GB1324755A - 1,4-benzothiazepines - Google Patents
1,4-benzothiazepinesInfo
- Publication number
- GB1324755A GB1324755A GB295072A GB295072A GB1324755A GB 1324755 A GB1324755 A GB 1324755A GB 295072 A GB295072 A GB 295072A GB 295072 A GB295072 A GB 295072A GB 1324755 A GB1324755 A GB 1324755A
- Authority
- GB
- United Kingdom
- Prior art keywords
- substituted
- alkyl
- radicals
- optionally substituted
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D281/02—Seven-membered rings
- C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
1324755 Benzothiazepines WARNERLAMBERT CO 21 Jan 1972 [22 Jan 1971] 2950/72 Heading C2C Compounds of the general Formula I (A = H, Ph, substituted Ph; B = OR 1 , NR 2 R 3 ; R 1 = C 1-6 alkyl optionally substituted by alkoxy, PhO or Ph radicals, cycloalkyl, Ph, substituted Ph; R 2,3 = H, OH, C 1-5 alkyl optionally substituted by NH 2 , alkylamino, dialkylamino, polymethyleneimino (the carbon chain of which can be interrupted by a heteroatom) or Ph radicals, Ph, substituted Ph, NH 2 optionally substituted by C 1-6 alkyl, alkylidene, carboxyalkylidene, acyl or aryl radicals, cyclic amino or NR 2 R 3 = unsubstituted or substituted, saturated 5-6 membered ring; or A and B, together with atoms 3 and 4 of the benzothiazepine ring, form a 5-7 membered ring) and their acid addition salts and quaternary ammonium compounds are prepared as follows: (R 4 = H, C 1-6 alkyl; Hal = halogen; X = anion), optionally followed by conversion to an acid addition salt or quaternary ammonium compound. These compounds possess anti-inflammatory activity, and may be administered in the form of pharmaceutical preparations containing them in association with a carrier.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE2103015 | 1971-01-22 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1324755A true GB1324755A (en) | 1973-07-25 |
Family
ID=5796657
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB295072A Expired GB1324755A (en) | 1971-01-22 | 1972-01-21 | 1,4-benzothiazepines |
Country Status (5)
| Country | Link |
|---|---|
| AU (1) | AU3810972A (en) |
| BE (1) | BE778335A (en) |
| ES (1) | ES399082A1 (en) |
| FR (1) | FR2122574A1 (en) |
| GB (1) | GB1324755A (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1986000618A1 (en) * | 1984-07-13 | 1986-01-30 | Takeda Chemical Industries, Ltd. | Condensed 7-membered ring compounds and process for their preparation |
-
1972
- 1972-01-20 AU AU38109/72A patent/AU3810972A/en not_active Expired
- 1972-01-21 GB GB295072A patent/GB1324755A/en not_active Expired
- 1972-01-21 ES ES399082A patent/ES399082A1/en not_active Expired
- 1972-01-21 FR FR7202008A patent/FR2122574A1/fr not_active Withdrawn
- 1972-01-21 BE BE778335A patent/BE778335A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BE778335A (en) | 1972-07-24 |
| AU3810972A (en) | 1973-07-26 |
| FR2122574A1 (en) | 1972-09-01 |
| ES399082A1 (en) | 1974-11-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| CSNS | Application of which complete specification have been accepted and published, but patent is not sealed |