GR78987B - - Google Patents
Info
- Publication number
- GR78987B GR78987B GR72382A GR830172382A GR78987B GR 78987 B GR78987 B GR 78987B GR 72382 A GR72382 A GR 72382A GR 830172382 A GR830172382 A GR 830172382A GR 78987 B GR78987 B GR 78987B
- Authority
- GR
- Greece
- Prior art keywords
- lopyridines
- ansiolytic
- pyrazo
- analgetic
- antiinflammatory
- Prior art date
Links
- 230000000202 analgesic effect Effects 0.000 abstract 1
- 230000003110 anti-inflammatory effect Effects 0.000 abstract 1
- 230000000949 anxiolytic effect Effects 0.000 abstract 1
- 239000003874 central nervous system depressant Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 150000005229 pyrazolopyridines Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT23375/82A IT1154024B (it) | 1982-09-22 | 1982-09-22 | Derivati pridinici e procedimento per la loro produzione |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GR78987B true GR78987B (enEXAMPLES) | 1984-10-02 |
Family
ID=11206534
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GR72382A GR78987B (enEXAMPLES) | 1982-09-22 | 1983-09-05 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US4612318A (enEXAMPLES) |
| EP (1) | EP0104522B1 (enEXAMPLES) |
| JP (1) | JPS5989679A (enEXAMPLES) |
| AT (1) | ATE63913T1 (enEXAMPLES) |
| CA (1) | CA1248532A (enEXAMPLES) |
| DE (1) | DE3382299D1 (enEXAMPLES) |
| ES (1) | ES525786A0 (enEXAMPLES) |
| GR (1) | GR78987B (enEXAMPLES) |
| IT (1) | IT1154024B (enEXAMPLES) |
| PT (1) | PT77370B (enEXAMPLES) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ208555A (en) * | 1983-06-23 | 1987-06-30 | American Cyanamid Co | (3-amino-1h-pyrazol-4-yl)-arylmethanone derivatives |
| US4751226A (en) * | 1985-09-12 | 1988-06-14 | Fujisawa Pharmaceutical Co., Ltd. | Pyrazoloisoquinoline derivatives, plant growth regulating compositions, and method of use therefor |
| JPH0615542B2 (ja) * | 1986-07-22 | 1994-03-02 | 吉富製薬株式会社 | ピラゾロピリジン化合物 |
| US5006520A (en) * | 1987-10-13 | 1991-04-09 | Yoshitomi Pharmaceutical Industries, Ltd. | Fused pyrazole compounds and pharmaceutical use thereof |
| TW370529B (en) | 1992-12-17 | 1999-09-21 | Pfizer | Pyrazolopyrimidines |
| PL181895B1 (pl) * | 1994-06-16 | 2001-10-31 | Pfizer | Nowe pirazolo-i pirolopirydyny _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ PL PL PL PL |
| AU2001264313A1 (en) * | 2000-06-20 | 2002-01-02 | Japan Tobacco Inc. | Pyrazolopyridine compounds and use thereof as drugs |
| WO2003020313A1 (fr) * | 2001-09-04 | 2003-03-13 | Ono Pharmaceutical Co., Ltd. | Medicaments contre les maladies respiratoires renfermant un agent de regulation du recepteur de la sphingosine-1-phosphate |
| PT1522314E (pt) * | 2002-06-26 | 2014-06-05 | Ono Pharmaceutical Co | Medicamentos para doenças causadas pela contracção ou dilatação vascular |
| RU2006134020A (ru) * | 2004-02-27 | 2008-04-10 | Ф.Хоффманн-Ля Рош Аг (Ch) | Конденсированные производные пиразола |
| EP1747202A1 (en) | 2004-02-27 | 2007-01-31 | F.Hoffmann-La Roche Ag | Indazole derivatives and pharmaceutical compositions containing them |
| RU2006134021A (ru) | 2004-02-27 | 2008-04-10 | Ф.Хоффманн-Ля Рош Аг (Ch) | Производные гетероарил-конденсированного пиразола |
| JP2009506007A (ja) | 2005-08-25 | 2009-02-12 | エフ．ホフマン−ラ ロシュ アーゲー | ｐ３８ＭＡＰキナーゼ阻害剤及びその使用方法 |
