GT200600365A - Aciltriptofanoles - Google Patents

Aciltriptofanoles

Info

Publication number
GT200600365A
GT200600365A GT200600365A GT200600365A GT200600365A GT 200600365 A GT200600365 A GT 200600365A GT 200600365 A GT200600365 A GT 200600365A GT 200600365 A GT200600365 A GT 200600365A GT 200600365 A GT200600365 A GT 200600365A
Authority
GT
Guatemala
Prior art keywords
aciltriptofanoles
anthogonists
aciltriptophenols
fsh
fertility
Prior art date
Application number
GT200600365A
Other languages
English (en)
Inventor
Wortmann Lars
Cleve Arwed
Menzenbach Bernd
Muhn Hans-Peter
Langer Gernot
Schrey Anna
Kuehne Ronald
Koppitz Marcus
Kosemund Dirk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT200600365A publication Critical patent/GT200600365A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/12Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Reproductive Health (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Pregnancy & Childbirth (AREA)
  • Gynecology & Obstetrics (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

LA PRESENTE INVENCIÓN SE REFIERE A ACILTRIPTOFENOLES DE FÓRMULA GENERAL (I), EN DONDE Q, X, Y, R1, R2, R3, R4, R5, R6 SON GRUPOS QUE SE ENCUENTRAN DEFINIDOS EN LA DESCRIPCIÓN. DICHOS COMPUESTOS SON EFICACES ANTAGONISTAS DE FSH Y SE PUEDEN USAR, POR EJEMPLO, PARA EL CONTROL DE LA FERTILIDAD EN EL HOMBRE O EN LA MUJER, O PARA LA PREVENCIÓN Y/O EL TRATAMIENTO DE OSTEOPOROSIS.
GT200600365A 2005-08-10 2006-08-09 Aciltriptofanoles GT200600365A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102005038632A DE102005038632B4 (de) 2005-08-10 2005-08-10 Acyltryptophanole

Publications (1)

Publication Number Publication Date
GT200600365A true GT200600365A (es) 2007-04-02

Family

ID=37681170

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200600365A GT200600365A (es) 2005-08-10 2006-08-09 Aciltriptofanoles

Country Status (7)

Country Link
AR (1) AR056190A1 (es)
DE (1) DE102005038632B4 (es)
DO (1) DOP2006000187A (es)
GT (1) GT200600365A (es)
PE (1) PE20070406A1 (es)
TW (1) TW200716098A (es)
UY (1) UY29737A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102008025893B4 (de) * 2008-05-26 2014-09-18 Technische Universität Dresden Verfahren zur Herstellung von Fettsäureamiden mit gesättigten, ungesättigten oder Hydroxy-Fettsäuren

Also Published As

Publication number Publication date
UY29737A1 (es) 2007-02-28
PE20070406A1 (es) 2007-05-12
AR056190A1 (es) 2007-09-26
DE102005038632B4 (de) 2008-03-27
DE102005038632A1 (de) 2007-02-15
DOP2006000187A (es) 2007-03-15
TW200716098A (en) 2007-05-01

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GT200600365A (es) Aciltriptofanoles