HK1185875A1 - Novel gpr 119 agonists gpr119 - Google Patents
Novel gpr 119 agonists gpr119Info
- Publication number
- HK1185875A1 HK1185875A1 HK13113263.8A HK13113263A HK1185875A1 HK 1185875 A1 HK1185875 A1 HK 1185875A1 HK 13113263 A HK13113263 A HK 13113263A HK 1185875 A1 HK1185875 A1 HK 1185875A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- gpr119
- agonists
- gpr
- novel
- novel gpr
- Prior art date
Links
- 229940100607 GPR119 agonist Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN2803MU2010 | 2010-10-08 | ||
PCT/IN2011/000694 WO2012046249A1 (en) | 2010-10-08 | 2011-10-05 | Novel gpr 119 agonists |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1185875A1 true HK1185875A1 (en) | 2014-02-28 |
Family
ID=45464048
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK13113263.8A HK1185875A1 (en) | 2010-10-08 | 2013-11-27 | Novel gpr 119 agonists gpr119 |
Country Status (18)
Country | Link |
---|---|
US (1) | US8785463B2 (xx) |
EP (1) | EP2625177B1 (xx) |
JP (1) | JP5814377B2 (xx) |
KR (1) | KR101563793B1 (xx) |
AP (1) | AP2013006812A0 (xx) |
AR (1) | AR083377A1 (xx) |
AU (1) | AU2011311183B2 (xx) |
BR (1) | BR112013007904A2 (xx) |
DK (1) | DK2625177T3 (xx) |
EA (1) | EA022501B1 (xx) |
ES (1) | ES2551183T3 (xx) |
HK (1) | HK1185875A1 (xx) |
MX (1) | MX2013003736A (xx) |
NZ (1) | NZ608708A (xx) |
PL (1) | PL2625177T3 (xx) |
SG (1) | SG188547A1 (xx) |
WO (1) | WO2012046249A1 (xx) |
ZA (1) | ZA201302249B (xx) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2012170867A1 (en) | 2011-06-09 | 2012-12-13 | Rhizen Pharmaceuticals Sa | Novel compounds as modulators of gpr-119 |
AU2013290100A1 (en) | 2012-07-11 | 2015-01-29 | Elcelyx Therapeutics, Inc. | Compositions comprising statins, biguanides and further agents for reducing cardiometabolic risk |
UY39222A (es) | 2020-05-19 | 2021-11-30 | Kallyope Inc | Activadores de la ampk |
EP4172162A4 (en) | 2020-06-26 | 2024-08-07 | Kallyope Inc | AMPK ACTIVATORS |
Family Cites Families (24)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6221660B1 (en) | 1999-02-22 | 2001-04-24 | Synaptic Pharmaceutical Corporation | DNA encoding SNORF25 receptor |
NZ547965A (en) | 2003-12-24 | 2009-12-24 | Prosidion Ltd | 1,2,4-Oxadiazole derivatives as GPCR receptor agonists |
GB0428514D0 (en) | 2004-12-31 | 2005-02-09 | Prosidion Ltd | Compounds |
MY148521A (en) * | 2005-01-10 | 2013-04-30 | Arena Pharm Inc | Substituted pyridinyl and pyrimidinyl derivatives as modulators of metabolism and the treatment of disorders related thereto |
CA2613236A1 (en) | 2005-06-30 | 2007-01-11 | Prosidion Limited | G-protein coupled receptor agonists |
BRPI0613505A2 (pt) | 2005-06-30 | 2011-01-11 | Prosidion Ltd | agonistas de gpcr |
JP2008545008A (ja) | 2005-06-30 | 2008-12-11 | プロシディオン・リミテッド | Gpcrアゴニスト |
EP1910294A1 (en) | 2005-07-27 | 2008-04-16 | Sandoz AG | A process for the preparation of substituted phenyl ether compounds and rosiglitazone |
CA2619093A1 (en) * | 2005-09-16 | 2007-03-29 | Arena Pharmaceuticals, Inc. | Modulators of metabolism and the treatment of disorders related thereto |
MX2008012814A (es) | 2006-04-06 | 2008-10-17 | Prosidion Ltd | Agonistas del receptor acoplado a la proteina g heterociclicos. |
GB0607196D0 (en) | 2006-04-11 | 2006-05-17 | Prosidion Ltd | G-protein coupled receptor agonists |
US8399485B2 (en) | 2006-12-14 | 2013-03-19 | Merck Sharp & Dohme Corp. | Acyl bipiperidinyl compounds useful as GPR 119 agonists |
