HK1182384A1 - 激酶抑制劑的結晶形式 - Google Patents

激酶抑制劑的結晶形式

Info

Publication number
HK1182384A1
HK1182384A1 HK13109691.8A HK13109691A HK1182384A1 HK 1182384 A1 HK1182384 A1 HK 1182384A1 HK 13109691 A HK13109691 A HK 13109691A HK 1182384 A1 HK1182384 A1 HK 1182384A1
Authority
HK
Hong Kong
Prior art keywords
kinase inhibitors
crystalline forms
crystalline
forms
kinase
Prior art date
Application number
HK13109691.8A
Other languages
English (en)
Inventor
Geoff G Z Zhang
Paul J Brackemeyer
Ahmad Y Sheikh
Original Assignee
Abbvie Bahamas Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbvie Bahamas Ltd filed Critical Abbvie Bahamas Ltd
Publication of HK1182384A1 publication Critical patent/HK1182384A1/zh

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/28—Compounds containing heavy metals
    • A61K31/282—Platinum compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HK13109691.8A 2010-06-09 2013-08-20 激酶抑制劑的結晶形式 HK1182384A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35305810P 2010-06-09 2010-06-09
PCT/US2011/039582 WO2011156461A1 (en) 2010-06-09 2011-06-08 Crystalline forms of kinase inhibitors

Publications (1)

Publication Number Publication Date
HK1182384A1 true HK1182384A1 (zh) 2013-11-29

Family

ID=44454740

Family Applications (1)

Application Number Title Priority Date Filing Date
HK13109691.8A HK1182384A1 (zh) 2010-06-09 2013-08-20 激酶抑制劑的結晶形式

Country Status (18)

Country Link
US (2) US8357804B2 (zh)
EP (1) EP2580219B1 (zh)
JP (1) JP5711814B2 (zh)
KR (1) KR20130112855A (zh)
CN (1) CN103025741A (zh)
AR (1) AR083722A1 (zh)
AU (1) AU2011264899B2 (zh)
BR (1) BR112012031469A2 (zh)
CA (1) CA2802064A1 (zh)
ES (1) ES2537708T3 (zh)
HK (1) HK1182384A1 (zh)
MX (1) MX2012014385A (zh)
NZ (1) NZ605436A (zh)
RU (1) RU2012157471A (zh)
SG (1) SG186249A1 (zh)
TW (1) TWI492949B (zh)
WO (1) WO2011156461A1 (zh)
ZA (1) ZA201209647B (zh)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2021012250A (es) * 2019-04-11 2022-01-18 Angion Biomedica Corp Formas solidas de (e)-3-[2-(2-tienil)vinil]-1h-pirazol.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050026944A1 (en) * 2003-07-24 2005-02-03 Patrick Betschmann Thienopyridine and furopyridine kinase inhibitors
GB0402518D0 (en) * 2004-02-05 2004-03-10 Astrazeneca Ab Therapeutic agents
US20070135387A1 (en) * 2005-12-08 2007-06-14 Michaelides Michael R Inhibitors of protein kinases
RU2498988C2 (ru) * 2008-03-05 2013-11-20 Метилджин, Инк. Ингибиторы активности протеинтирозинкиназы
MY179042A (en) 2008-12-05 2020-10-26 Abbvie Bahamas Ltd Kinase inhibitors with improved cyp safety profile

Also Published As

Publication number Publication date
WO2011156461A1 (en) 2011-12-15
ES2537708T3 (es) 2015-06-11
NZ605436A (en) 2014-11-28
JP5711814B2 (ja) 2015-05-07
US20120149726A1 (en) 2012-06-14
SG186249A1 (en) 2013-01-30
RU2012157471A (ru) 2014-07-20
US8592589B2 (en) 2013-11-26
AU2011264899A1 (en) 2013-01-10
AR083722A1 (es) 2013-03-20
TW201204736A (en) 2012-02-01
JP2013528220A (ja) 2013-07-08
AU2011264899B2 (en) 2015-01-22
CN103025741A (zh) 2013-04-03
US8357804B2 (en) 2013-01-22
EP2580219A1 (en) 2013-04-17
EP2580219B1 (en) 2015-02-25
MX2012014385A (es) 2013-05-01
TWI492949B (zh) 2015-07-21
BR112012031469A2 (pt) 2016-11-01
KR20130112855A (ko) 2013-10-14
ZA201209647B (en) 2014-02-26
US20130136804A1 (en) 2013-05-30
CA2802064A1 (en) 2011-12-15

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20190607