GT200900284A - Dosis intravenosa y oral de un inhibidor p2y12 de accion directa y reversible.- - Google Patents
Dosis intravenosa y oral de un inhibidor p2y12 de accion directa y reversible.-Info
- Publication number
- GT200900284A GT200900284A GT200900284A GT200900284A GT200900284A GT 200900284 A GT200900284 A GT 200900284A GT 200900284 A GT200900284 A GT 200900284A GT 200900284 A GT200900284 A GT 200900284A GT 200900284 A GT200900284 A GT 200900284A
- Authority
- GT
- Guatemala
- Prior art keywords
- reversible
- direct
- intravenous
- inhibitor
- oral dose
- Prior art date
Links
- 230000002441 reversible effect Effects 0.000 title abstract 2
- 239000002172 P2Y12 inhibitor Substances 0.000 title 1
- 238000001990 intravenous administration Methods 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- BSYNRYMUTXBXSQ-UHFFFAOYSA-N Aspirin Chemical compound CC(=O)OC1=CC=CC=C1C(O)=O BSYNRYMUTXBXSQ-UHFFFAOYSA-N 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 230000005764 inhibitory process Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Emergency Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US91564907P | 2007-05-02 | 2007-05-02 | |
| US94792107P | 2007-07-03 | 2007-07-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GT200900284A true GT200900284A (es) | 2012-01-31 |
Family
ID=39587015
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GT200900284A GT200900284A (es) | 2007-05-02 | 2009-10-30 | Dosis intravenosa y oral de un inhibidor p2y12 de accion directa y reversible.- |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US20090048216A1 (enExample) |
| EP (1) | EP2079464A2 (enExample) |
| JP (1) | JP2010526101A (enExample) |
| KR (1) | KR20100029746A (enExample) |
| CN (1) | CN101795682A (enExample) |
| AU (1) | AU2008247483A1 (enExample) |
| BR (1) | BRPI0811476A2 (enExample) |
| CA (1) | CA2686203A1 (enExample) |
| CO (1) | CO6241104A2 (enExample) |
| EA (1) | EA200901473A1 (enExample) |
| EC (1) | ECSP099778A (enExample) |
| GT (1) | GT200900284A (enExample) |
| IL (1) | IL201834A0 (enExample) |
| MA (1) | MA31663B1 (enExample) |
| MX (1) | MX2009011843A (enExample) |
| TN (1) | TN2009000451A1 (enExample) |
| WO (1) | WO2008137753A2 (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5509406B2 (ja) * | 2005-11-03 | 2014-06-04 | ポートラ ファーマシューティカルズ， インコーポレイテッド | ［４−（６−ハロ−７−置換−２，４−ジオキソ−１，４−ジヒドロ−２ｈ−キナゾリン−３−イル）−フェニル］−５−クロロ−チオフェン−２−イル−スルホニル尿素、ならびにそれに関連する形態および方法 |
| US8633211B2 (en) * | 2007-03-06 | 2014-01-21 | Novartis Ag | Bicyclic organic compounds suitable for the treatment of inflammatory or allergic conditions |
| MX2009011836A (es) * | 2007-05-02 | 2010-05-20 | Portola Pharm Inc | Sales de [4-(6-fluoro-7-metilamino-2,4-dioxo-1,4-dihidro-2h-quinaz olin-3-il)-fenil]-5-cloro-tiofen-2-il-sulfonilurea, en diferentes formas cristalinas, y composiciones farmaceuticas de las mismas. |
| US20090156620A1 (en) * | 2007-05-02 | 2009-06-18 | Portola Pharmaceuticals, Inc. | [4-(6-fluoro-7-methylamino-2,4-dioxo-1,4-dihydro-2h-quinazolin-3-yl)-phenyl]-5-chloro-thiophen-2-yl-sulfonylurea salts, forms and methods related thereto |
| US9427448B2 (en) * | 2009-11-11 | 2016-08-30 | The Medicines Company | Methods of treating, reducing the incidence of, and/or preventing ischemic events |
| CN102271685A (zh) * | 2008-12-30 | 2011-12-07 | 斯若姆博洛捷克有限公司 | 鉴定发展成器官功能衰竭的风险提高的危重患者的方法及用于其治疗的化合物 |
| US10376532B2 (en) | 2009-11-11 | 2019-08-13 | Chiesi Farmaceutici, S.P.A. | Methods of treating, reducing the incidence of, and/or preventing ischemic events |
| WO2011060066A2 (en) | 2009-11-11 | 2011-05-19 | The Medicines Company | Methods of treating or preventing stent thrombosis |
