FR2369296A1 - Derives de 5-fluorouracile, leur procede de preparation et leur application therapeutique - Google Patents
Derives de 5-fluorouracile, leur procede de preparation et leur application therapeutiqueInfo
- Publication number
- FR2369296A1 FR2369296A1 FR7732748A FR7732748A FR2369296A1 FR 2369296 A1 FR2369296 A1 FR 2369296A1 FR 7732748 A FR7732748 A FR 7732748A FR 7732748 A FR7732748 A FR 7732748A FR 2369296 A1 FR2369296 A1 FR 2369296A1
- Authority
- FR
- France
- Prior art keywords
- preparation process
- therapeutic application
- fluorouracil derivatives
- fluorouracil
- positions
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- GHASVSINZRGABV-UHFFFAOYSA-N Fluorouracil Chemical class FC1=CNC(=O)NC1=O GHASVSINZRGABV-UHFFFAOYSA-N 0.000 title abstract 3
- 238000002360 preparation method Methods 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
- 230000000259 anti-tumor effect Effects 0.000 abstract 1
- 239000002246 antineoplastic agent Substances 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- -1 glycosyl halide Chemical class 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000002184 metal Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP13020076A JPS5356677A (en) | 1976-10-28 | 1976-10-28 | 5-fluorouracil derivatives |
| JP4321477A JPS53135987A (en) | 1977-04-15 | 1977-04-15 | 5-fluorouracil derivative |
| JP5849277A JPS53144582A (en) | 1977-05-20 | 1977-05-20 | 5-fluorouracil derivatives |
| JP11037077A JPS5444681A (en) | 1977-09-13 | 1977-09-13 | 5-fluororacil derivative |
| JP11086777A JPS5444682A (en) | 1977-09-14 | 1977-09-14 | 5-fluorouracil derivative |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2369296A1 true FR2369296A1 (fr) | 1978-05-26 |
| FR2369296B1 FR2369296B1 (enrdf_load_stackoverflow) | 1982-06-11 |
Family
ID=27522306
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7732748A Granted FR2369296A1 (fr) | 1976-10-28 | 1977-10-28 | Derives de 5-fluorouracile, leur procede de preparation et leur application therapeutique |
Country Status (6)
| Country | Link |
|---|---|
| CH (3) | CH642974A5 (enrdf_load_stackoverflow) |
| DE (1) | DE2748562A1 (enrdf_load_stackoverflow) |
| DK (1) | DK149818C (enrdf_load_stackoverflow) |
| FR (1) | FR2369296A1 (enrdf_load_stackoverflow) |
| GB (1) | GB1541185A (enrdf_load_stackoverflow) |
| NL (1) | NL7711911A (enrdf_load_stackoverflow) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE204878T1 (de) * | 1995-06-23 | 2001-09-15 | Oxford Glycosciences Uk Ltd | Therapeutische verbindungen |
| GB9626450D0 (en) * | 1996-12-20 | 1997-02-05 | Oxford Glycosciences Uk Ltd | Therapeutic compounds |
| WO2003000712A1 (fr) | 2001-06-20 | 2003-01-03 | Kissei Pharmaceutical Co., Ltd. | Derive heterocyclique azote, composition medicinale contenant ce derive, leur utilisation medicinale et intermediaire associe |
-
1977
- 1977-10-27 DK DK478177A patent/DK149818C/da not_active IP Right Cessation
- 1977-10-28 FR FR7732748A patent/FR2369296A1/fr active Granted
- 1977-10-28 CH CH1318477A patent/CH642974A5/de not_active IP Right Cessation
- 1977-10-28 GB GB44960/77A patent/GB1541185A/en not_active Expired
- 1977-10-28 NL NL7711911A patent/NL7711911A/xx not_active Application Discontinuation
- 1977-10-28 DE DE19772748562 patent/DE2748562A1/de not_active Ceased
- 1977-10-28 CH CH2395/84A patent/CH650006A5/de not_active IP Right Cessation
-
1981
- 1981-12-15 CH CH800481A patent/CH643272A5/de not_active IP Right Cessation
Non-Patent Citations (2)
| Title |
|---|
| CA1978 * |
