HK1213256A1 - 作為多巴胺 配體的雜芳族化合物 - Google Patents

作為多巴胺 配體的雜芳族化合物

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Publication number
HK1213256A1
HK1213256A1 HK16101174.8A HK16101174A HK1213256A1 HK 1213256 A1 HK1213256 A1 HK 1213256A1 HK 16101174 A HK16101174 A HK 16101174A HK 1213256 A1 HK1213256 A1 HK 1213256A1
Authority
HK
Hong Kong
Prior art keywords
dopamine
ligands
heteroaromatic compounds
heteroaromatic
compounds
Prior art date
Application number
HK16101174.8A
Other languages
English (en)
Inventor
‧達沃倫
.杜奈
.葉夫列莫夫
.格雷
.門特
.奧尼爾
.羅杰斯
.蘇布拉曼亞姆
.張
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49955424&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1213256(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of HK1213256A1 publication Critical patent/HK1213256A1/zh

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Addiction (AREA)
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  • Endocrinology (AREA)
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  • Emergency Medicine (AREA)
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  • Ophthalmology & Optometry (AREA)
  • Child & Adolescent Psychology (AREA)
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  • Reproductive Health (AREA)
HK16101174.8A 2012-11-08 2016-02-02 作為多巴胺 配體的雜芳族化合物 HK1213256A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261723995P 2012-11-08 2012-11-08
PCT/IB2013/059768 WO2014072882A1 (en) 2012-11-08 2013-10-30 Heteroaromatic compounds as dopamine d1 ligands

Publications (1)

Publication Number Publication Date
HK1213256A1 true HK1213256A1 (zh) 2016-06-30

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ID=49955424

Family Applications (1)

Application Number Title Priority Date Filing Date
HK16101174.8A HK1213256A1 (zh) 2012-11-08 2016-02-02 作為多巴胺 配體的雜芳族化合物

Country Status (30)

Country Link
US (3) US8822494B2 (zh)
EP (1) EP2917216B1 (zh)
JP (1) JP5823657B1 (zh)
KR (1) KR101660664B1 (zh)
CN (1) CN104837839A (zh)
AP (1) AP3861A (zh)
AR (1) AR095359A1 (zh)
AU (1) AU2013343105B2 (zh)
BR (1) BR112015010412A2 (zh)
CA (1) CA2889572C (zh)
CL (1) CL2015001233A1 (zh)
CO (1) CO7350619A2 (zh)
CR (1) CR20150237A (zh)
EA (1) EA201500402A1 (zh)
ES (1) ES2652514T3 (zh)
GE (1) GEP201606598B (zh)
HK (1) HK1213256A1 (zh)
IL (1) IL238712A0 (zh)
MA (1) MA38069A1 (zh)
MD (1) MD20150037A2 (zh)
MX (1) MX2015005506A (zh)
NI (1) NI201500066A (zh)
PE (1) PE20150966A1 (zh)
PH (1) PH12015500883A1 (zh)
SG (1) SG11201502884TA (zh)
TN (1) TN2015000167A1 (zh)
TW (1) TWI577678B (zh)
UA (1) UA111687C2 (zh)
UY (1) UY35129A (zh)
WO (1) WO2014072882A1 (zh)

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EP3137469B1 (en) * 2014-04-28 2019-10-09 Pfizer Inc Heterocyclic compounds and their use as dopamine d1 ligands
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CN115340500A (zh) * 2021-05-14 2022-11-15 广东东阳光药业有限公司 一种含硫化合物的制备方法
WO2023143321A1 (zh) * 2022-01-29 2023-08-03 苏州科睿思制药有限公司 他伐帕敦的晶型及其制备方法和用途
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JP2015535276A (ja) 2015-12-10
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US20140128374A1 (en) 2014-05-08
PE20150966A1 (es) 2015-06-21
US20140336176A1 (en) 2014-11-13
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UA111687C2 (uk) 2016-05-25
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