HK1175780A1 - 晶體 抑制劑鹽 - Google Patents

晶體 抑制劑鹽

Info

Publication number
HK1175780A1
HK1175780A1 HK13103038.3A HK13103038A HK1175780A1 HK 1175780 A1 HK1175780 A1 HK 1175780A1 HK 13103038 A HK13103038 A HK 13103038A HK 1175780 A1 HK1175780 A1 HK 1175780A1
Authority
HK
Hong Kong
Prior art keywords
cdc7
crystalline
inhibitor salts
salts
inhibitor
Prior art date
Application number
HK13103038.3A
Other languages
English (en)
Inventor
.贊姆皮裡
.瓦諾蒂
.西瓦羅裡
.弗納雷托
Original Assignee
內爾維阿諾醫學科學有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 內爾維阿諾醫學科學有限公司 filed Critical 內爾維阿諾醫學科學有限公司
Publication of HK1175780A1 publication Critical patent/HK1175780A1/zh

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Transplantation (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK13103038.3A 2009-11-11 2013-03-12 晶體 抑制劑鹽 HK1175780A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP09175648 2009-11-11
PCT/EP2010/066873 WO2011057960A1 (en) 2009-11-11 2010-11-05 Crystalline cdc7 inhibitor salts

Publications (1)

Publication Number Publication Date
HK1175780A1 true HK1175780A1 (zh) 2013-07-12

Family

ID=43513935

Family Applications (1)

Application Number Title Priority Date Filing Date
HK13103038.3A HK1175780A1 (zh) 2009-11-11 2013-03-12 晶體 抑制劑鹽

Country Status (9)

Country Link
US (1) US8658662B2 (zh)
EP (1) EP2499128B1 (zh)
JP (1) JP5856971B2 (zh)
CN (1) CN102666528B (zh)
AR (1) AR078960A1 (zh)
ES (1) ES2543098T3 (zh)
HK (1) HK1175780A1 (zh)
TW (1) TW201125861A (zh)
WO (1) WO2011057960A1 (zh)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112013026137B1 (pt) * 2011-04-19 2020-12-01 Nerviano Medical Sciences S.R.L pirimidinil-pirróis substituídos ativos como inibidores da quinase
JP6016915B2 (ja) * 2011-07-28 2016-10-26 ネルビアーノ・メデイカル・サイエンシーズ・エツセ・エルレ・エルレ キナーゼ阻害剤として活性なアルキニル置換ピリミジニルピロール

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0202463D0 (sv) * 2002-08-14 2002-08-14 Astrazeneca Ab Novel compounds
MX2008012422A (es) * 2006-03-27 2008-10-09 Nerviano Medical Sciences Srl Derivados de furano y tiofeno, pirrol substituido con pirimidinil y piridil como inhibidores de cinasa.
TWI426074B (zh) * 2008-04-30 2014-02-11 Nerviano Medical Sciences Srl 5-(2-胺基-嘧啶-4-基)-2-芳基-1h-吡咯-3-羧醯胺之製造方法

Also Published As

Publication number Publication date
TW201125861A (en) 2011-08-01
CN102666528B (zh) 2014-04-16
EP2499128A1 (en) 2012-09-19
US20120245189A1 (en) 2012-09-27
CN102666528A (zh) 2012-09-12
JP5856971B2 (ja) 2016-02-10
ES2543098T3 (es) 2015-08-14
WO2011057960A1 (en) 2011-05-19
US8658662B2 (en) 2014-02-25
AR078960A1 (es) 2011-12-14
EP2499128B1 (en) 2015-06-03
JP2013510811A (ja) 2013-03-28

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