GB1471235A - Amoxycillin derivatives - Google Patents
Amoxycillin derivativesInfo
- Publication number
- GB1471235A GB1471235A GB4066174A GB4066174A GB1471235A GB 1471235 A GB1471235 A GB 1471235A GB 4066174 A GB4066174 A GB 4066174A GB 4066174 A GB4066174 A GB 4066174A GB 1471235 A GB1471235 A GB 1471235A
- Authority
- GB
- United Kingdom
- Prior art keywords
- compounds
- amoxycillin
- sept
- prepared
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- LSQZJLSUYDQPKJ-NJBDSQKTSA-N amoxicillin Chemical class C1([C@@H](N)C(=O)N[C@H]2[C@H]3SC([C@@H](N3C2=O)C(O)=O)(C)C)=CC=C(O)C=C1 LSQZJLSUYDQPKJ-NJBDSQKTSA-N 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 3
- HTSGKJQDMSTCGS-UHFFFAOYSA-N 1,4-bis(4-chlorophenyl)-2-(4-methylphenyl)sulfonylbutane-1,4-dione Chemical compound C1=CC(C)=CC=C1S(=O)(=O)C(C(=O)C=1C=CC(Cl)=CC=1)CC(=O)C1=CC=C(Cl)C=C1 HTSGKJQDMSTCGS-UHFFFAOYSA-N 0.000 abstract 1
- QGZKDVFQNNGYKY-UHFFFAOYSA-O Ammonium Chemical class [NH4+] QGZKDVFQNNGYKY-UHFFFAOYSA-O 0.000 abstract 1
- BVKZGUZCCUSVTD-UHFFFAOYSA-M Bicarbonate Chemical compound OC([O-])=O BVKZGUZCCUSVTD-UHFFFAOYSA-M 0.000 abstract 1
- BVKZGUZCCUSVTD-UHFFFAOYSA-L Carbonate Chemical compound [O-]C([O-])=O BVKZGUZCCUSVTD-UHFFFAOYSA-L 0.000 abstract 1
- 229960003022 amoxicillin Drugs 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 239000012736 aqueous medium Substances 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 238000007327 hydrogenolysis reaction Methods 0.000 abstract 1
- 230000007062 hydrolysis Effects 0.000 abstract 1
- 238000006460 hydrolysis reaction Methods 0.000 abstract 1
- 150000002500 ions Chemical class 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- LSQZJLSUYDQPKJ-UHFFFAOYSA-N p-Hydroxyampicillin Natural products O=C1N2C(C(O)=O)C(C)(C)SC2C1NC(=O)C(N)C1=CC=C(O)C=C1 LSQZJLSUYDQPKJ-UHFFFAOYSA-N 0.000 abstract 1
- 125000006239 protecting group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
- A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Priority Applications (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB4066174A GB1471235A (en) | 1974-09-18 | 1974-09-18 | Amoxycillin derivatives |
| US05/611,199 US3980639A (en) | 1974-09-18 | 1975-09-08 | Amoxicillin derivatives |
| BE159884A BE833237A (fr) | 1974-09-18 | 1975-09-09 | Penicillines |
| FR7527707A FR2285127A1 (fr) | 1974-09-18 | 1975-09-10 | Penicillines |
| DE19752540523 DE2540523A1 (de) | 1974-09-18 | 1975-09-11 | Derivate von amoxycillin, verfahren zu ihrer herstellung und diese derivate enthaltende arzneimittel |
| JP50112483A JPS5159892A (enExample) | 1974-09-18 | 1975-09-17 | |
| US05/664,083 US4024244A (en) | 1974-09-18 | 1976-03-05 | Amoxicillin derivatives |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB4066174A GB1471235A (en) | 1974-09-18 | 1974-09-18 | Amoxycillin derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1471235A true GB1471235A (en) | 1977-04-21 |
Family
ID=10416004
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB4066174A Expired GB1471235A (en) | 1974-09-18 | 1974-09-18 | Amoxycillin derivatives |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US3980639A (enExample) |
| JP (1) | JPS5159892A (enExample) |
| BE (1) | BE833237A (enExample) |
| DE (1) | DE2540523A1 (enExample) |
| FR (1) | FR2285127A1 (enExample) |
| GB (1) | GB1471235A (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1576731A (en) * | 1976-08-10 | 1980-10-15 | Beecham Group Ltd | Process for the preparation of sodium amoxycillin |
| DE2737673A1 (de) * | 1977-08-20 | 1979-02-22 | Bayer Ag | Synergistische kombinationen von penicillinen |
| FR2503710B1 (fr) * | 1981-04-10 | 1985-07-05 | Bristol Myers Co | Procede de production du sel de sodium de l'amoxicilline |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3654265A (en) * | 1970-11-27 | 1972-04-04 | Bristol Myers Co | Synthetic penicillin |
| GB1380741A (en) * | 1971-02-05 | 1975-01-15 | Squibb & Sons Inc | Antibiotic compositions and their preparation |
| BE786924A (fr) * | 1971-07-28 | 1973-01-29 | Squibb & Sons Inc | Antibiotiques, leur preparation et leurs utilisations therapeutiques |
-
1974
- 1974-09-18 GB GB4066174A patent/GB1471235A/en not_active Expired
-
1975
- 1975-09-08 US US05/611,199 patent/US3980639A/en not_active Expired - Lifetime
- 1975-09-09 BE BE159884A patent/BE833237A/xx not_active IP Right Cessation
- 1975-09-10 FR FR7527707A patent/FR2285127A1/fr active Granted
- 1975-09-11 DE DE19752540523 patent/DE2540523A1/de not_active Withdrawn
- 1975-09-17 JP JP50112483A patent/JPS5159892A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| DE2540523A1 (de) | 1976-04-08 |
| FR2285127A1 (fr) | 1976-04-16 |
| US3980639A (en) | 1976-09-14 |
| BE833237A (fr) | 1976-03-09 |
| FR2285127B1 (enExample) | 1979-09-14 |
| JPS5159892A (enExample) | 1976-05-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed [section 19, patents act 1949] | ||
| PCNP | Patent ceased through non-payment of renewal fee |