GB1112723A - Pyrazino[2,3-d][1,3]oxazin-4-one 8-oxides - Google Patents
Pyrazino[2,3-d][1,3]oxazin-4-one 8-oxidesInfo
- Publication number
- GB1112723A GB1112723A GB3179365D GB3179365D GB1112723A GB 1112723 A GB1112723 A GB 1112723A GB 3179365 D GB3179365 D GB 3179365D GB 3179365 D GB3179365 D GB 3179365D GB 1112723 A GB1112723 A GB 1112723A
- Authority
- GB
- United Kingdom
- Prior art keywords
- alkyl
- phenyl
- hydrogen
- pyrazino
- alkylsulphonyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D241/24—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D241/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with nitrogen atoms directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D475/00—Heterocyclic compounds containing pteridine ring systems
- C07D475/02—Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D475/00—Heterocyclic compounds containing pteridine ring systems
- C07D475/02—Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4
- C07D475/04—Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
1,112,723. Pyrazino-oxazines. MERCK & CO. Inc. 7 Sept., 1965 [8 July, 1965], No. 31793/67. Divided out of 1,112,721. Heading C2C. Novel compounds of the formula in which R<SP>5</SP> is a hydrogen atom or a C 1-5 alkyl or phenyl-substituted C 1-5 alkyl radical and X is a hydrogen, chlorine or bromine atom or a trifluoromethyl, C 1-5 alkyl, C 3-6 cycloalkyl, mononuclear aryl, C 1-5 alkoxy, C 1-5 alkylthio, phenyl-Bubstituted C 1-5 alkylthio, C 1-5 alkylsulphonyl, phenyl-substituted C 1-5 alkylsulphonyl or di-(C 1-5 alkyl) amino group, are prepared by heating a 3-amino-6-X-pyrazinoic acid 4-oxide with an organic acid anhydride of formula (R<SP>5</SP>CO) 2 O or, when R<SP>5</SP> is to be hydrogen, with a mixture of formic acid and acetic anhydride.
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US395046A US3249610A (en) | 1964-09-08 | 1964-09-08 | Synthesis of 3-amino, 5-chloro, 6-substituted-pyrazinoates |
| US426203A US3327287A (en) | 1965-01-18 | 1965-01-18 | Apparatus for converting lineal seismogram sections into an areally presented seismogram |
| US47035065A | 1965-07-08 | 1965-07-08 | |
| US47056365A | 1965-07-08 | 1965-07-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1112723A true GB1112723A (en) | 1968-05-08 |
Family
ID=27503371
Family Applications (5)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB3179365D Expired GB1112723A (en) | 1964-09-08 | 1965-09-07 | Pyrazino[2,3-d][1,3]oxazin-4-one 8-oxides |
| GB3816765A Expired GB1112722A (en) | 1964-09-08 | 1965-09-07 | Alkyl aminochloropyrazinoates |
| GB3816665A Expired GB1112721A (en) | 1964-09-08 | 1965-09-07 | 3-aminopyrazinoic acid n-oxide compounds and their derivatives |
| GB3179467A Expired GB1112724A (en) | 1964-09-08 | 1965-09-07 | Pteridine n-oxides |
| GB2907666A Expired GB1115406A (en) | 1964-09-08 | 1966-06-29 | 3(aminopyrazinoyl)guanidine 4-oxide derivatives and their preparation and use |
Family Applications After (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB3816765A Expired GB1112722A (en) | 1964-09-08 | 1965-09-07 | Alkyl aminochloropyrazinoates |
| GB3816665A Expired GB1112721A (en) | 1964-09-08 | 1965-09-07 | 3-aminopyrazinoic acid n-oxide compounds and their derivatives |
| GB3179467A Expired GB1112724A (en) | 1964-09-08 | 1965-09-07 | Pteridine n-oxides |
| GB2907666A Expired GB1115406A (en) | 1964-09-08 | 1966-06-29 | 3(aminopyrazinoyl)guanidine 4-oxide derivatives and their preparation and use |
Country Status (8)
| Country | Link |
|---|---|
| BE (2) | BE668496A (en) |
| BR (3) | BR6572769D0 (en) |
| CH (3) | CH466293A (en) |
| DE (3) | DE1595952A1 (en) |
| GB (5) | GB1112723A (en) |
| IL (3) | IL24098A (en) |
| NL (3) | NL6511644A (en) |
| SE (1) | SE329629B (en) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN113200985B (en) * | 2021-05-18 | 2022-09-09 | 南开大学 | Pteridinone compound and preparation method and application thereof |
| CN117946013B (en) * | 2024-01-25 | 2024-07-02 | 白银康寓信生物科技有限公司 | Method for synthesizing 5, 6-dihalogen-3-aminopyrazine-2-methyl formate by one-pot method |
-
1965
- 1965-08-06 IL IL2409865A patent/IL24098A/en unknown
- 1965-08-06 IL IL2409765A patent/IL24097A/en unknown
- 1965-08-06 IL IL3178765A patent/IL31787A/en unknown
- 1965-08-19 BE BE668496D patent/BE668496A/xx unknown
- 1965-08-19 BE BE668495D patent/BE668495A/xx unknown
- 1965-08-24 DE DE19651595952 patent/DE1595952A1/en active Pending
- 1965-08-24 DE DE19651595953 patent/DE1595953A1/en active Pending
- 1965-08-31 BR BR17276965A patent/BR6572769D0/en unknown
- 1965-08-31 BR BR17274165A patent/BR6572741D0/en unknown
- 1965-09-07 NL NL6511644A patent/NL6511644A/xx unknown
- 1965-09-07 GB GB3179365D patent/GB1112723A/en not_active Expired
- 1965-09-07 CH CH1075068A patent/CH466293A/en unknown
- 1965-09-07 GB GB3816765A patent/GB1112722A/en not_active Expired
- 1965-09-07 SE SE1164765A patent/SE329629B/xx unknown
- 1965-09-07 NL NL6511643A patent/NL6511643A/xx unknown
- 1965-09-07 GB GB3816665A patent/GB1112721A/en not_active Expired
- 1965-09-07 CH CH1243565A patent/CH467271A/en unknown
- 1965-09-07 CH CH1243465A patent/CH475262A/en not_active IP Right Cessation
- 1965-09-07 GB GB3179467A patent/GB1112724A/en not_active Expired
-
1966
- 1966-06-07 DE DE19661620020 patent/DE1620020A1/en active Pending
- 1966-06-29 GB GB2907666A patent/GB1115406A/en not_active Expired
- 1966-07-06 BR BR18106066A patent/BR6681060D0/en unknown
- 1966-07-08 NL NL6609629A patent/NL6609629A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GB1112722A (en) | 1968-05-08 |
| BE668495A (en) | 1966-02-21 |
| GB1115406A (en) | 1968-05-29 |
| BR6572769D0 (en) | 1973-12-26 |
| BE668496A (en) | 1966-02-21 |
| BR6572741D0 (en) | 1973-08-07 |
| DE1595953A1 (en) | 1970-07-09 |
| BR6681060D0 (en) | 1973-12-26 |
| IL24097A (en) | 1969-11-12 |
| CH475262A (en) | 1969-07-15 |
| CH466293A (en) | 1968-12-15 |
| NL6511643A (en) | 1966-03-09 |
| SE329629B (en) | 1970-10-19 |
| NL6511644A (en) | 1966-03-09 |
| GB1112724A (en) | 1968-05-08 |
| DE1595952A1 (en) | 1970-05-14 |
| IL24098A (en) | 1969-03-27 |
| NL6609629A (en) | 1967-01-09 |
| DE1620020A1 (en) | 1970-02-12 |
| CH467271A (en) | 1969-01-15 |
| IL31787A (en) | 1969-07-30 |
| GB1112721A (en) | 1968-05-08 |
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