GB1234058A - - Google Patents

Info

Publication number
GB1234058A
GB1234058A GB1234058DA GB1234058A GB 1234058 A GB1234058 A GB 1234058A GB 1234058D A GB1234058D A GB 1234058DA GB 1234058 A GB1234058 A GB 1234058A
Authority
GB
United Kingdom
Prior art keywords
group
atom
quaternary ammonium
reaction
general formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GB1234058A publication Critical patent/GB1234058A/en
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
GB1234058D 1968-10-21 1968-10-21 Expired GB1234058A (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4979868 1968-10-21

Publications (1)

Publication Number Publication Date
GB1234058A true GB1234058A (ja) 1971-06-03

Family

ID=10453571

Family Applications (1)

Application Number Title Priority Date Filing Date
GB1234058D Expired GB1234058A (ja) 1968-10-21 1968-10-21

Country Status (4)

Country Link
DE (1) DE1804450A1 (ja)
FR (1) FR1593614A (ja)
GB (1) GB1234058A (ja)
NL (1) NL6815409A (ja)

Cited By (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4182766A (en) * 1977-09-19 1980-01-08 Hoffmann-La Roche Inc. Naphth[2,3-d]imidazoles
WO1987005296A1 (en) * 1986-03-07 1987-09-11 Pfizer Inc. 2-[(2-pyridyl)methylsulfinyl]thienoimidazoles and related compounds as antiulcer agents
EP0254588A1 (en) * 1986-07-25 1988-01-27 Tokyo Tanabe Company Limited Imidazo[4,5-b] pyridine compounds, process for preparing same and pharmaceutical compositions containing same
US4738974A (en) * 1983-03-04 1988-04-19 Aktiebolaget Hassle Base addition salts of omeprazole
US4738970A (en) * 1984-12-18 1988-04-19 Otsuka Pharmaceutical Co., Ltd. Benzimidazolyl-thio-tetrahydroquinolines and anti-peptic ulcer compositions containing the same
US4758579A (en) * 1984-06-16 1988-07-19 Byk Gulden Lomberg Chemische Fabrik Gmbh Fluoroalkoxy substituted benzimidazoles useful as gastric acid secretion inhibitors
US4791114A (en) * 1986-01-20 1988-12-13 501 Laboratorios Del, Dr. Esteve 2-Benzimidazolylalkylthio (or -sulfinyl or -sulfonyl) derivatives, their preparation and their application as medicinal products
GB2161160B (en) * 1984-07-06 1989-05-24 Fisons Plc Heterocyclic sulphinyl compounds
US4873337A (en) * 1985-07-31 1989-10-10 The Upjohn Company N-substituted derivatives of 2-(pyridylalkenesulfinyl) benzimidazoles as gastric antisecretory agents
US5053417A (en) * 1986-02-12 1991-10-01 Tanabe Seiyaku Co., Ltd. Imidazole derivatives and preparation thereof
US5114955A (en) * 1987-11-13 1992-05-19 Hoechst Aketiengesellschaft Substituted thienoimidazole derivatives
US5389664A (en) * 1992-07-08 1995-02-14 Monsanto Company Alleviating stomach ulcers in swine
JP2679745B2 (ja) 1989-06-29 1997-11-19 明治製菓株式会社 アゾール誘導体及びそれらを有効成分とする抗潰瘍剤
US5703097A (en) * 1994-02-28 1997-12-30 Il-Yang Pharm. Co., Ltd. 5-pyrrolyl-2-pyridylmethylsulfinyl benzimidazole derivatives
US5859030A (en) * 1994-06-10 1999-01-12 Byk Gulden Lomberg Chemische Fabrik Gmbh Substituted arylalkylthioalkylthiopyridines for use in the control of helicobacter bacteria
US6077541A (en) * 1997-11-14 2000-06-20 Andrx Pharmaceuticals, Inc. Omeprazole formulation
US6174548B1 (en) 1998-08-28 2001-01-16 Andrx Pharmaceuticals, Inc. Omeprazole formulation
US6733778B1 (en) 1999-08-27 2004-05-11 Andrx Pharmaceuticals, Inc. Omeprazole formulation
EP3050565A1 (en) * 2015-01-27 2016-08-03 Ecole Polytechnique Fédérale de Lausanne (EPFL) Benzimidazole sulfide derivatives for the treatment or prevention of tuberculosis

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1259525B (de) * 1961-11-21 1968-01-25 Bauermann & Soehne G M B H W Befestigungsvorrichtung fuer ein einstellbares Schutzdach an einer Sitz- bzw. Liegeschaukel
SE418966B (sv) * 1974-02-18 1981-07-06 Haessle Ab Analogiforfarande for framstellning av foreningar med magsyrasekretionsinhiberande verkan
US4045564A (en) * 1974-02-18 1977-08-30 Ab Hassle Benzimidazole derivatives useful as gastric acid secretion inhibitors
SE416649B (sv) * 1974-05-16 1981-01-26 Haessle Ab Forfarande for framstellning av foreningar som paverkar magsyrasekretionen
SE7804231L (sv) * 1978-04-14 1979-10-15 Haessle Ab Magsyrasekretionsmedel
DE3216843C2 (de) * 1982-05-05 1986-10-23 Ludwig Heumann & Co GmbH, 8500 Nürnberg 3-Thiomethyl-pyridin-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
CA1260474A (en) * 1984-12-03 1989-09-26 Raymond A. Stokbroekx Benzoxazol- and benzothiazolamine derivatives
SE8500996D0 (sv) * 1985-03-01 1985-03-01 Haessle Ab Method of treatment
DK399389A (da) * 1988-08-18 1990-02-19 Takeda Chemical Industries Ltd Injicerbare oploesninger

