FR2395994A1 - Nouveaux derives d'aminoacides a-acetyleniques et leur utilisation therapeutique - Google Patents

Nouveaux derives d'aminoacides a-acetyleniques et leur utilisation therapeutique

Info

Publication number
FR2395994A1
FR2395994A1 FR7819345A FR7819345A FR2395994A1 FR 2395994 A1 FR2395994 A1 FR 2395994A1 FR 7819345 A FR7819345 A FR 7819345A FR 7819345 A FR7819345 A FR 7819345A FR 2395994 A1 FR2395994 A1 FR 2395994A1
Authority
FR
France
Prior art keywords
acetylenicaminoacids
therapeutic use
new derivatives
new
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7819345A
Other languages
English (en)
Other versions
FR2395994B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merrell Toraude et Cie
Original Assignee
Merrell Toraude et Cie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Toraude et Cie filed Critical Merrell Toraude et Cie
Publication of FR2395994A1 publication Critical patent/FR2395994A1/fr
Application granted granted Critical
Publication of FR2395994B1 publication Critical patent/FR2395994B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C243/00—Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D209/20—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals substituted additionally by nitrogen atoms, e.g. tryptophane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D317/30—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Abstract

Les nouveaux composé selon l'invention répondent à la formule générale :
FR7819345A 1977-07-01 1978-06-28 Nouveaux derives d'aminoacides a-acetyleniques et leur utilisation therapeutique Granted FR2395994A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/812,052 US4180509A (en) 1977-07-01 1977-07-01 α-Ethynyl tryptophanes

Publications (2)

Publication Number Publication Date
FR2395994A1 true FR2395994A1 (fr) 1979-01-26
FR2395994B1 FR2395994B1 (fr) 1980-10-31

Family

ID=25208350

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7819345A Granted FR2395994A1 (fr) 1977-07-01 1978-06-28 Nouveaux derives d'aminoacides a-acetyleniques et leur utilisation therapeutique

Country Status (7)

Country Link
US (1) US4180509A (fr)
AU (1) AU515468B2 (fr)
BE (1) BE868589A (fr)
FR (1) FR2395994A1 (fr)
IT (1) IT1105058B (fr)
NZ (1) NZ187540A (fr)
ZA (1) ZA783353B (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2310369A1 (fr) * 2008-06-24 2011-04-20 Valeant Pharmaceuticals International Dérivés de benzyloxy anilide utiles en tant que modulateurs du canal potassique

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZW19381A1 (en) * 1980-08-12 1983-03-09 Glaxo Group Ltd Heterocyclic compounds
US4537907A (en) * 1980-10-06 1985-08-27 University Of Illinois Foundation Hypnotic composition and method of inducing sleep
NZ551511A (en) * 2004-06-04 2010-09-30 Xenoport Inc Levodopa prodrugs, and compositions and uses thereof
WO2005121070A1 (fr) * 2004-06-04 2005-12-22 Xenoport, Inc. Promedicaments de levodopa, et compositions et leurs utilisations
CN101365439B (zh) * 2005-12-05 2012-12-26 克塞诺波特公司 左旋多巴前体药物甲磺酸盐、其组合物及其用途
US7829592B2 (en) * 2006-12-21 2010-11-09 Xenoport, Inc. Catechol protected levodopa diester prodrugs, compositions, and methods of use
JP2011502953A (ja) * 2006-12-21 2011-01-27 ゼノポート，インコーポレーテッド ジメチル置換されたレボドパジエステルのプロドラッグ、組成物及び使用方法
CN102186804A (zh) * 2008-10-20 2011-09-14 克塞诺波特公司 合成左旋多巴酯前药的方法
US8399513B2 (en) 2008-10-20 2013-03-19 Xenoport, Inc. Levodopa prodrug mesylate hydrate
AU2010315892B2 (en) 2009-11-09 2014-09-18 Xenoport, Inc. Pharmaceutical compositions and oral dosage forms of a levodopa prodrug and methods of use

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA557705A (fr) * 1958-05-20 R. Snyder Harold Preparation de n-acyle-tryptophanes
US3079345A (en) * 1959-04-30 1963-02-26 Dow Chemical Co Propargyl compounds as corrosion inhibitors
US4041041A (en) * 1975-03-18 1977-08-09 Merrell Toraude Et Compagnie Acetylene derivatives of amino acids

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2310369A1 (fr) * 2008-06-24 2011-04-20 Valeant Pharmaceuticals International Dérivés de benzyloxy anilide utiles en tant que modulateurs du canal potassique
EP2310369A4 (fr) * 2008-06-24 2014-02-19 Valeant Pharmaceuticals Int Dérivés de benzyloxy anilide utiles en tant que modulateurs du canal potassique

Also Published As

Publication number Publication date
AU3732478A (en) 1980-01-03
BE868589A (fr) 1978-10-16
US4180509A (en) 1979-12-25
FR2395994B1 (fr) 1980-10-31
ZA783353B (en) 1979-06-27
IT7850018A0 (it) 1978-06-26
NZ187540A (en) 1982-05-25
AU515468B2 (en) 1981-04-02
IT1105058B (it) 1985-10-28

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Legal Events

Date Code Title Description
ST Notification of lapse