FR2608601B2 - NOVEL CARBOXAMIDE INDOLE DERIVATIVES, SALTS THEREOF, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, APPLICATION AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM - Google Patents

NOVEL CARBOXAMIDE INDOLE DERIVATIVES, SALTS THEREOF, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, APPLICATION AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM

Info

Publication number
FR2608601B2
FR2608601B2 FR868617810A FR8617810A FR2608601B2 FR 2608601 B2 FR2608601 B2 FR 2608601B2 FR 868617810 A FR868617810 A FR 868617810A FR 8617810 A FR8617810 A FR 8617810A FR 2608601 B2 FR2608601 B2 FR 2608601B2
Authority
FR
France
Prior art keywords
medicaments
intermediates
salts
preparation
application
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR868617810A
Other languages
French (fr)
Other versions
FR2608601A2 (en
Inventor
Francois Clemence
Jacques Guillaume
Gilles Hamon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8510648A external-priority patent/FR2584713B1/en
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Priority to FR868617810A priority Critical patent/FR2608601B2/en
Priority to ES87402892T priority patent/ES2059402T3/en
Priority to EP87402892A priority patent/EP0275762B1/en
Priority to AT87402892T priority patent/ATE97403T1/en
Priority to DE87402892T priority patent/DE3788207T2/en
Priority to DK668687A priority patent/DK169328B1/en
Priority to ZA879523A priority patent/ZA879523B/en
Priority to JP62319123A priority patent/JPS63233972A/en
Priority to FI875586A priority patent/FI85139C/en
Priority to HU875870A priority patent/HU199792B/en
Priority to AU82805/87A priority patent/AU617094B2/en
Priority to IE344187A priority patent/IE61987B1/en
Priority to KR870014617A priority patent/KR880007459A/en
Priority to US07/136,118 priority patent/US4908367A/en
Publication of FR2608601A2 publication Critical patent/FR2608601A2/en
Publication of FR2608601B2 publication Critical patent/FR2608601B2/en
Application granted granted Critical
Priority to US07/438,525 priority patent/US5084455A/en
Priority to US08/066,565 priority patent/US5380722A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/08Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/32Oxygen atoms
    • C07D209/34Oxygen atoms in position 2
FR868617810A 1985-07-11 1986-12-19 NOVEL CARBOXAMIDE INDOLE DERIVATIVES, SALTS THEREOF, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, APPLICATION AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM Expired FR2608601B2 (en)

Priority Applications (16)

Application Number Priority Date Filing Date Title
FR868617810A FR2608601B2 (en) 1985-07-11 1986-12-19 NOVEL CARBOXAMIDE INDOLE DERIVATIVES, SALTS THEREOF, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, APPLICATION AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM
ES87402892T ES2059402T3 (en) 1986-12-19 1987-12-17 DERIVATIVES OF INDOL-CARBOXAMIDE AS WELL AS ITS SALTS, PROCEDURE AND INTERMEDIATE PRODUCTS FOR ITS PREPARATION, APPLICATION AS DRUGS OF THESE DERIVATIVES AND COMPOSITIONS THAT CONTAIN THEM.
EP87402892A EP0275762B1 (en) 1986-12-19 1987-12-17 Indole carboxamide derivatives and their salts, process and intermediates for their preparation, their use as medicines and compositions containing them
AT87402892T ATE97403T1 (en) 1986-12-19 1987-12-17 INDOL CARBOXAMIDE DERIVATIVES AND THEIR SALTS, PROCESSES AND INTERMEDIATE PRODUCTS FOR THE MANUFACTURE, MEDICINAL USE AND COMPOSITIONS CONTAINING THEM.
DE87402892T DE3788207T2 (en) 1986-12-19 1987-12-17 Indole carboxamide derivatives and their salts, processes and intermediates for their preparation, use as medicines and compositions containing them.
FI875586A FI85139C (en) 1986-12-19 1987-12-18 Process for the preparation of novel therapeutically useful indole carboxamide derivatives and their salts
ZA879523A ZA879523B (en) 1986-12-19 1987-12-18 Indolecarboxamide derivatives
JP62319123A JPS63233972A (en) 1986-12-19 1987-12-18 Novel indole carboxamide derivatives and salts, manufacture and intermediates, use for medicines and composition
DK668687A DK169328B1 (en) 1986-12-19 1987-12-18 Indole carboxamide derivatives, their preparation and pharmaceutical preparations containing them
HU875870A HU199792B (en) 1986-12-19 1987-12-18 Process for producing new indolecarboxamide derivatives and pharmaceutical compositions comprising such compounds
AU82805/87A AU617094B2 (en) 1986-12-19 1987-12-18 New indolecarboxamide derivatives as well as salts thereof, process and intermediates for preparation, application of these derivatives by way of medicinal products and compositions containing them
IE344187A IE61987B1 (en) 1986-12-19 1987-12-18 New indolecarboxamide derivatives as well as salts thereof, process and intermediates for preparation, application of these derivatives by way of medicinal products and compositions containing same
KR870014617A KR880007459A (en) 1986-12-19 1987-12-19 Indole carboxyamide derivatives, salts thereof, preparation methods and intermediates thereof, use of such derivatives as pharmaceuticals and compositions containing them
US07/136,118 US4908367A (en) 1985-07-11 1987-12-21 N-(1H-indole-4-yl)-benzamides
US07/438,525 US5084455A (en) 1985-07-11 1989-11-17 Novel indole carboxamides
US08/066,565 US5380722A (en) 1985-07-11 1993-05-25 Indole carboxamides

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8510648A FR2584713B1 (en) 1985-07-11 1985-07-11 NOVEL CARBOXAMIDE INDOLE DERIVATIVES, SALTS THEREOF, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, APPLICATION AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM
FR868617810A FR2608601B2 (en) 1985-07-11 1986-12-19 NOVEL CARBOXAMIDE INDOLE DERIVATIVES, SALTS THEREOF, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, APPLICATION AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM

Publications (2)

Publication Number Publication Date
FR2608601A2 FR2608601A2 (en) 1988-06-24
FR2608601B2 true FR2608601B2 (en) 1989-04-14

Family

ID=26224613

Family Applications (1)

Application Number Title Priority Date Filing Date
FR868617810A Expired FR2608601B2 (en) 1985-07-11 1986-12-19 NOVEL CARBOXAMIDE INDOLE DERIVATIVES, SALTS THEREOF, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, APPLICATION AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM

Country Status (1)

Country Link
FR (1) FR2608601B2 (en)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2528043A1 (en) * 1982-06-03 1983-12-09 Roussel Uclaf NOVEL 1,3-DIHYDRO 4- / 1-HYDROXY-2-AMINO-ETHYL / 2H-INDOL-2-ONE DERIVATIVES, THEIR SALTS, PREPARATION METHOD, MEDICAMENT APPLICATION AND COMPOSITIONS COMPRISING THE SAME
US4853408A (en) * 1985-04-23 1989-08-01 Roussel Uclaf 4-phenylpropyl-indoles having antiarythmic activity
FR2583047B1 (en) * 1985-06-05 1988-01-08 Roussel Uclaf PROCESS FOR THE PREPARATION OF INDOLE 4-PHENYLPROPYL DERIVATIVES AND INTERMEDIATES

Also Published As

Publication number Publication date
FR2608601A2 (en) 1988-06-24

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