GB1570374A - Indoles - Google Patents

Indoles Download PDF

Info

Publication number
GB1570374A
GB1570374A GB902078A GB902078A GB1570374A GB 1570374 A GB1570374 A GB 1570374A GB 902078 A GB902078 A GB 902078A GB 902078 A GB902078 A GB 902078A GB 1570374 A GB1570374 A GB 1570374A
Authority
GB
United Kingdom
Prior art keywords
indole
indoles
acetyl
piperazino
piperonylpiperazino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB902078A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SAUBA LAB
Original Assignee
SAUBA LAB
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SAUBA LAB filed Critical SAUBA LAB
Publication of GB1570374A publication Critical patent/GB1570374A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/40—Nitrogen atoms, not forming part of a nitro radical, e.g. isatin semicarbazone

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
GB902078A 1977-03-17 1978-03-07 Indoles Expired GB1570374A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7707993A FR2421900A1 (fr) 1977-03-17 1977-03-17 Piperazino-3-indoles, leur procede de preparation et leurs applications therapeutiques

Publications (1)

Publication Number Publication Date
GB1570374A true GB1570374A (en) 1980-07-02

Family

ID=9188218

Family Applications (1)

Application Number Title Priority Date Filing Date
GB902078A Expired GB1570374A (en) 1977-03-17 1978-03-07 Indoles

Country Status (4)

Country Link
DE (1) DE2811031C2 (de)
ES (1) ES467954A1 (de)
FR (1) FR2421900A1 (de)
GB (1) GB1570374A (de)

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4382935A (en) 1980-02-14 1983-05-10 Andre Buzas Analgesic drug containing a derivative of benzylpiperazine
EP0200322B1 (de) * 1985-04-10 1990-02-28 H. Lundbeck A/S Heterocyclische Verbindungen
US5532372A (en) * 1990-07-06 1996-07-02 Sumitomo Pharmaceuticals Company, Ltd. Imide derivatives, and their production and use
WO2004106346A1 (en) * 2003-05-30 2004-12-09 Janssen Pharmaceutica N.V. Indole derivatives with an improved antipsychotic activity
JP2010507621A (ja) * 2006-10-27 2010-03-11 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規な置換ピペリジル−プロパン−チオール
JP2010507620A (ja) * 2006-10-27 2010-03-11 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ピペリジル−プロパン−チオールｃｃｒ３モジュレーター
JP2010521438A (ja) * 2007-03-15 2010-06-24 ノバルティス アーゲー 有機化合物およびその使用
US9409871B2 (en) 2008-07-18 2016-08-09 Novartis Ag Pyridazinyl derivatives as SMO inhibitors

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2524884A1 (fr) * 1982-04-07 1983-10-14 Delalande Sa Nouvelles piperazines substituees par un groupe heterocyclique du type benzotriazolyle ou indolyle, leur procede de preparation et leur application en therapeutique
DK181190D0 (da) * 1990-07-30 1990-07-30 Lundbeck & Co As H 3-aryl-indol- eller 3-aryl-indazolderivater
US5643784A (en) * 1990-12-04 1997-07-01 H, Lundbeck A/S Indan derivatives
NZ243065A (en) * 1991-06-13 1995-07-26 Lundbeck & Co As H Piperidine derivatives and pharmaceutical compositions
ES2063700B1 (es) * 1993-04-28 1995-07-16 Vita Invest Sa Agente activo sobre el sistema nervioso central, proceso para su preparacion y composiciones farmaceuticas que lo contengan.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1135461B (de) * 1959-05-08 1962-08-30 Knoll Ag Verfahren zur Herstellung von basisch substituierten Phthalimidinen
NL133995C (de) * 1965-08-21
DE2138865A1 (de) * 1970-08-15 1973-02-22 Sumitomo Chemical Co 3-indolylpiperazine, verfahren zu ihrer herstellung und arzneimittel
US3751416A (en) * 1971-05-27 1973-08-07 American Cyanamid Co 3-(2-(4-phenyl-1-piperazinyl)-ethyl)indolines
FR2140260B1 (de) * 1971-06-07 1974-08-30 Delalande Sa
BE790679A (fr) * 1971-11-03 1973-04-27 Ici Ltd Derives de l'indole
FR2191895B1 (de) * 1972-07-17 1975-10-17 Bellon Labor Sa Roger

Cited By (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4382935A (en) 1980-02-14 1983-05-10 Andre Buzas Analgesic drug containing a derivative of benzylpiperazine
EP0200322B1 (de) * 1985-04-10 1990-02-28 H. Lundbeck A/S Heterocyclische Verbindungen
USRE34299E (en) * 1985-04-10 1993-06-29 H. Lundbeck A/S 1-(4'-fluorophenyl)-3,5-substituted indoles useful in the treatment of psychic disorders and pharmaceutical compositions thereof
US5780632A (en) * 1990-06-07 1998-07-14 Sumitomo Pharmaceuticals Company, Limited Imide derivatives and their production and use
US5532372A (en) * 1990-07-06 1996-07-02 Sumitomo Pharmaceuticals Company, Ltd. Imide derivatives, and their production and use
WO2004106346A1 (en) * 2003-05-30 2004-12-09 Janssen Pharmaceutica N.V. Indole derivatives with an improved antipsychotic activity
WO2004106298A1 (en) * 2003-05-30 2004-12-09 Janssen Pharmaceutica N.V. Indole derivatives with an improved antipsychotic activity
JP2010507621A (ja) * 2006-10-27 2010-03-11 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規な置換ピペリジル−プロパン−チオール
JP2010507620A (ja) * 2006-10-27 2010-03-11 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ピペリジル−プロパン−チオールｃｃｒ３モジュレーター
JP2010521438A (ja) * 2007-03-15 2010-06-24 ノバルティス アーゲー 有機化合物およびその使用
US9409871B2 (en) 2008-07-18 2016-08-09 Novartis Ag Pyridazinyl derivatives as SMO inhibitors

Also Published As

Publication number Publication date
DE2811031A1 (de) 1978-09-21
DE2811031C2 (de) 1984-11-29
FR2421900A1 (fr) 1979-11-02
ES467954A1 (es) 1978-11-01
FR2421900B1 (de) 1980-10-10

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Legal Events

Date Code Title Description
PS Patent sealed
PCNP Patent ceased through non-payment of renewal fee