic acid derivatives on the pyridine ring as fungicides, intermediates, preparation and use thereof

Country Status (10)

Country Link
US (1) US5968875A (hu)
EP (1) EP0961771A1 (hu)
JP (1) JP2001511146A (hu)
KR (1) KR100514941B1 (hu)
CN (1) CN1126742C (hu)
AU (1) AU729160B2 (hu)
BR (1) BR9807145B1 (hu)
CA (1) CA2278851C (hu)
HU (1) HUP0001957A3 (hu)
WO (1) WO1998033772A1 (hu)

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WO2000015635A1 (en) * 1998-09-16 2000-03-23 Dow Agrosciences Llc 2-methoxyimino -2-(pyridinyloxymethyl) phenyl acetamides useful as fungicides
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AU6049199A (en) 1998-09-16 2000-04-03 Dow Agrosciences Llc 2-methoxyimino-2-(pyridinyloxymethyl)phenyl acetamides with (derivatised) hydroxyalkyl derivatives on the pyridine ring
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WO2012152741A1 (de) 2011-05-10 2012-11-15 Bayer Intellectual Property Gmbh Bicyclische (thio)carbonylamidine
EP2871180B1 (en) 2012-07-04 2018-03-21 Agro-Kanesho Co., Ltd. 2-aminonicotinic acid ester derivative and bactericide containing same as active ingredient
EA030128B1 (ru) 2012-09-26 2018-06-29 Арагон Фармасьютикалз, Инк. Способ лечения неметастатического кастрационно-резистентного рака простаты
JOP20200097A1 (ar) 2013-01-15 2017-06-16 Aragon Pharmaceuticals Inc معدل مستقبل أندروجين واستخداماته
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GB9602623D0 (en) * 1996-02-09 1996-04-10 Zeneca Ltd Fungicides

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AU6254398A (en) 1998-08-25
EP0961771A1 (en) 1999-12-08
KR20000070702A (ko) 2000-11-25
WO1998033772A1 (en) 1998-08-06
KR100514941B1 (ko) 2005-09-15
AU729160B2 (en) 2001-01-25
CN1126742C (zh) 2003-11-05
BR9807145A (pt) 2000-03-14
HUP0001957A3 (en) 2000-12-28
CA2278851C (en) 2009-04-07
CA2278851A1 (en) 1998-08-06
US5968875A (en) 1999-10-19
JP2001511146A (ja) 2001-08-07
BR9807145B1 (pt) 2010-06-29

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