GR3034458T3 - A specific crystalline form of zilpaterol hydrochloride, process for its preparation and intermediates used - Google Patents

A specific crystalline form of zilpaterol hydrochloride, process for its preparation and intermediates used

Info

Publication number
GR3034458T3
GR3034458T3 GR20000402058T GR20000402058T GR3034458T3 GR 3034458 T3 GR3034458 T3 GR 3034458T3 GR 20000402058 T GR20000402058 T GR 20000402058T GR 20000402058 T GR20000402058 T GR 20000402058T GR 3034458 T3 GR3034458 T3 GR 3034458T3
Authority
GR
Greece
Prior art keywords
trihydrate
soln
degrees
water
satd
Prior art date
Application number
GR20000402058T
Other languages
Greek (el)
English (en)
Inventor
Yves Chevremont
Jean-Yves Godard
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of GR3034458T3 publication Critical patent/GR3034458T3/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23K—FODDER
    • A23K20/00—Accessory food factors for animal feeding-stuffs
    • A23K20/10—Organic substances
    • A23K20/116—Heterocyclic compounds
    • A23K20/137—Heterocyclic compounds containing two hetero atoms, of which at least one is nitrogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S426/00—Food or edible material: processes, compositions, and products
    • Y10S426/807—Poultry or ruminant feed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Polymers & Plastics (AREA)
  • Food Science & Technology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Zoology (AREA)
  • Animal Husbandry (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Fodder In General (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Saccharide Compounds (AREA)
GR20000402058T 1995-06-13 2000-09-21 A specific crystalline form of zilpaterol hydrochloride, process for its preparation and intermediates used GR3034458T3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9506966A FR2735474B1 (fr) 1995-06-13 1995-06-13 Chlorhydrate de zilpaterol sous une forme cristallisee particuliere, son procede de preparation et les produits intermediaires mis en oeuvre

Publications (1)

Publication Number Publication Date
GR3034458T3 true GR3034458T3 (en) 2000-12-29

Family

ID=9479897

Family Applications (1)

Application Number Title Priority Date Filing Date
GR20000402058T GR3034458T3 (en) 1995-06-13 2000-09-21 A specific crystalline form of zilpaterol hydrochloride, process for its preparation and intermediates used

Country Status (21)

Country Link
US (2) US5731028A (enExample)
EP (1) EP0753518B1 (enExample)
JP (1) JP4249273B2 (enExample)
KR (1) KR100395204B1 (enExample)
CN (2) CN1164591C (enExample)
AT (1) ATE196471T1 (enExample)
AU (1) AU701653B2 (enExample)
BR (1) BR9602788A (enExample)
CA (1) CA2178783C (enExample)
DE (1) DE69610374T2 (enExample)
DK (1) DK0753518T3 (enExample)
EA (1) EA000011B1 (enExample)
ES (1) ES2151999T3 (enExample)
FR (1) FR2735474B1 (enExample)
GR (1) GR3034458T3 (enExample)
HU (1) HU220461B1 (enExample)
IN (1) IN2014DE02233A (enExample)
MX (1) MX9602307A (enExample)
PT (1) PT753518E (enExample)
UA (1) UA48941C2 (enExample)
ZA (1) ZA964977B (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4956308A (en) * 1987-01-20 1990-09-11 Itt Corporation Method of making self-aligned field-effect transistor
KR100344157B1 (ko) * 2000-01-06 2002-07-31 주식회사 하이테크 그라스 배경무늬 형성을 위한 장식판 도포제재 및 장식판의배경무늬 형성방법
US7207289B2 (en) * 2004-05-20 2007-04-24 Intervet International B.V. Method of feeding the cattle with feed additives that increases beef production and reduces liver abscess
RU2433131C2 (ru) 2007-02-01 2011-11-10 Интервет Интернэшнл Б.В. ЭНАНТИОСЕЛЕКТИВНЫЙ СИНТЕЗ 6-АМИНО-7-ГИДРОКСИ-4,5,6,7-ТЕТРАГИДРОИМИДАЗО[4,5,1-jk][1]БЕНЗАЗЕПИН-2[1H]-ОНА И ЗИЛПАТЕРОЛА
US8362006B2 (en) * 2007-03-31 2013-01-29 Intervet International B.V. Processes for making zilpaterol and salts thereof
CN105037275B (zh) 2007-03-31 2019-05-10 英特威国际有限公司 制备齐帕特罗及其盐的方法
JP5856990B2 (ja) * 2007-03-31 2016-02-10 インターベット インターナショナル ベー． フェー． ジルパテロールおよびこの塩の製造方法
MX2010006223A (es) 2007-12-06 2010-08-10 Intervet Int Bv Terapias de combinacion usando acetato de melengestrol y zilpaterol o sus sales.
TW201033217A (en) * 2008-12-17 2010-09-16 Intervet Int Bv Process for making a crystalline zilpaterol salt
BR112014028449A2 (pt) 2012-05-18 2017-06-27 Intervet Int Bv método para intensificar o desempenho de frangos de corte.
AU2013363731B2 (en) 2012-12-18 2018-04-19 Intervet International B.V. An improved process for making zilpaterol
BR112015022345A2 (pt) 2013-03-15 2017-07-18 Intervet Int Bv método para aumentar a eficiência de produção de carne bovina, composição para alimento de gado bovino, artigo medicinal, alimento medicinal, e, alimento de componente medicinal
US9364483B2 (en) 2014-06-20 2016-06-14 Laboratorios Virbac Pre-mix composition for cattle
CN105334323A (zh) * 2014-08-07 2016-02-17 暨南大学 一种检测齐帕特罗的方法和试纸条及其应用
MX2018000862A (es) * 2015-07-21 2018-05-15 Intervet Int Bv Una novedosa formulacion de premezcla animal de zilpaterol.
EP3488705A1 (en) 2017-11-23 2019-05-29 Saviela AG Solubilized growth promoting product to be applied orally to animals and method for the respective feed preparation