Cited By (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4182766A (en) * 1977-09-19 1980-01-08 Hoffmann-La Roche Inc. Naphth[2,3-d]imidazoles
US4248880A (en) 1977-09-19 1981-02-03 Hoffmann-La Roche Inc. Treatment of gastric ulcers with naphthimidazole derivatives
US4738974A (en) * 1983-03-04 1988-04-19 Aktiebolaget Hassle Base addition salts of omeprazole
US4758579A (en) * 1984-06-16 1988-07-19 Byk Gulden Lomberg Chemische Fabrik Gmbh Fluoroalkoxy substituted benzimidazoles useful as gastric acid secretion inhibitors
GB2161160B (en) * 1984-07-06 1989-05-24 Fisons Plc Heterocyclic sulphinyl compounds
US4738970A (en) * 1984-12-18 1988-04-19 Otsuka Pharmaceutical Co., Ltd. Benzimidazolyl-thio-tetrahydroquinolines and anti-peptic ulcer compositions containing the same
US4880815A (en) * 1984-12-18 1989-11-14 Otsuka Pharmaceutical Co., Ltd. Imidazopyridyl-alkylthio-pyridines and anti-peptic ulcer compositions containing the same
US4873337A (en) * 1985-07-31 1989-10-10 The Upjohn Company N-substituted derivatives of 2-(pyridylalkenesulfinyl) benzimidazoles as gastric antisecretory agents
US4791114A (en) * 1986-01-20 1988-12-13 501 Laboratorios Del, Dr. Esteve 2-Benzimidazolylalkylthio (or -sulfinyl or -sulfonyl) derivatives, their preparation and their application as medicinal products
US5053417A (en) * 1986-02-12 1991-10-01 Tanabe Seiyaku Co., Ltd. Imidazole derivatives and preparation thereof
WO1987005296A1 (en) * 1986-03-07 1987-09-11 Pfizer Inc. 2-[(2-pyridyl)methylsulfinyl]thienoimidazoles and related compounds as antiulcer agents
EP0254588A1 (en) * 1986-07-25 1988-01-27 Tokyo Tanabe Company Limited Imidazo[4,5-b] pyridine compounds, process for preparing same and pharmaceutical compositions containing same
US5114955A (en) * 1987-11-13 1992-05-19 Hoechst Aketiengesellschaft Substituted thienoimidazole derivatives
JP2679745B2 (ja) 1989-06-29 1997-11-19 明治製菓株式会社 アゾール誘導体及びそれらを有効成分とする抗潰瘍剤
US5389664A (en) * 1992-07-08 1995-02-14 Monsanto Company Alleviating stomach ulcers in swine
US5703097A (en) * 1994-02-28 1997-12-30 Il-Yang Pharm. Co., Ltd. 5-pyrrolyl-2-pyridylmethylsulfinyl benzimidazole derivatives
US5859030A (en) * 1994-06-10 1999-01-12 Byk Gulden Lomberg Chemische Fabrik Gmbh Substituted arylalkylthioalkylthiopyridines for use in the control of helicobacter bacteria
US6077541A (en) * 1997-11-14 2000-06-20 Andrx Pharmaceuticals, Inc. Omeprazole formulation
US6780435B2 (en) 1997-11-14 2004-08-24 Andrx Pharmaceuticals, Inc. Omeprazole formulation
US6174548B1 (en) 1998-08-28 2001-01-16 Andrx Pharmaceuticals, Inc. Omeprazole formulation
US6855336B2 (en) 1998-08-28 2005-02-15 Andrx Pharmaceuticals, Inc. Omeprazole formulation
US6733778B1 (en) 1999-08-27 2004-05-11 Andrx Pharmaceuticals, Inc. Omeprazole formulation
EP3050565A1 (en) * 2015-01-27 2016-08-03 Ecole Polytechnique Fédérale de Lausanne (EPFL) Benzimidazole sulfide derivatives for the treatment or prevention of tuberculosis
WO2016120259A1 (en) * 2015-01-27 2016-08-04 Ecole Polytechnique Federale De Lausanne (Epfl) Benzimidazole sulfide derivatives for the treatment or prevention of tuberculosis
US10137116B2 (en) 2015-01-27 2018-11-27 École Polytechnique Fédérale De Lausanne (Epfl) Benzimidazole sulfide derivatives for the treatment or prevention of tuberculosis

Also Published As

Publication number Publication date
DE1804450A1 (de) 1970-05-27
NL6815409A (ja) 1970-05-04
FR1593614A (ja) 1970-06-01

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Legal Events

Date Code Title Description
PS Patent sealed
PLNP Patent lapsed through nonpayment of renewal fees