HK1176236A1 - Thiazolo[5,4-d] pyrimidines and their use as agrochemicals [54-d] - Google Patents

Thiazolo[5,4-d] pyrimidines and their use as agrochemicals [54-d]

Info

Publication number
HK1176236A1
HK1176236A1 HK13103749.3A HK13103749A HK1176236A1 HK 1176236 A1 HK1176236 A1 HK 1176236A1 HK 13103749 A HK13103749 A HK 13103749A HK 1176236 A1 HK1176236 A1 HK 1176236A1
Authority
HK
Hong Kong
Prior art keywords
thiazolo
agrochemicals
pyrimidines
Prior art date
Application number
HK13103749.3A
Other languages
English (en)
Chinese (zh)
Inventor
William Brewster
Carla Klittich
Brent Rieder
Thomas Siddall
Chenglin Yao
Original Assignee
陶氏益農公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 陶氏益農公司 filed Critical 陶氏益農公司
Publication of HK1176236A1 publication Critical patent/HK1176236A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Zoology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
HK13103749.3A 2010-01-07 2013-03-26 Thiazolo[5,4-d] pyrimidines and their use as agrochemicals [54-d] HK1176236A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US29301410P 2010-01-07 2010-01-07
PCT/US2011/020351 WO2011085084A1 (en) 2010-01-07 2011-01-06 THIAZOLO[5,4-d] PYRIMIDINES AND THEIR USE AS AGROCHEMICALS

Publications (1)

Publication Number Publication Date
HK1176236A1 true HK1176236A1 (en) 2013-07-26

Family

ID=44225056

Family Applications (1)

Application Number Title Priority Date Filing Date
HK13103749.3A HK1176236A1 (en) 2010-01-07 2013-03-26 Thiazolo[5,4-d] pyrimidines and their use as agrochemicals [54-d]

Country Status (19)

Country Link
US (1) US8921382B2 (el)
EP (1) EP2521452B1 (el)
JP (1) JP5781090B2 (el)
KR (1) KR101814835B1 (el)
CN (1) CN102791135B (el)
BR (1) BR112012016866A2 (el)
CA (1) CA2786250A1 (el)
CL (1) CL2012001851A1 (el)
CO (1) CO6612238A2 (el)
ES (1) ES2529247T3 (el)
HK (1) HK1176236A1 (el)
IN (1) IN2012DN06323A (el)
MX (1) MX2012007954A (el)
PL (1) PL2521452T3 (el)
PT (1) PT2521452E (el)
RU (1) RU2547721C2 (el)
UA (1) UA109780C2 (el)
WO (1) WO2011085084A1 (el)
ZA (1) ZA201204871B (el)

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ME01838B (me) 2009-06-29 2014-12-20 Lncyte Holdings Corp Pirimidinoni kao inhibitori pi3k
AR088218A1 (es) 2011-07-19 2014-05-21 Infinity Pharmaceuticals Inc Compuestos heterociclicos utiles como inhibidores de pi3k
WO2013031694A1 (ja) * 2011-08-26 2013-03-07 富山化学工業株式会社 アミン化合物またはその塩
KR102371532B1 (ko) 2011-09-02 2022-03-07 인사이트 홀딩스 코포레이션 Pi3k 억제제로서 헤테로시클릴아민
AU2013214353A1 (en) 2012-02-03 2014-08-21 Basf Se Fungicidal pyrimidine compounds
IN2014DN07220A (el) 2012-02-03 2015-04-24 Basf Se
WO2013135672A1 (en) 2012-03-13 2013-09-19 Basf Se Fungicidal pyrimidine compounds
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
CN103668956B (zh) * 2012-09-21 2015-08-12 上海韬鸿化工科技有限公司 防螨虫整理剂、织物的防螨虫整理方法及防螨虫织物
BR112015023640A2 (pt) * 2013-03-15 2017-07-18 Univ California métodos para identificar repelentes e atraentes de artrópodes e compostos e composições identificados por tais métodos
US10077277B2 (en) 2014-06-11 2018-09-18 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
CN105594748A (zh) * 2014-10-15 2016-05-25 浙江新安化工集团股份有限公司 一种精准定向、高效的防治鳞翅目害虫的杀虫组合物及其使用方法
CN104391070B (zh) * 2014-12-05 2016-06-08 山东省城市供排水水质监测中心 一种水中烷基汞的检测方法
NZ734993A (en) 2015-02-27 2024-03-22 Incyte Holdings Corp Salts of pi3k inhibitor and processes for their preparation
WO2016149567A1 (en) 2015-03-18 2016-09-22 The Regents Of The University Of California Anthropod repellent chemicals
US9988401B2 (en) 2015-05-11 2018-06-05 Incyte Corporation Crystalline forms of a PI3K inhibitor
CN105606755A (zh) * 2016-01-30 2016-05-25 郭庆龙 一种胺苯吡唑酮残留量的gc-nci-ms测定方法
CA3050864A1 (en) 2017-01-26 2018-08-02 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
EP3611166B1 (en) 2017-04-10 2022-09-21 Mitsui Chemicals Agro, Inc. Pyridone compound, and agricultural and horticultural fungicide having this as active component
US11147272B2 (en) 2017-04-10 2021-10-19 Mitsui Chemicals Argro, Inc. Pyridone compounds and agricultural and horticultural fungicides comprising the same as active ingredients
CN110234627B (zh) 2017-04-11 2023-09-01 三井化学植保株式会社 吡啶酮化合物及以吡啶酮化合物作为有效成分的农园艺用杀菌剂
WO2018225829A1 (ja) 2017-06-08 2018-12-13 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
TWI828725B (zh) 2018-07-25 2024-01-11 日商三井化學植保股份有限公司 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑
CN112010848B (zh) * 2020-09-29 2021-12-24 南通大学 含三氟甲基吡啶联芳氧基结构的1,3,4-噁二唑类化合物的制备方法和应用
CN116250525A (zh) * 2023-03-08 2023-06-13 内蒙古民族大学 一种小型哺乳类剥制标本安全防腐剂及其制备方法

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Also Published As

Publication number Publication date
MX2012007954A (es) 2012-08-03
ES2529247T3 (es) 2015-02-18
BR112012016866A2 (pt) 2015-09-01
US20110166164A1 (en) 2011-07-07
ZA201204871B (en) 2013-09-25
JP2013516476A (ja) 2013-05-13
EP2521452B1 (en) 2014-12-24
CL2012001851A1 (es) 2012-12-14
JP5781090B2 (ja) 2015-09-16
PT2521452E (pt) 2015-02-24
IN2012DN06323A (el) 2015-10-02
RU2012133570A (ru) 2014-02-20
CO6612238A2 (es) 2013-02-01
UA109780C2 (uk) 2015-10-12
CN102791135B (zh) 2015-05-20
CA2786250A1 (en) 2011-07-14
RU2547721C2 (ru) 2015-04-10
WO2011085084A1 (en) 2011-07-14
CN102791135A (zh) 2012-11-21
KR101814835B1 (ko) 2018-01-04
EP2521452A4 (en) 2013-07-03
PL2521452T3 (pl) 2015-05-29
EP2521452A1 (en) 2012-11-14
KR20120115538A (ko) 2012-10-18
US8921382B2 (en) 2014-12-30

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PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20200106