| EXBK/ * |
Also Published As
| Publication number | Publication date |
|---|---|
| CH642974A5 (en) | 1984-05-15 |
| DK149818C (da) | 1987-04-06 |
| CH643272A5 (en) | 1984-05-30 |
| DK478177A (da) | 1978-04-29 |
| DK149818B (da) | 1986-10-06 |
| NL7711911A (nl) | 1978-05-03 |
| CH650006A5 (en) | 1985-06-28 |
| GB1541185A (en) | 1979-02-21 |
| FR2369296B1 (enrdf_load_stackoverflow) | 1982-06-11 |
| DE2748562A1 (de) | 1978-05-03 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FR2426695A1 (fr) | Nouvelles cephalosporines, leur procede de preparation et leur application therapeutique | |
| OA06064A (fr) | Produits d'hydrogénation sélective des composés C-076 et leurs dérivés. | |
| OA05914A (fr) | Procédé de préparation de nouveaux dérivés de la taurine à activité neuro-musculaire renforcée. | |
| BE903334A (fr) | Nouveaux derives naphtaleniques a action retinoique, leurs procedes de preparation et compositions medicamenteuse et cosmetique les contenant | |
| BE900842A (fr) | Nouveaux complexes de platine et leur application en therapeutique. | |
| FR2434156A2 (fr) | Composes d'imidazolium quaternaire, leur procede de preparation et compositions, notamment microbicides les contenant | |
| FR2426694A1 (fr) | Cephalosporines perfectionnees, leur procede de preparation et leur application therapeutique | |
| FR2374307A1 (fr) | Derives de la 1,4-dihydropyridine, leur procede d'obtention et composition pharmaceutique les contenant | |
| FR2394542A1 (fr) | Derives de 3-(1-pyrazolyl)-pyridazine et leur procede de preparation et nouveaux medicaments les contenant | |
| FR2369296A1 (fr) | Derives de 5-fluorouracile, leur procede de preparation et leur application therapeutique | |
| BE903376A (fr) | Derives de la vitamine d et precurseurs de ceux-ci et compositions pharmaceutiques en contenant | |
| GB1309679A (en) | Substituted sulphonanilides | |
| FR2422667A1 (fr) | Derives de 7a-methoxycephalosporine, leur procede de preparation et leur application en therapeutique | |
| FR2368479A1 (fr) | Procede pour monoacyler des acides aminohydroxynaphtalene-sulfoniques avec une 2,4,6-trifluoro-s-triazine | |
| ES299418A1 (es) | Procedimiento para la preparación de nucleósidos de fluoropirimidina | |
| FR2428045A1 (fr) | Derives silyles de naphtacenones utilisables notamment dans la synthese d'agents antitumeurs | |
| JPS57179197A (en) | 17 alpha-alkyne-17 beta-hydroxy-1 alpha- methyl-4-androstene-3-one, manufacture and medicine having anti-androgenic activity and fat production inhibiting activity | |
| OA05777A (fr) | Compositions biocides à base de dérivés aryles d'hydrazone pour lutter contre les maladies des plantes. | |
| BE1000719A4 (fr) | Derives de 3-(hydroxymethyl)-isoquinoleine, procede pour les preparer et compositions pharmaceutiques les contenant. | |
| SE332172B (enrdf_load_stackoverflow) | ||
| ES8305717A1 (es) | Procedimiento para la obtencion de derivados de 2-amino-3,4-dihidropiridina sustituidos. | |
| BE905751A (fr) | Nitro-anthracycline, aglycone correspondante, procedes pour les preparer, composition pharmaceutique correspondante. | |
| BE903438A (fr) | Nouveaux derives de la phenethylaminoalcoyle-6 furo-(3,4-c)-pyridine, leur preparation et compositions therapeutiques a base de ceux-ci | |
| BE902710A (fr) | Procede stereospecifique pour la preparation d'azetidinones. | |
| FR2392006A1 (fr) | B-lactames monocycliques, leur procede de preparation et leur application en therapeutique |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |