GB2040291A - Trifluoromethylated dipeptides - Google Patents

Trifluoromethylated dipeptides Download PDF

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Publication number
GB2040291A
GB2040291A GB7944621A GB7944621A GB2040291A GB 2040291 A GB2040291 A GB 2040291A GB 7944621 A GB7944621 A GB 7944621A GB 7944621 A GB7944621 A GB 7944621A GB 2040291 A GB2040291 A GB 2040291A
Authority
GB
United Kingdom
Prior art keywords
formula
compounds
ala
assumes
leu
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
GB7944621A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Delalande SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR7901410A external-priority patent/FR2416883A2/fr
Application filed by Delalande SA filed Critical Delalande SA
Publication of GB2040291A publication Critical patent/GB2040291A/en
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
GB7944621A 1979-01-19 1979-12-31 Trifluoromethylated dipeptides Withdrawn GB2040291A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7901410A FR2416883A2 (fr) 1977-02-18 1979-01-19 Nouveaux oligopeptides trifluoromethyles, leur procede de preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
GB2040291A true GB2040291A (en) 1980-08-28

Family

ID=9220984

Family Applications (1)

Application Number Title Priority Date Filing Date
GB7944621A Withdrawn GB2040291A (en) 1979-01-19 1979-12-31 Trifluoromethylated dipeptides

Country Status (8)

Country Link
JP (1) JPS55100347A (es)
AU (1) AU5474980A (es)
ES (1) ES487622A0 (es)
GB (1) GB2040291A (es)
GR (1) GR73130B (es)
IT (1) IT1149281B (es)
NL (1) NL8000345A (es)
ZA (1) ZA8079B (es)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4499082A (en) * 1983-12-05 1985-02-12 E. I. Du Pont De Nemours And Company α-Aminoboronic acid peptides
EP0168769A2 (en) * 1984-07-16 1986-01-22 Merck & Co. Inc. Process for preparing carboxyalkyl dipeptides
US5693617A (en) * 1994-03-15 1997-12-02 Proscript, Inc. Inhibitors of the 26s proteolytic complex and the 20s proteasome contained therein
CN113861240A (zh) * 2021-10-20 2021-12-31 中国科学院大学 一种三氟甲基试剂及其合成方法与应用

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4499082A (en) * 1983-12-05 1985-02-12 E. I. Du Pont De Nemours And Company α-Aminoboronic acid peptides
EP0168769A2 (en) * 1984-07-16 1986-01-22 Merck & Co. Inc. Process for preparing carboxyalkyl dipeptides
EP0168769A3 (en) * 1984-07-16 1989-02-08 Merck & Co. Inc. Process for preparing carboxyalkyl dipeptides
US5693617A (en) * 1994-03-15 1997-12-02 Proscript, Inc. Inhibitors of the 26s proteolytic complex and the 20s proteasome contained therein
CN113861240A (zh) * 2021-10-20 2021-12-31 中国科学院大学 一种三氟甲基试剂及其合成方法与应用
CN113861240B (zh) * 2021-10-20 2023-10-31 中国科学院大学 一种三氟甲基试剂及其合成方法与应用

Also Published As

Publication number Publication date
GR73130B (es) 1984-02-07
NL8000345A (nl) 1980-07-22
ZA8079B (en) 1981-01-28
ES8202786A1 (es) 1980-12-16
JPS55100347A (en) 1980-07-31
IT8019070A0 (it) 1980-01-08
ES487622A0 (es) 1980-12-16
AU5474980A (en) 1980-07-24
IT1149281B (it) 1986-12-03

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Legal Events

Date Code Title Description
WAP Application withdrawn, taken to be withdrawn or refused ** after publication under section 16(1)