HRP20160744T1 - Heterocikličke tvari i njihova uporaba kao modulatora receptora tirozin kinaza tipa iii - Google Patents

Heterocikličke tvari i njihova uporaba kao modulatora receptora tirozin kinaza tipa iii

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Publication number
HRP20160744T1
HRP20160744T1 HRP20160744TT HRP20160744T HRP20160744T1 HR P20160744 T1 HRP20160744 T1 HR P20160744T1 HR P20160744T T HRP20160744T T HR P20160744TT HR P20160744 T HRP20160744 T HR P20160744T HR P20160744 T1 HRP20160744 T1 HR P20160744T1
Authority
HR
Croatia
Prior art keywords
modulators
type iii
receptor tyrosine
heterocyclic compounds
tyrosine kinases
Prior art date
Application number
HRP20160744TT
Other languages
English (en)
Inventor
Michael J. Hadd
Michael D. Hocker
Mark W. Holladay
Gang Liu
Martin W. Rowbottom
Shimin Xu
Original Assignee
Ambit Biosciences Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ambit Biosciences Corporation filed Critical Ambit Biosciences Corporation
Publication of HRP20160744T1 publication Critical patent/HRP20160744T1/hr
Publication of HRP20160744T2 publication Critical patent/HRP20160744T2/hr

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
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    • C07—ORGANIC CHEMISTRY
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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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