HU176023B - Process for producing meso-ionic degehydro derivatives of 1,7-dihydro-1-substituted-3h-pyrasolo-square bracket-4,3-e-square bracket closed-1,2,4-triazolo-square bracket-4,3-c-square bracket closed-pyrimidine-3-thiones and 3-thionones - Google Patents

Process for producing meso-ionic degehydro derivatives of 1,7-dihydro-1-substituted-3h-pyrasolo-square bracket-4,3-e-square bracket closed-1,2,4-triazolo-square bracket-4,3-c-square bracket closed-pyrimidine-3-thiones and 3-thionones Download PDF

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Publication number
HU176023B
HU176023B HU78SU991A HUSU000991A HU176023B HU 176023 B HU176023 B HU 176023B HU 78SU991 A HU78SU991 A HU 78SU991A HU SU000991 A HUSU000991 A HU SU000991A HU 176023 B HU176023 B HU 176023B
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HU
Hungary
Prior art keywords
pyrimidine
pyrazolo
dihydro
methyl
ionic
Prior art date
Application number
HU78SU991A
Other languages
English (en)
Hungarian (hu)
Inventor
Uwe D Treuner
Hermann Breuer
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/833,103 external-priority patent/US4124764A/en
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of HU176023B publication Critical patent/HU176023B/hu

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
HU78SU991A 1977-09-13 1978-09-11 Process for producing meso-ionic degehydro derivatives of 1,7-dihydro-1-substituted-3h-pyrasolo-square bracket-4,3-e-square bracket closed-1,2,4-triazolo-square bracket-4,3-c-square bracket closed-pyrimidine-3-thiones and 3-thionones HU176023B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/833,103 US4124764A (en) 1976-04-21 1977-09-13 Meso-ionic didehydro derivatives of 1,7-dehydro-1-substituted-3H-pyrazolo[4,]-1,2,4-triazolo[4,3-c]pyrimidine-3-thiones and 3-ones

Publications (1)

Publication Number Publication Date
HU176023B true HU176023B (en) 1980-11-28

Family

ID=25263436

Family Applications (1)

Application Number Title Priority Date Filing Date
HU78SU991A HU176023B (en) 1977-09-13 1978-09-11 Process for producing meso-ionic degehydro derivatives of 1,7-dihydro-1-substituted-3h-pyrasolo-square bracket-4,3-e-square bracket closed-1,2,4-triazolo-square bracket-4,3-c-square bracket closed-pyrimidine-3-thiones and 3-thionones

Country Status (13)

Country Link
JP (1) JPS5452098A (no)
AU (1) AU3914178A (no)
BE (1) BE870456A (no)
CA (1) CA1095907A (no)
DE (1) DE2838029A1 (no)
DK (1) DK402178A (no)
FR (1) FR2402658A1 (no)
GB (1) GB2004278B (no)
HU (1) HU176023B (no)
IT (1) IT1099031B (no)
NL (1) NL7809035A (no)
NO (1) NO783086L (no)
SE (1) SE7809601L (no)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4053474A (en) * 1976-04-21 1977-10-11 E. R. Squibb & Sons, Inc. Pyrazolo[4,3-e][1,2,4]triazolo[4,3-c]pyrimidine

Also Published As

Publication number Publication date
DK402178A (da) 1979-03-14
SE7809601L (sv) 1979-03-14
DE2838029A1 (de) 1979-03-22
BE870456A (fr) 1979-03-13
AU3914178A (en) 1980-02-28
GB2004278A (en) 1979-03-28
JPS5452098A (en) 1979-04-24
FR2402658A1 (fr) 1979-04-06
NL7809035A (nl) 1979-03-15
IT7827559A0 (it) 1978-09-12
GB2004278B (en) 1982-01-13
CA1095907A (en) 1981-02-17
IT1099031B (it) 1985-09-18
NO783086L (no) 1979-03-14

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