| EP2633857B1 (en) * | 2009-12-23 | 2015-08-12 | ratiopharm GmbH | Solid pharmaceutical dosage form of ticagrelor and acetylsalicylic acid |
| WO2011088152A1 (en) | 2010-01-12 | 2011-07-21 | Portola Pharmaceuticals, Inc. | Pharmaceutical composition and dosage forms of elinogrel and methods of use thereof |
| WO2011137459A1 (en) * | 2010-04-30 | 2011-11-03 | Portola Pharmaceuticals, Inc. | Dosage forms of elinogrel and methods of injectable administration thereof |
| EP2646827A1 (en) * | 2010-12-01 | 2013-10-09 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Method and kits for determining platelet susceptibility to activation in a patient |
| WO2012072824A1 (en) * | 2010-12-03 | 2012-06-07 | Novartis Ag | Pharmaceutical compositions, dosage forms and new forms of the compound of formula (i), and methods of use thereof |
| MX393334B (es) | 2017-03-15 | 2025-03-24 | Idorsia Pharmaceuticals Ltd | Administración subcutánea de un antagonista del receptor p2y12. |
| MA49452A (fr) | 2017-06-23 | 2021-05-05 | Chiesi Farm Spa | Procédé de prévention de thrombose de shunt de l'artère systémique-pulmonaire |
| CN107462648B (zh) * | 2017-08-21 | 2019-09-27 | 盐城锦明药业有限公司 | 一种Cangrelor中间体腺苷-2-硫酮的高效液相色谱检测方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6906063B2 (en) * | 2000-02-04 | 2005-06-14 | Portola Pharmaceuticals, Inc. | Platelet ADP receptor inhibitors |
| JP5509406B2 (ja) | 2005-11-03 | 2014-06-04 | ポートラ ファーマシューティカルズ， インコーポレイテッド | ［４−（６−ハロ−７−置換−２，４−ジオキソ−１，４−ジヒドロ−２ｈ−キナゾリン−３−イル）−フェニル］−５−クロロ−チオフェン−２−イル−スルホニル尿素、ならびにそれに関連する形態および方法 |
-
2008
- 2008-05-02 EA EA200901473A patent/EA200901473A1/ru unknown
- 2008-05-02 BR BRPI0811476-5A2A patent/BRPI0811476A2/pt not_active IP Right Cessation
- 2008-05-02 WO PCT/US2008/062518 patent/WO2008137753A2/en not_active Ceased
- 2008-05-02 JP JP2010506688A patent/JP2010526101A/ja not_active Withdrawn
- 2008-05-02 EP EP08747561A patent/EP2079464A2/en not_active Withdrawn
- 2008-05-02 MX MX2009011843A patent/MX2009011843A/es not_active Application Discontinuation
- 2008-05-02 KR KR1020097025059A patent/KR20100029746A/ko not_active Withdrawn
- 2008-05-02 CN CN200880023071A patent/CN101795682A/zh active Pending
- 2008-05-02 US US12/114,630 patent/US20090048216A1/en not_active Abandoned
- 2008-05-02 AU AU2008247483A patent/AU2008247483A1/en not_active Abandoned
- 2008-05-02 CA CA002686203A patent/CA2686203A1/en not_active Abandoned
-
2009
- 2009-10-29 IL IL201834A patent/IL201834A0/en unknown
- 2009-10-30 TN TNP2009000451A patent/TN2009000451A1/fr unknown
- 2009-10-30 GT GT200900284A patent/GT200900284A/es unknown
- 2009-11-26 MA MA32377A patent/MA31663B1/fr unknown
- 2009-12-02 EC EC2009009778A patent/ECSP099778A/es unknown
- 2009-12-02 CO CO09137697A patent/CO6241104A2/es not_active Application Discontinuation
-
2011
- 2011-09-16 US US13/235,305 patent/US20120009172A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN101795682A (zh) | 2010-08-04 |
| MX2009011843A (es) | 2010-04-22 |
| EP2079464A2 (en) | 2009-07-22 |
| IL201834A0 (en) | 2010-06-16 |
| WO2008137753A2 (en) | 2008-11-13 |
| ECSP099778A (es) | 2010-01-29 |
| CO6241104A2 (es) | 2011-01-20 |
| BRPI0811476A2 (pt) | 2014-11-04 |
| WO2008137753A3 (en) | 2009-02-12 |
| MA31663B1 (fr) | 2010-09-01 |
| AU2008247483A1 (en) | 2008-11-13 |
| TN2009000451A1 (en) | 2011-03-31 |
| CA2686203A1 (en) | 2008-11-13 |
| US20090048216A1 (en) | 2009-02-19 |
| KR20100029746A (ko) | 2010-03-17 |
| US20120009172A1 (en) | 2012-01-12 |
| EA200901473A1 (ru) | 2010-06-30 |
| JP2010526101A (ja) | 2010-07-29 |
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