FR3041638A1 - Methode pour ameliorer la capacite d’un compose a traverser les membranes. - Google Patents

Methode pour ameliorer la capacite d’un compose a traverser les membranes. Download PDF

Info

Publication number
FR3041638A1
FR3041638A1 FR1559130A FR1559130A FR3041638A1 FR 3041638 A1 FR3041638 A1 FR 3041638A1 FR 1559130 A FR1559130 A FR 1559130A FR 1559130 A FR1559130 A FR 1559130A FR 3041638 A1 FR3041638 A1 FR 3041638A1
Authority
FR
France
Prior art keywords
compound
peptide
formula
amine function
lysine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
FR1559130A
Other languages
English (en)
French (fr)
Inventor
Nicolas Inguimbert
Haj Salah Khoubaib Ben
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
De Perpignan Via Domitia, University of
Centre National de la Recherche Scientifique CNRS
Universite de Montpellier I
Universite de Perpignan
Universite de Montpellier
Original Assignee
De Perpignan Via Domitia, University of
Centre National de la Recherche Scientifique CNRS
Universite de Montpellier I
Universite de Perpignan
Universite de Montpellier
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by De Perpignan Via Domitia, University of, Centre National de la Recherche Scientifique CNRS, Universite de Montpellier I, Universite de Perpignan, Universite de Montpellier filed Critical De Perpignan Via Domitia, University of
Priority to FR1559130A priority Critical patent/FR3041638A1/fr
Priority to EP16779025.2A priority patent/EP3356383A1/de
Priority to PCT/EP2016/073002 priority patent/WO2017055286A1/fr
Publication of FR3041638A1 publication Critical patent/FR3041638A1/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • C07K1/1072—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups
    • C07K1/1077—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups by covalent attachment of residues other than amino acids or peptide residues, e.g. sugars, polyols, fatty acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Analytical Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
FR1559130A 2015-09-28 2015-09-28 Methode pour ameliorer la capacite d’un compose a traverser les membranes. Withdrawn FR3041638A1 (fr)

Priority Applications (3)

Application Number Priority Date Filing Date Title
FR1559130A FR3041638A1 (fr) 2015-09-28 2015-09-28 Methode pour ameliorer la capacite d’un compose a traverser les membranes.
EP16779025.2A EP3356383A1 (de) 2015-09-28 2016-09-27 Verfahren zur verbesserung der fähigkeit einer verbindung zum durchlaufen von membranen
PCT/EP2016/073002 WO2017055286A1 (fr) 2015-09-28 2016-09-27 Méthode pour améliorer la capacité d'un composé à traverser les membranes

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR1559130A FR3041638A1 (fr) 2015-09-28 2015-09-28 Methode pour ameliorer la capacite d’un compose a traverser les membranes.

Publications (1)

Publication Number Publication Date
FR3041638A1 true FR3041638A1 (fr) 2017-03-31

Family

ID=54707983

Family Applications (1)

Application Number Title Priority Date Filing Date
FR1559130A Withdrawn FR3041638A1 (fr) 2015-09-28 2015-09-28 Methode pour ameliorer la capacite d’un compose a traverser les membranes.

Country Status (3)

Country Link
EP (1) EP3356383A1 (de)
FR (1) FR3041638A1 (de)
WO (1) WO2017055286A1 (de)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001067867A2 (de) * 2000-03-17 2001-09-20 Basf Aktiengesellschaft Ionenkanal-bildende peptaibole als resistenzinduktoren

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001067867A2 (de) * 2000-03-17 2001-09-20 Basf Aktiengesellschaft Ionenkanal-bildende peptaibole als resistenzinduktoren

Non-Patent Citations (3)

* Cited by examiner, † Cited by third party
Title
IBAI E. VALVERDE ET AL: "1,2,3-Triazoles as Amide Bond Mimics: Triazole Scan Yields Protease-Resistant Peptidomimetics for Tumor Targeting", ANGEWANDTE CHEMIE INTERNATIONAL EDITION, vol. 52, no. 34, 5 July 2013 (2013-07-05), DE, pages 8957 - 8960, XP055288655, ISSN: 1433-7851, DOI: 10.1002/anie.201303108 *
IMMA GÜELL ET AL: "Peptidotriazoles with antimicrobial activity against bacterial and fungal plant pathogens", PEPTIDES, ELSEVIER, AMSTERDAM, NL, vol. 33, no. 1, 7 December 2011 (2011-12-07), pages 9 - 17, XP028439857, ISSN: 0196-9781, [retrieved on 20111216], DOI: 10.1016/J.PEPTIDES.2011.12.003 *
OXANA RYABTSOVA ET AL: "Acylated Gly-(2-cyano)pyrrolidines as inhibitors of fibroblast activation protein (FAP) and the issue of FAP/prolyl oligopeptidase (PREP)-selectivity", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, AMSTERDAM, NL, vol. 22, no. 10, 29 March 2012 (2012-03-29), pages 3412 - 3417, XP028479271, ISSN: 0960-894X, [retrieved on 20120404], DOI: 10.1016/J.BMCL.2012.03.107 *

Also Published As

Publication number Publication date
EP3356383A1 (de) 2018-08-08
WO2017055286A1 (fr) 2017-04-06

Similar Documents

Publication Publication Date Title
US9181302B2 (en) WT1 antigen peptide conjugate vaccine
CN101663044B (zh) 三唑大环系统
US9060513B2 (en) Antibiotic peptides
DE60119714T2 (de) Peptidderivat
EP1254162B1 (de) Kahalalide f und verwandte verbindungen
KR20110120917A (ko) 항생 펩티드
HUE031681T2 (en) CMAP27 based antimicrobial peptides
JP5763082B2 (ja) 新規のバシトラシン抗生物質
FR3041638A1 (fr) Methode pour ameliorer la capacite d’un compose a traverser les membranes.
Niederhafner et al. Melectin MAPs: the influence of dendrimerization on antimicrobial and hemolytic activity
US20130130994A1 (en) Antimicrobial peptides and peptide derivatives derived from oncopeltus fasciatus
WO2000075178A1 (fr) Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme antifongiques
DK2493843T3 (en) 2-amino-3-methyl-hex-5-enoic acid and their use in the preparation of peptides, such as bacitracins
US20230103890A1 (en) Photooxygenation Catalyst Compound and Medicine Comprising Same
KR20050072337A (ko) 개구린 5로부터 합성 및 제조된 항생 펩타이드 유도체
HUE033371T2 (en) Process for the preparation of peptide products containing a ring imide
EP1189933A1 (de) Echinocandinderivate, deren herstellung und deren verwendung als fungizid
Levengood et al. Engineering of lantibiotic peptides through the incorporation of nonproteinogenic amino acids

Legal Events

Date Code Title Description
PLFP Fee payment

Year of fee payment: 2

PLSC Publication of the preliminary search report

Effective date: 20170331

PLFP Fee payment

Year of fee payment: 3

PLFP Fee payment

Year of fee payment: 4

ST Notification of lapse

Effective date: 20200906