US7638541B2 (en) | 2006-12-28 | 2009-12-29 | Metabolex Inc. | 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine |
EP2170864B1 (en) | 2007-07-17 | 2011-09-14 | Bristol-Myers Squibb Company | Pyridone gpr119 g protein-coupled receptor agonists |
WO2009046416A1 (en) * | 2007-10-05 | 2009-04-09 | Targegen Inc. | Anilinopyrimidines as jak kinase inhibitors |
CN101896481B (zh) | 2007-10-16 | 2014-04-30 | 第一三共株式会社 | 嘧啶基二氢吲哚化合物 |
WO2009106561A1 (en) | 2008-02-27 | 2009-09-03 | Biovitrum Ab (Publ) | Pyrazine compounds for treating gpr119 related disorders |
US8188098B2 (en) | 2008-05-19 | 2012-05-29 | Hoffmann-La Roche Inc. | GPR119 receptor agonists |
WO2009150144A1 (en) | 2008-06-10 | 2009-12-17 | Inovacia Ab | New gpr119modulators |
MX2011000392A (es) | 2008-07-11 | 2011-03-01 | Irm Llc | 4-fenoxi-metil-piperidinas como moduladoras de la actividad de gpr119. |
TW201006821A (en) | 2008-07-16 | 2010-02-16 | Bristol Myers Squibb Co | Pyridone and pyridazone analogues as GPR119 modulators |
WO2010048149A2 (en) | 2008-10-20 | 2010-04-29 | Kalypsys, Inc. | Heterocyclic modulators of gpr119 for treatment of disease |
JP2012513470A (ja) * | 2008-12-23 | 2012-06-14 | シェーリング コーポレイション | 二環式複素環誘導体及びその使用方法 |
US8742117B2 (en) | 2008-12-24 | 2014-06-03 | Cadila Healthcare Limited | Oxime derivatives |
-
2011
- 2011-10-05 EA EA201390488A patent/EA022501B1/ru not_active IP Right Cessation
- 2011-10-05 NZ NZ608708A patent/NZ608708A/en not_active IP Right Cessation
- 2011-10-05 PL PL11805633T patent/PL2625177T3/pl unknown
- 2011-10-05 BR BR112013007904A patent/BR112013007904A2/pt not_active IP Right Cessation
- 2011-10-05 DK DK11805633.2T patent/DK2625177T3/en active
- 2011-10-05 KR KR1020137008931A patent/KR101563793B1/ko not_active IP Right Cessation
- 2011-10-05 ES ES11805633.2T patent/ES2551183T3/es active Active
- 2011-10-05 AU AU2011311183A patent/AU2011311183B2/en not_active Ceased
- 2011-10-05 MX MX2013003736A patent/MX2013003736A/es active IP Right Grant
- 2011-10-05 SG SG2013019062A patent/SG188547A1/en unknown
- 2011-10-05 EP EP11805633.2A patent/EP2625177B1/en active Active
- 2011-10-05 AP AP2013006812A patent/AP2013006812A0/xx unknown
- 2011-10-05 JP JP2013532319A patent/JP5814377B2/ja not_active Expired - Fee Related
- 2011-10-05 WO PCT/IN2011/000694 patent/WO2012046249A1/en active Application Filing
- 2011-10-05 US US13/824,552 patent/US8785463B2/en not_active Expired - Fee Related
- 2011-10-11 AR ARP110103746A patent/AR083377A1/es unknown
-
2013
- 2013-03-26 ZA ZA2013/02249A patent/ZA201302249B/en unknown
- 2013-11-27 HK HK13113263.8A patent/HK1185875A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
EA201390488A1 (ru) | 2013-08-30 |
US8785463B2 (en) | 2014-07-22 |
KR20130064801A (ko) | 2013-06-18 |
NZ608708A (en) | 2015-05-29 |
KR101563793B1 (ko) | 2015-10-27 |
EP2625177A1 (en) | 2013-08-14 |
PL2625177T3 (pl) | 2015-12-31 |
SG188547A1 (en) | 2013-04-30 |
BR112013007904A2 (pt) | 2019-09-24 |
US20130252980A1 (en) | 2013-09-26 |
WO2012046249A1 (en) | 2012-04-12 |
ES2551183T3 (es) | 2015-11-16 |
ZA201302249B (en) | 2013-12-23 |
AU2011311183B2 (en) | 2014-09-25 |
AP2013006812A0 (en) | 2013-04-30 |
JP2013538870A (ja) | 2013-10-17 |
EP2625177B1 (en) | 2015-07-29 |
AR083377A1 (es) | 2013-02-21 |
MX2013003736A (es) | 2013-05-09 |
JP5814377B2 (ja) | 2015-11-17 |
AU2011311183A1 (en) | 2013-04-04 |
DK2625177T3 (en) | 2015-10-12 |
EA022501B1 (ru) | 2016-01-29 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20191008 |