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2534257A1 (fr) * 1982-10-12 1984-04-13 Roussel Uclaf Nouveaux derives de la 6-amino 7-hydroxy 4,5,6,7-tetrahydro-imidazo/4,5,1-j-k/ /1/ benzazepin-2(1h)-one, leurs sels, application a titre de medicaments, compositions les renfermant et un intermediaire
US4497779A (en) * 1983-10-14 1985-02-05 Amax Inc. Production of potassium hexafluotitanates using dilute hydrofluoric acid
IE60588B1 (en) * 1986-07-30 1994-07-27 Sumitomo Pharma Carbapenem compound in crystalline form, and its production and use
IE60964B1 (en) * 1986-12-11 1994-09-07 Roussel Uclaf Zootechnical compositions containing a beta-adrenergic
FR2608046B1 (fr) * 1986-12-11 1989-03-31 Roussel Uclaf Compositions zootechniques renfermant un derive de la 6-amino 7-hydroxy 4,5,6,7-tetrahydroimidazo /4,5, 1-j-k/ /1/benzazepin-2-(1h)-one
US5015639A (en) * 1987-03-27 1991-05-14 Schering Corporation Substituted benzazepines, their preparation and pharmaceutical compositions containing them
FR2647310B1 (fr) * 1989-05-29 1992-01-17 Roussel Uclaf Utilisation de beta-adrenergiques pour la fabrication de compositions zootechniques
WO1994013680A1 (en) * 1992-12-04 1994-06-23 Janssen Pharmaceutica N.V. ANTIALLERGIC IMIDAZO[1,2-a](PYRROLO, THIENO OR FURANO)[2,3-d]AZEPINE DERIVATIVES

Also Published As

Publication number Publication date
EA199600027A2 (ru) 1996-12-30
FR2735474A1 (fr) 1996-12-20
UA48941C2 (uk) 2002-09-16
CA2178783C (fr) 2005-04-12
FR2735474B1 (fr) 1997-08-08
DE69610374T2 (de) 2001-01-25
US5847124A (en) 1998-12-08
MX9602307A (es) 1998-04-30
EA000011B1 (ru) 1997-12-30
CN1164591C (zh) 2004-09-01
CN1147902A (zh) 1997-04-23
CA2178783A1 (fr) 1996-12-14
US5731028A (en) 1998-03-24
HU9601617D0 (en) 1996-08-28
IN2014DE02233A (enExample) 2015-06-19
DK0753518T3 (da) 2001-01-29
KR100395204B1 (ko) 2003-11-17
EA199600027A3 (ru) 1997-03-31
ZA964977B (en) 1997-06-12
HUP9601617A2 (en) 1997-06-30
JPH093069A (ja) 1997-01-07
AU5592596A (en) 1997-01-02
HUP9601617A3 (en) 1999-07-28
JP4249273B2 (ja) 2009-04-02
DE69610374D1 (de) 2000-10-26
EP0753518B1 (fr) 2000-09-20
ATE196471T1 (de) 2000-10-15
PT753518E (pt) 2000-12-29
ES2151999T3 (es) 2001-01-16
CN1083244C (zh) 2002-04-24
HU220461B1 (hu) 2002-02-28
KR970001215A (ko) 1997-01-21
AU701653B2 (en) 1999-02-04
BR9602788A (pt) 1998-09-08
EP0753518A1 (fr) 1997-01-15
CN1396165A (zh) 2003-02-12

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