FR2717804B1 - Sels de composés hétéroaromatiques azotés substitués, procédé pour leur préparation et compositions pharmaceutiques en contenant. - Google Patents

Sels de composés hétéroaromatiques azotés substitués, procédé pour leur préparation et compositions pharmaceutiques en contenant.

Info

Publication number
FR2717804B1
FR2717804B1 FR9403561A FR9403561A FR2717804B1 FR 2717804 B1 FR2717804 B1 FR 2717804B1 FR 9403561 A FR9403561 A FR 9403561A FR 9403561 A FR9403561 A FR 9403561A FR 2717804 B1 FR2717804 B1 FR 2717804B1
Authority
FR
France
Prior art keywords
salts
preparation
pharmaceutical compositions
compositions containing
substituted nitrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9403561A
Other languages
English (en)
Other versions
FR2717804A1 (fr
Inventor
Nathalie Chabert
Xavier Emonds-Alt
Vincenzo Proietto
Didier Van Broeck
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi SA
Original Assignee
Sanofi SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR9403561A priority Critical patent/FR2717804B1/fr
Application filed by Sanofi SA filed Critical Sanofi SA
Priority to AU21421/95A priority patent/AU2142195A/en
Priority to PCT/FR1995/000368 priority patent/WO1995026339A1/fr
Priority to US08/545,772 priority patent/US5665886A/en
Priority to HU9503377A priority patent/HU216843B/hu
Priority to JP7525002A priority patent/JPH08511276A/ja
Priority to EP95914414A priority patent/EP0700387A1/fr
Publication of FR2717804A1 publication Critical patent/FR2717804A1/fr
Application granted granted Critical
Publication of FR2717804B1 publication Critical patent/FR2717804B1/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/06Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
    • C07D213/16Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom containing only one pyridine ring
    • C07D213/18Salts thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR9403561A 1994-03-25 1994-03-25 Sels de composés hétéroaromatiques azotés substitués, procédé pour leur préparation et compositions pharmaceutiques en contenant. Expired - Fee Related FR2717804B1 (fr)

Priority Applications (7)

Application Number Priority Date Filing Date Title
FR9403561A FR2717804B1 (fr) 1994-03-25 1994-03-25 Sels de composés hétéroaromatiques azotés substitués, procédé pour leur préparation et compositions pharmaceutiques en contenant.
PCT/FR1995/000368 WO1995026339A1 (fr) 1994-03-25 1995-03-24 Sels de composes heteroaromatiques azotes substitues, procede pour leur preparation et compositions pharmaceutiques en contenant
US08/545,772 US5665886A (en) 1994-03-25 1995-03-24 Salts of substituted nitrogenous heteroaromatic compounds, a process for their preparation and pharmaceutical compositions containing them
HU9503377A HU216843B (hu) 1994-03-25 1995-03-24 Szubsztituált piridiniumsók, eljárás előállításukra és ezeket tartalmazó gyógyászati készítmények
AU21421/95A AU2142195A (en) 1994-03-25 1995-03-24 Salts of substituted heteroaromatic nitrogen compounds, method for their preparation and pharmaceutical compounds containing same
JP7525002A JPH08511276A (ja) 1994-03-25 1995-03-24 置換された窒素性ヘテロ芳香族化合物の塩、これらの製造方法及びこれらを含有する薬学的組成物
EP95914414A EP0700387A1 (fr) 1994-03-25 1995-03-24 Sels de composes heteroaromatiques azotes substitues, procede pour leur preparation et compositions pharmaceutiques en contenant

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9403561A FR2717804B1 (fr) 1994-03-25 1994-03-25 Sels de composés hétéroaromatiques azotés substitués, procédé pour leur préparation et compositions pharmaceutiques en contenant.

Publications (2)

Publication Number Publication Date
FR2717804A1 FR2717804A1 (fr) 1995-09-29
FR2717804B1 true FR2717804B1 (fr) 1996-06-21

Family

ID=9461452

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9403561A Expired - Fee Related FR2717804B1 (fr) 1994-03-25 1994-03-25 Sels de composés hétéroaromatiques azotés substitués, procédé pour leur préparation et compositions pharmaceutiques en contenant.

Country Status (7)

Country Link
US (1) US5665886A (fr)
EP (1) EP0700387A1 (fr)
JP (1) JPH08511276A (fr)
AU (1) AU2142195A (fr)
FR (1) FR2717804B1 (fr)
HU (1) HU216843B (fr)
WO (1) WO1995026339A1 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2759584B1 (fr) * 1997-02-17 1999-06-11 Sanofi Sa Composition pharmaceutique pour l'administration orale de composes heterocycliques sous forme ammonium quaternaire
FR2759585B1 (fr) * 1997-02-17 1999-06-11 Sanofi Sa Formulations pharmaceutiques presentees sous forme seche pour l'administration orale d'un compose ammonium quaternaire cyclique

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2676055B1 (fr) * 1991-05-03 1993-09-03 Sanofi Elf Composes polycycliques amines et leurs enantiomeres, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2688219B1 (fr) * 1992-03-03 1994-07-08 Sanofi Elf Sels d'ammonium quaternaires de composes aromatiques amines, leur preparation et compositions pharmaceutiques les contenant.
FR2696178B1 (fr) * 1992-09-30 1994-12-30 Sanofi Elf Amides basiques quaternaires, procédé pour leur préparation et compositions pharmaceutiques en contenant.

Also Published As

Publication number Publication date
JPH08511276A (ja) 1996-11-26
FR2717804A1 (fr) 1995-09-29
EP0700387A1 (fr) 1996-03-13
HUT73530A (en) 1996-08-28
US5665886A (en) 1997-09-09
HU9503377D0 (en) 1996-02-28
AU2142195A (en) 1995-10-17
WO1995026339A1 (fr) 1995-10-05
HU216843B (hu) 1999-09-28

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Legal Events

Date Code Title Description
ST Notification of lapse