HU183050B - Process for producing n-acyl-derivatives of aminoglycoside antibiotics - Google Patents

Process for producing n-acyl-derivatives of aminoglycoside antibiotics Download PDF

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Publication number
HU183050B
HU183050B HU79ZA414A HUZA000414A HU183050B HU 183050 B HU183050 B HU 183050B HU 79ZA414 A HU79ZA414 A HU 79ZA414A HU ZA000414 A HUZA000414 A HU ZA000414A HU 183050 B HU183050 B HU 183050B
Authority
HU
Hungary
Prior art keywords
zinc
kanamycin
acylated
complex
aminoglycoside antibiotic
Prior art date
Application number
HU79ZA414A
Other languages
English (en)
Hungarian (hu)
Inventor
Hamao Umezawa
Sumio Umezawa
Tsutomu Tsuchiya
Yasushi Takagi
Tomo Jikihara
Original Assignee
Zaidan Hojin Biseibutsu
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zaidan Hojin Biseibutsu filed Critical Zaidan Hojin Biseibutsu
Publication of HU183050B publication Critical patent/HU183050B/hu

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H23/00—Compounds containing boron, silicon, or a metal, e.g. chelates, vitamin B12
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
HU79ZA414A 1978-11-11 1979-11-09 Process for producing n-acyl-derivatives of aminoglycoside antibiotics HU183050B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP13840278A JPS5564598A (en) 1978-11-11 1978-11-11 Preparation of aminoglycoside antibiotic having selectively protected amino group

Publications (1)

Publication Number Publication Date
HU183050B true HU183050B (en) 1984-04-28

Family

ID=15221109

Family Applications (1)

Application Number Title Priority Date Filing Date
HU79ZA414A HU183050B (en) 1978-11-11 1979-11-09 Process for producing n-acyl-derivatives of aminoglycoside antibiotics

Country Status (5)

Country Link
JP (1) JPS5564598A (ja)
BE (1) BE879925A (ja)
CS (1) CS261853B2 (ja)
HU (1) HU183050B (ja)
ZA (1) ZA795691B (ja)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4136254A (en) * 1976-06-17 1979-01-23 Schering Corporation Process of selectively blocking amino functions in aminoglycosides using transition metal salts and intermediates used thereby
EP0446670B1 (en) * 1990-03-08 1994-09-21 Biochimica Opos Spa Method of preparation of amikacin precursors
KR100450607B1 (ko) * 2002-07-11 2004-09-30 경동제약 주식회사 가라민 유도체의 제조방법

Also Published As

Publication number Publication date
CS771179A2 (en) 1988-06-15
BE879925A (fr) 1980-03-03
JPS5564598A (en) 1980-05-15
CS261853B2 (en) 1989-02-10
JPS631319B2 (ja) 1988-01-12
ZA795691B (en) 1980-11-26

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Legal Events

Date Code Title Description
HU90 Patent valid on 900628