| CN101421268B (zh) * | 2006-02-15 | 2016-01-06 | Abbvie公司 | 作为有效parp抑制剂的吡唑并喹诺酮 |
| MX2011006959A (es) | 2008-12-30 | 2011-12-06 | Arqule Inc | Compuestos substituidos de 5,6-dihidro-6-fenilbenzo [f] isoquinolina-2-amina. |
| WO2010078427A1 (en) * | 2008-12-30 | 2010-07-08 | Arqule, Inc. | Substituted pyrazolo [3, 4-b] pyridine compounds |
| WO2011159864A1 (en) * | 2010-06-17 | 2011-12-22 | Bracco Imaging S.P.A. | Jte013 analogs and methods of making and using same |
| RU2495039C1 (ru) * | 2012-07-31 | 2013-10-10 | Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Пермский государственный национальный исследовательский университет" | МЕТИЛ 3-МЕТИЛ-5-[2-(4-АРИЛАМИНО)-2-ОКСОАЦЕТИЛ]-1,6-ДИФЕНИЛ-1Н-ПИРАЗОЛО[3,4-b]ПИРИДИН-4-КАРБОКСИЛАТЫ И МЕТИЛ 3-МЕТИЛ-5-[2-(4-АРИЛАМИНО)-2-ОКСОАЦЕТИЛ]-6-СТИРИЛ-1-ФЕНИЛ-1Н-ПИРАЗОЛО[3,4-b]ПИРИДИН-4-КАРБОКСИЛАТЫ И СПОСОБ ИХ ПОЛУЧЕНИЯ |
| TWI785101B (zh) * | 2017-08-23 | 2022-12-01 | 瑞典商斯普林特生物科技公司 | 氮雜吲哚基吡啶酮及二氮雜吲哚基吡啶酮化合物 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3403158A (en) * | 1966-03-11 | 1968-09-24 | Upjohn Co | 1h-pyrazolo[3, 4-b]pyridines |
| US3681368A (en) * | 1970-10-15 | 1972-08-01 | Abbott Lab | Pyrazolo naphthridines |
| BE787249A (fr) * | 1971-08-05 | 1973-02-05 | Squibb & Sons Inc | Derives amino d'acides pyrazolopyridine carboxyliques, leurs esters et les sels de ces composes, ainsi que leurs procedes de preparation |
| US3891630A (en) * | 1974-03-04 | 1975-06-24 | Abbott Lab | Substituted pyrazolo{8 3,4-e{9 {8 1,4{9 thiazepines and isoxazolo{8 5,4-e{9 {8 1,4{9 thiazepines |
| US3903096A (en) * | 1974-03-29 | 1975-09-02 | Squibb & Sons Inc | New derivatives of sulfonyl-, sulfinyl- and sulfenyl-1H-pyrazolo {8 3,4-b{9 -pyridines |
| EP0005745B1 (en) * | 1978-05-26 | 1982-07-14 | Gruppo Lepetit S.P.A. | Pyrazolo (3,4-c) and thiazolo (5,4-c) isoquinolines, methods for preparing them, these compounds for use as antiinflammatory, cns-depressant and anti-anxiety agents and pharmaceutical compositions thereof |
-
1982
- 1982-09-22 IT IT23375/82A patent/IT1154024B/it active
-
1983
- 1983-09-05 GR GR72382A patent/GR78987B/el unknown
- 1983-09-10 EP EP83108942A patent/EP0104522B1/en not_active Expired - Lifetime
- 1983-09-10 DE DE8383108942T patent/DE3382299D1/de not_active Expired - Fee Related
- 1983-09-10 AT AT83108942T patent/ATE63913T1/de not_active IP Right Cessation
- 1983-09-19 US US06/533,909 patent/US4612318A/en not_active Expired - Fee Related
- 1983-09-21 CA CA000437174A patent/CA1248532A/en not_active Expired
- 1983-09-21 ES ES83525786A patent/ES525786A0/es active Granted
- 1983-09-21 PT PT77370A patent/PT77370B/pt not_active IP Right Cessation
- 1983-09-22 JP JP58176193A patent/JPS5989679A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| PT77370A (en) | 1983-10-01 |
| PT77370B (en) | 1986-04-21 |
| ATE63913T1 (de) | 1991-06-15 |
| EP0104522A2 (en) | 1984-04-04 |
| ES8503685A1 (es) | 1985-03-01 |
| EP0104522B1 (en) | 1991-05-29 |
| US4612318A (en) | 1986-09-16 |
| ES525786A0 (es) | 1985-03-01 |
| IT8223375A0 (it) | 1982-09-22 |
| CA1248532A (en) | 1989-01-10 |
| DE3382299D1 (de) | 1991-07-04 |
| JPS5989679A (ja) | 1984-05-23 |
| EP0104522A3 (en) | 1985-06-19 |
| IT1154024B (it) | 1987-01-21 |
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