FR3048884B1 - Composition pour l'administration par voie orale d'au moins un principe actif a un sujet - Google Patents

Composition pour l'administration par voie orale d'au moins un principe actif a un sujet Download PDF

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Publication number
FR3048884B1
FR3048884B1 FR1652329A FR1652329A FR3048884B1 FR 3048884 B1 FR3048884 B1 FR 3048884B1 FR 1652329 A FR1652329 A FR 1652329A FR 1652329 A FR1652329 A FR 1652329A FR 3048884 B1 FR3048884 B1 FR 3048884B1
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France
Prior art keywords
composition
subject
oral administration
active substance
active principle
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Active
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FR1652329A
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English (en)
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FR3048884A1 (fr
Inventor
Victor Roullier
Arnaud Picot
Anthony Gourdon
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Capsulae Fr
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Capsulae SAS
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Priority to FR1652329A priority Critical patent/FR3048884B1/fr
Publication of FR3048884A1 publication Critical patent/FR3048884A1/fr
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Publication of FR3048884B1 publication Critical patent/FR3048884B1/fr
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1652Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1658Proteins, e.g. albumin, gelatin

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  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

L'invention concerne une composition pour l'administration par voie orale d'au moins un principe actif à un sujet. Cette composition comprend des particules d'hydrogel, avantageusement sous forme humide ou sèche, comprenant : - ledit au moins un principe actif, - au moins un polysaccharide gélifiant, - au moins un agent de charge, et - au moins un agent protecteur, choisi parmi les protéines et/ou les résines alimentaires, aptes à conférer une protection dudit au moins un principe actif dans un milieu dont le pH est inférieur à 5,5, lesquelles particules sont aptes à libérer au moins une partie dudit au moins un principe actif dans un milieu dont le pH est supérieur à 5,5.
FR1652329A 2016-03-18 2016-03-18 Composition pour l'administration par voie orale d'au moins un principe actif a un sujet Active FR3048884B1 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR1652329A FR3048884B1 (fr) 2016-03-18 2016-03-18 Composition pour l'administration par voie orale d'au moins un principe actif a un sujet

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR1652329A FR3048884B1 (fr) 2016-03-18 2016-03-18 Composition pour l'administration par voie orale d'au moins un principe actif a un sujet

Publications (2)

Publication Number Publication Date
FR3048884A1 FR3048884A1 (fr) 2017-09-22
FR3048884B1 true FR3048884B1 (fr) 2021-07-30

Family

ID=56555469

Family Applications (1)

Application Number Title Priority Date Filing Date
FR1652329A Active FR3048884B1 (fr) 2016-03-18 2016-03-18 Composition pour l'administration par voie orale d'au moins un principe actif a un sujet

Country Status (1)

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FR (1) FR3048884B1 (fr)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050226905A1 (en) * 2001-05-22 2005-10-13 Tien Canh L Biocompatible compositions as carriers or excipients for pharmaceutical and nutraceutical formulations and for food protection
ITMI20031617A1 (it) * 2003-08-06 2005-02-07 Fond Carlo E Dirce Callerio Onlus Microcapsule a doppio strato di polisaccaridi utilizzabili
US9089152B2 (en) * 2009-04-13 2015-07-28 TEAGASC—Agriculture and Food Development Authority Method of producing microbeads
CN101856604A (zh) * 2010-06-04 2010-10-13 上海理工大学 一种用静电喷雾制备益生菌微胶囊的方法
US9788563B2 (en) * 2011-04-15 2017-10-17 Pepsico, Inc. Encapsulation system for protection of probiotics during processing
CN103110153A (zh) * 2013-02-05 2013-05-22 浙江大学 一种果蔬复合颗粒饮料及其制备方法
CN104911171A (zh) * 2015-05-25 2015-09-16 淮阴工学院 以海藻酸钠、明胶复合凹土制备益生菌微胶囊的方法

Also Published As

Publication number Publication date
FR3048884A1 (fr) 2017-09-22

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