FR2382452A1 - 3, 7-dihydro- et 1, 7-dihydro-4h-pyrazolo (4', 3':5, 6) pyrido (4, 3-d) pyrimidin-4-ones et leur utilisation comme medicaments - Google Patents

3, 7-dihydro- et 1, 7-dihydro-4h-pyrazolo (4', 3':5, 6) pyrido (4, 3-d) pyrimidin-4-ones et leur utilisation comme medicaments

Info

Publication number
FR2382452A1
FR2382452A1 FR7806020A FR7806020A FR2382452A1 FR 2382452 A1 FR2382452 A1 FR 2382452A1 FR 7806020 A FR7806020 A FR 7806020A FR 7806020 A FR7806020 A FR 7806020A FR 2382452 A1 FR2382452 A1 FR 2382452A1
Authority
FR
France
Prior art keywords
dihydro
pyrazolo
pyrido
pyrimidin
ones
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7806020A
Other languages
English (en)
Other versions
FR2382452B1 (fr
Inventor
Theodor Denzel
Hans Hoehn
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of FR2382452A1 publication Critical patent/FR2382452A1/fr
Application granted granted Critical
Publication of FR2382452B1 publication Critical patent/FR2382452B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Anesthesiology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne de nouvelles 3,7-dihydro et 1,7-dihydro-4H-pyrazolo Ø4', 3':5, 6õ pyrido Ø4, 3-dõ pyrimidin-4-ones de formule :
FR7806020A 1977-03-02 1978-03-02 3, 7-dihydro- et 1, 7-dihydro-4h-pyrazolo (4', 3':5, 6) pyrido (4, 3-d) pyrimidin-4-ones et leur utilisation comme medicaments Granted FR2382452A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/773,562 US4072681A (en) 1977-03-02 1977-03-02 3,7-Dihydro- and 1,7-dihydro-4H-pyrazolo[4',3':5,6]pyrido[4,3-d]pyrimidin-4-ones

Publications (2)

Publication Number Publication Date
FR2382452A1 true FR2382452A1 (fr) 1978-09-29
FR2382452B1 FR2382452B1 (fr) 1980-12-19

Family

ID=25098664

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7806020A Granted FR2382452A1 (fr) 1977-03-02 1978-03-02 3, 7-dihydro- et 1, 7-dihydro-4h-pyrazolo (4', 3':5, 6) pyrido (4, 3-d) pyrimidin-4-ones et leur utilisation comme medicaments

Country Status (6)

Country Link
US (1) US4072681A (fr)
JP (1) JPS53109000A (fr)
CA (1) CA1091667A (fr)
DE (1) DE2809033A1 (fr)
FR (1) FR2382452A1 (fr)
GB (1) GB1597091A (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58138166U (ja) * 1982-03-11 1983-09-17 株式会社東芝 自動改札装置
US4511568A (en) * 1982-05-12 1985-04-16 Ici Americas Inc. CNS-Depressant pyrazolopyridines
JP2002540102A (ja) 1999-03-22 2002-11-26 ブリストル−マイヤーズ スクイブ カンパニー ｃＧＭＰホスホジエステラーゼの縮合ピリドピリダジン阻害剤
GB0119828D0 (en) * 2001-08-14 2001-10-10 Merck Sharp & Dohme Therapeutic agents
GB0405937D0 (en) * 2004-03-16 2004-04-21 Glaxo Group Ltd Compounds
WO2012127506A1 (fr) * 2011-03-22 2012-09-27 Advinus Therapeutics Limited Composés tricycliques substitués; compositions et applications médicinales correspondantes

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3894021A (en) * 1974-01-28 1975-07-08 Squibb & Sons Inc Derivatives of 1,7-dihydro-2H-pyrazolo{8 4{40 ,3{40 :5,6{9 pyrido{8 4,3-D{9 pyrimidine-2,4-(3H)-diones

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3894021A (en) * 1974-01-28 1975-07-08 Squibb & Sons Inc Derivatives of 1,7-dihydro-2H-pyrazolo{8 4{40 ,3{40 :5,6{9 pyrido{8 4,3-D{9 pyrimidine-2,4-(3H)-diones

Also Published As

Publication number Publication date
US4072681A (en) 1978-02-07
GB1597091A (en) 1981-09-03
FR2382452B1 (fr) 1980-12-19
DE2809033A1 (de) 1978-09-07
CA1091667A (fr) 1980-12-16
JPS53109000A (en) 1978-09-22

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Legal Events

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