FR2384498A1 - Nouveaux derives sulfonylamino thiazoliques et leurs applications en medecine humaine et veterinaire - Google Patents
Nouveaux derives sulfonylamino thiazoliques et leurs applications en medecine humaine et veterinaireInfo
- Publication number
- FR2384498A1 FR2384498A1 FR7536118A FR7536118A FR2384498A1 FR 2384498 A1 FR2384498 A1 FR 2384498A1 FR 7536118 A FR7536118 A FR 7536118A FR 7536118 A FR7536118 A FR 7536118A FR 2384498 A1 FR2384498 A1 FR 2384498A1
- Authority
- FR
- France
- Prior art keywords
- prepd
- sulphonamido
- isothiocyanato
- butyne
- thiazole
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- -1 sulphonamido thiazole Chemical compound 0.000 title abstract 5
- 230000000844 anti-bacterial effect Effects 0.000 title abstract 2
- 229940121375 antifungal agent Drugs 0.000 title abstract 2
- 230000002218 hypoglycaemic effect Effects 0.000 title abstract 2
- KHBQMWCZKVMBLN-UHFFFAOYSA-N Benzenesulfonamide Chemical compound NS(=O)(=O)C1=CC=CC=C1 KHBQMWCZKVMBLN-UHFFFAOYSA-N 0.000 title 1
- ZNOPAVGGORUIHN-UHFFFAOYSA-N N(=C=S)C#CCC Chemical compound N(=C=S)C#CCC ZNOPAVGGORUIHN-UHFFFAOYSA-N 0.000 title 1
- 230000000843 anti-fungal effect Effects 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- BWHMMNNQKKPAPP-UHFFFAOYSA-L potassium carbonate Chemical compound [K+].[K+].[O-]C([O-])=O BWHMMNNQKKPAPP-UHFFFAOYSA-L 0.000 abstract 2
- FPIDKDMAINJQKV-UHFFFAOYSA-N 4-(4-isothiocyanatobut-2-ynyl)morpholine Chemical compound S=C=NCC#CCN1CCOCC1 FPIDKDMAINJQKV-UHFFFAOYSA-N 0.000 abstract 1
- 125000000218 acetic acid group Chemical group C(C)(=O)* 0.000 abstract 1
- 125000004442 acylamino group Chemical group 0.000 abstract 1
- 229940088710 antibiotic agent Drugs 0.000 abstract 1
- 239000003429 antifungal agent Substances 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 229910000027 potassium carbonate Inorganic materials 0.000 abstract 1
- 235000015320 potassium carbonate Nutrition 0.000 abstract 1
- LMYRWZFENFIFIT-UHFFFAOYSA-N toluene-4-sulfonamide Chemical compound CC1=CC=C(S(N)(=O)=O)C=C1 LMYRWZFENFIFIT-UHFFFAOYSA-N 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/50—Nitrogen atoms bound to hetero atoms
- C07D277/52—Nitrogen atoms bound to hetero atoms to sulfur atoms, e.g. sulfonamides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7536118A FR2384498A1 (fr) | 1975-11-26 | 1975-11-26 | Nouveaux derives sulfonylamino thiazoliques et leurs applications en medecine humaine et veterinaire |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7536118A FR2384498A1 (fr) | 1975-11-26 | 1975-11-26 | Nouveaux derives sulfonylamino thiazoliques et leurs applications en medecine humaine et veterinaire |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2384498A1 true FR2384498A1 (fr) | 1978-10-20 |
| FR2384498B1 FR2384498B1 (https=) | 1979-09-28 |
Family
ID=9162918
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7536118A Granted FR2384498A1 (fr) | 1975-11-26 | 1975-11-26 | Nouveaux derives sulfonylamino thiazoliques et leurs applications en medecine humaine et veterinaire |
Country Status (1)
| Country | Link |
|---|---|
| FR (1) | FR2384498A1 (https=) |
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2001090090A1 (en) * | 2000-05-22 | 2001-11-29 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| WO2003043999A1 (en) * | 2001-11-22 | 2003-05-30 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| US7074788B2 (en) | 2001-11-22 | 2006-07-11 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| US7094792B2 (en) | 2001-11-22 | 2006-08-22 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| AU2007205749B2 (en) * | 2001-11-22 | 2009-04-23 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| US8541593B2 (en) | 2007-06-21 | 2013-09-24 | Amgen Inc. | Process for making substituted 2-amino-thiazolones |
-
1975
- 1975-11-26 FR FR7536118A patent/FR2384498A1/fr active Granted
Non-Patent Citations (1)
| Title |
|---|
| NEANT * |
Cited By (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2001090090A1 (en) * | 2000-05-22 | 2001-11-29 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| US7030135B2 (en) | 2000-05-22 | 2006-04-18 | Biovitrum Ab | Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 |
| US7132436B2 (en) | 2000-05-22 | 2006-11-07 | Biovitrum Ab | Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 |
| US7618961B2 (en) | 2000-05-22 | 2009-11-17 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| WO2003043999A1 (en) * | 2001-11-22 | 2003-05-30 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| JP2005509675A (ja) * | 2001-11-22 | 2005-04-14 | ビオヴィトルム・アクチボラゲット | １１−ベータ−ヒドロキシステロイド脱水素酵素タイプ１のインヒビター |
| US7074788B2 (en) | 2001-11-22 | 2006-07-11 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| US7094792B2 (en) | 2001-11-22 | 2006-08-22 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| AU2007205749B2 (en) * | 2001-11-22 | 2009-04-23 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| US7671051B2 (en) | 2001-11-22 | 2010-03-02 | Biovitrum Ab | Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 |
| US8541593B2 (en) | 2007-06-21 | 2013-09-24 | Amgen Inc. | Process for making substituted 2-amino-thiazolones |
Also Published As
| Publication number | Publication date |
|---|---|
| FR2384498B1 (https=) | 1979-09-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |