HRP20030853B1 - Crystalline form of omeprazole - Google Patents
Crystalline form of omeprazoleInfo
- Publication number
- HRP20030853B1 HRP20030853B1 HR20030853A HRP20030853A HRP20030853B1 HR P20030853 B1 HRP20030853 B1 HR P20030853B1 HR 20030853 A HR20030853 A HR 20030853A HR P20030853 A HRP20030853 A HR P20030853A HR P20030853 B1 HRP20030853 B1 HR P20030853B1
- Authority
- HR
- Croatia
- Prior art keywords
- omeprazole
- crystalline form
- powder
- values
- ray diffraction
- Prior art date
Links
- SUBDBMMJDZJVOS-UHFFFAOYSA-N 5-methoxy-2-{[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]sulfinyl}-1H-benzimidazole Chemical compound N=1C2=CC(OC)=CC=C2NC=1S(=O)CC1=NC=C(C)C(OC)=C1C SUBDBMMJDZJVOS-UHFFFAOYSA-N 0.000 title abstract 2
- 229960000381 omeprazole Drugs 0.000 title abstract 2
- 238000000634 powder X-ray diffraction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SI200100111A SI20875A (sl) | 2001-04-25 | 2001-04-25 | Kristalna oblika omeprazola |
PCT/IB2002/001350 WO2002085889A1 (en) | 2001-04-25 | 2002-04-24 | Crystalline form of omeprazole |
Publications (2)
Publication Number | Publication Date |
---|---|
HRP20030853A2 HRP20030853A2 (en) | 2005-08-31 |
HRP20030853B1 true HRP20030853B1 (en) | 2011-11-30 |
Family
ID=20432882
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HR20030853A HRP20030853B1 (en) | 2001-04-25 | 2003-10-20 | Crystalline form of omeprazole |
Country Status (26)
Country | Link |
---|---|
US (2) | US20040122056A1 (sl) |
EP (1) | EP1390360B1 (sl) |
JP (1) | JP4455815B2 (sl) |
KR (1) | KR20030094358A (sl) |
CN (1) | CN1531533B (sl) |
AT (1) | ATE346063T1 (sl) |
AU (1) | AU2002307892B2 (sl) |
BG (1) | BG108287A (sl) |
BR (1) | BR0209103A (sl) |
CA (1) | CA2445251C (sl) |
CZ (1) | CZ20032911A3 (sl) |
DE (1) | DE60216273T2 (sl) |
HR (1) | HRP20030853B1 (sl) |
HU (1) | HUP0303928A2 (sl) |
IL (1) | IL158561A0 (sl) |
MX (1) | MXPA03009789A (sl) |
NO (1) | NO20034715L (sl) |
NZ (1) | NZ528917A (sl) |
PL (1) | PL366471A1 (sl) |
RS (1) | RS50880B (sl) |
RU (1) | RU2286991C2 (sl) |
SI (2) | SI20875A (sl) |
SK (1) | SK13192003A3 (sl) |
UA (1) | UA77671C2 (sl) |
WO (1) | WO2002085889A1 (sl) |
ZA (1) | ZA200307988B (sl) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8993599B2 (en) | 2003-07-18 | 2015-03-31 | Santarus, Inc. | Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them |
US8815916B2 (en) | 2004-05-25 | 2014-08-26 | Santarus, Inc. | Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them |
US8906940B2 (en) | 2004-05-25 | 2014-12-09 | Santarus, Inc. | Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them |
ES2246149B1 (es) * | 2004-07-02 | 2007-06-01 | Esteve Quimica, S.A. | Formas solidas de la sal magnesica de s-omeprazol y procedimientos para su preparacion. |
EP1904064A4 (en) * | 2005-07-07 | 2009-12-02 | Reddys Lab Ltd Dr | OMEPRAZOLE OF FORM B |
EP1988163B1 (en) * | 2006-02-22 | 2012-06-27 | International Institute of Cancer Immunology, Inc. | Hla-a*3303-restricted wt1 peptide and pharmaceutical composition comprising the same |
WO2008067037A2 (en) | 2006-10-05 | 2008-06-05 | Santarus, Inc. | Novel formulations of proton pump inhibitors and methods of using these formulations |
EP2086543A2 (en) | 2006-10-27 | 2009-08-12 | The Curators of the University of Missouri | Compositions comprising at least one acid labile proton pump inhibiting agents, optionally other pharmaceutically active agents and methods of using same |
WO2008092939A2 (en) | 2007-01-31 | 2008-08-07 | Krka, Tovarna Zdravil, D.D., Novo Mesto | Process for the preparation of optically pure omeprazole via salt formation with a chiral amine or treatment with an entiomer converting enzyme and chromatographic separation |
WO2010134099A1 (en) | 2009-05-21 | 2010-11-25 | Cadila Healthcare Limited | One pot process for preparing omeprazole and related compounds |
CN102786513A (zh) * | 2011-05-18 | 2012-11-21 | 中国医学科学院药物研究所 | 奥美拉唑晶e型物质及制备方法与在药品和保健品中应用 |
CN102351846B (zh) * | 2011-09-07 | 2012-08-22 | 周晓东 | 一种新的奥美拉唑钠化合物及其药物组合物 |
KR101459088B1 (ko) * | 2012-08-02 | 2014-12-02 | 대화제약 주식회사 | 알-라베프라졸, 이의 금속염의 제조방법 |
