HU186877B - Process for preparing new hormone antagonists releasing luteinizing hormone and acid addition salts thereof - Google Patents

Process for preparing new hormone antagonists releasing luteinizing hormone and acid addition salts thereof Download PDF

Info

Publication number
HU186877B
HU186877B HU823976A HU397682A HU186877B HU 186877 B HU186877 B HU 186877B HU 823976 A HU823976 A HU 823976A HU 397682 A HU397682 A HU 397682A HU 186877 B HU186877 B HU 186877B
Authority
HU
Hungary
Prior art keywords
formula
protected
phe
resin
peptide
Prior art date
Application number
HU823976A
Other languages
English (en)
Hungarian (hu)
Inventor
David H Coy
Andrew V Schally
Original Assignee
Coy David Howard
Schally Andrew Victor
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Coy David Howard, Schally Andrew Victor filed Critical Coy David Howard
Publication of HU186877B publication Critical patent/HU186877B/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
HU823976A 1981-12-10 1982-12-09 Process for preparing new hormone antagonists releasing luteinizing hormone and acid addition salts thereof HU186877B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32952681A 1981-12-10 1981-12-10
US36870282A 1982-04-15 1982-04-15

Publications (1)

Publication Number Publication Date
HU186877B true HU186877B (en) 1985-10-28

Family

ID=26986839

Family Applications (1)

Application Number Title Priority Date Filing Date
HU823976A HU186877B (en) 1981-12-10 1982-12-09 Process for preparing new hormone antagonists releasing luteinizing hormone and acid addition salts thereof

Country Status (9)

Country Link
EP (1) EP0081877B1 (forum.php)
AU (1) AU9102582A (forum.php)
DE (1) DE3270899D1 (forum.php)
DK (1) DK549882A (forum.php)
ES (1) ES8406418A1 (forum.php)
FI (1) FI824235A7 (forum.php)
GR (1) GR77102B (forum.php)
HU (1) HU186877B (forum.php)
PT (1) PT75955B (forum.php)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4444759A (en) * 1982-07-26 1984-04-24 The Salk Institute For Biological Studies GnRH Antagonists II
IL70888A0 (en) * 1983-03-10 1984-05-31 Salk Inst For Biological Studi Gn rh antagonist peptides and pharmaceutical compositions containing them
DE3467173D1 (en) * 1983-08-16 1987-12-10 Akzo Nv Lh- rh antagonists
US4547370A (en) * 1983-11-29 1985-10-15 The Salk Institute For Biological Studies GnRH Antagonists
IL74827A (en) * 1984-05-21 1989-06-30 Salk Inst For Biological Studi Peptides active as gnrh antagonists and pharmaceutical compositions containing them
US4565804A (en) * 1984-09-07 1986-01-21 The Salk Institute For Biological Studies GnRH Antagonists VI
ZA862570B (en) * 1985-04-09 1986-12-30 Univ Tulane Therapeutic decapeptides
US4866160A (en) * 1985-04-09 1989-09-12 The Administrators Of The Tulane Educational Fund Therapeutic decapeptides
US4800191A (en) * 1987-07-17 1989-01-24 Schally Andrew Victor LHRH antagonists
US4935491A (en) * 1987-08-24 1990-06-19 Board Of Regents, The University Of Texas System Effective antagonists of the luteinizing hormone releasing hormone which release negligible histamine
US5084443A (en) * 1989-12-04 1992-01-28 Biomeasure, Inc. Promoting expression of acetylcholine receptors with lhrh antagonist
US5480969A (en) * 1992-09-15 1996-01-02 The Administrators Of The Tulane Educational Fund Antagonists of LHRH
US5656727A (en) * 1992-09-15 1997-08-12 The Administrators Of The Tulane Educational Fund Antagonists of LHRH
GB0307777D0 (en) 2003-04-04 2003-05-07 Medical Res Council Conjugate compounds
WO2004093807A2 (en) 2003-04-22 2004-11-04 Societe De Conseils De Recherches Et D'applications Scientifiques S.A.S. Somatostatin vectors

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4317815A (en) * 1979-06-13 1982-03-02 Coy David Howard LH-RH Antagonists
ATE8988T1 (de) * 1980-06-02 1984-09-15 Andrew Victor Schally Lh-rh antagonisten.

Also Published As

Publication number Publication date
PT75955A (en) 1983-01-01
DE3270899D1 (en) 1986-06-05
FI824235A0 (fi) 1982-12-09
PT75955B (en) 1985-11-11
EP0081877B1 (en) 1986-04-30
FI824235L (fi) 1983-06-11
ES518060A0 (es) 1984-08-01
DK549882A (da) 1983-06-11
GR77102B (forum.php) 1984-09-06
ES8406418A1 (es) 1984-08-01
AU9102582A (en) 1983-06-16
EP0081877A1 (en) 1983-06-22
FI824235A7 (fi) 1983-06-11

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Legal Events

Date Code Title Description
HU90 Patent valid on 900628