WO2023079094A1 (en) * | 2021-11-05 | 2023-05-11 | Cinclus Pharma Holding AB (publ) | Polymorphs of the hydrochloride salt of linaprazan glurate |
WO2024075017A1 (en) | 2022-10-04 | 2024-04-11 | Zabirnyk Arsenii | Inhibition of aortic valve calcification |
Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0005129A1 (en) * | 1978-04-14 | 1979-10-31 | Aktiebolaget Hässle | Substituted pyridylsulfinylbenzimidazoles having gastric acid secretion properties, pharmaceutical preparations containing same, and intermediates for their preparation |
WO1998028294A1 (en) * | 1996-12-20 | 1998-07-02 | Astra Aktiebolag | A novel compound form |
WO1999008500A2 (en) * | 1998-11-10 | 1999-02-25 | Astrazeneca Ab | New crystalline form of omeprazole |
WO2002000876A1 (en) * | 2000-06-28 | 2002-01-03 | Commonwealth Scientific And Industrial Research Organisation | Truncated egf receptor |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IE67187B1 (en) * | 1990-06-15 | 1996-03-06 | Merck & Co Inc | A crystallization method to improve crystal structure and size |
SI20019A (sl) * | 1998-07-13 | 2000-02-29 | LEK, tovarna farmacevtskih in kemi�nih izdelkov, d.d. | Izboljšan postopek sinteze 5-metoksi -2-/(4-metoksi-3,5-dimetil-2-piridil)metil/ sulfinil-1H-benzimidazola |
US6166213A (en) * | 1998-08-11 | 2000-12-26 | Merck & Co., Inc. | Omeprazole process and compositions thereof |
US6627646B2 (en) * | 2001-07-17 | 2003-09-30 | Sepracor Inc. | Norastemizole polymorphs |
-
2001
- 2001-04-25 SI SI200100111A patent/SI20875A/sl not_active IP Right Cessation
-
2002
- 2002-04-24 IL IL15856102A patent/IL158561A0/xx unknown
- 2002-04-24 EP EP02764081A patent/EP1390360B1/en not_active Expired - Lifetime
- 2002-04-24 CN CN028089553A patent/CN1531533B/zh not_active Expired - Lifetime
- 2002-04-24 RU RU2003133213/04A patent/RU2286991C2/ru active
- 2002-04-24 SI SI200230491T patent/SI1390360T1/sl unknown
- 2002-04-24 UA UA2003109492A patent/UA77671C2/uk unknown
- 2002-04-24 AU AU2002307892A patent/AU2002307892B2/en not_active Expired
- 2002-04-24 NZ NZ528917A patent/NZ528917A/en unknown
- 2002-04-24 SK SK1319-2003A patent/SK13192003A3/sk unknown
- 2002-04-24 HU HU0303928A patent/HUP0303928A2/hu unknown
- 2002-04-24 PL PL02366471A patent/PL366471A1/xx not_active Application Discontinuation
- 2002-04-24 US US10/475,239 patent/US20040122056A1/en not_active Abandoned
- 2002-04-24 KR KR10-2003-7013767A patent/KR20030094358A/ko not_active Application Discontinuation
- 2002-04-24 RS YUP-840/03A patent/RS50880B/sr unknown
- 2002-04-24 MX MXPA03009789A patent/MXPA03009789A/es active IP Right Grant
- 2002-04-24 WO PCT/IB2002/001350 patent/WO2002085889A1/en active IP Right Grant
- 2002-04-24 DE DE60216273T patent/DE60216273T2/de not_active Expired - Lifetime
- 2002-04-24 CZ CZ20032911A patent/CZ20032911A3/cs unknown
- 2002-04-24 JP JP2002583416A patent/JP4455815B2/ja not_active Expired - Lifetime
- 2002-04-24 AT AT02764081T patent/ATE346063T1/de active
- 2002-04-24 CA CA2445251A patent/CA2445251C/en not_active Expired - Lifetime
- 2002-04-24 BR BR0209103-8A patent/BR0209103A/pt not_active Application Discontinuation
-
2003
- 2003-10-14 ZA ZA200307988A patent/ZA200307988B/xx unknown
- 2003-10-20 HR HR20030853A patent/HRP20030853B1/xx not_active IP Right Cessation
- 2003-10-21 NO NO20034715A patent/NO20034715L/no not_active Application Discontinuation
- 2003-10-24 BG BG108287A patent/BG108287A/bg unknown
-
2005
- 2005-10-12 US US11/248,461 patent/US7553856B2/en not_active Expired - Lifetime
Patent Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0005129A1 (en) * | 1978-04-14 | 1979-10-31 | Aktiebolaget Hässle | Substituted pyridylsulfinylbenzimidazoles having gastric acid secretion properties, pharmaceutical preparations containing same, and intermediates for their preparation |
WO1998028294A1 (en) * | 1996-12-20 | 1998-07-02 | Astra Aktiebolag | A novel compound form |
WO1999008500A2 (en) * | 1998-11-10 | 1999-02-25 | Astrazeneca Ab | New crystalline form of omeprazole |
WO2002000876A1 (en) * | 2000-06-28 | 2002-01-03 | Commonwealth Scientific And Industrial Research Organisation | Truncated egf receptor |
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