FR2358414A1 - Derives peptidiques, leur preparation et leur application comme agents antibacteriens - Google Patents
Derives peptidiques, leur preparation et leur application comme agents antibacteriensInfo
- Publication number
- FR2358414A1 FR2358414A1 FR7721280A FR7721280A FR2358414A1 FR 2358414 A1 FR2358414 A1 FR 2358414A1 FR 7721280 A FR7721280 A FR 7721280A FR 7721280 A FR7721280 A FR 7721280A FR 2358414 A1 FR2358414 A1 FR 2358414A1
- Authority
- FR
- France
- Prior art keywords
- phosphonic acid
- antibacterial
- activity against
- gram positive
- against gram
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 108090000765 processed proteins & peptides Proteins 0.000 title abstract 3
- ABLZXFCXXLZCGV-UHFFFAOYSA-N Phosphorous acid Chemical compound OP(O)=O ABLZXFCXXLZCGV-UHFFFAOYSA-N 0.000 title 1
- 230000000844 anti-bacterial effect Effects 0.000 title 1
- 230000000694 effects Effects 0.000 title 1
- 241000147019 Enterobacter sp. Species 0.000 abstract 1
- 241000588724 Escherichia coli Species 0.000 abstract 1
- 241000606768 Haemophilus influenzae Species 0.000 abstract 1
- 241000588915 Klebsiella aerogenes Species 0.000 abstract 1
- 241000293869 Salmonella enterica subsp. enterica serovar Typhimurium Species 0.000 abstract 1
- 241000607715 Serratia marcescens Species 0.000 abstract 1
- 230000002378 acidificating effect Effects 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 150000001413 amino acids Chemical class 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- GRKSQRAVWODMGW-UHFFFAOYSA-N ethylphosphonic acid Chemical compound [CH2]CP(O)(O)=O GRKSQRAVWODMGW-UHFFFAOYSA-N 0.000 abstract 1
- 229940047650 haemophilus influenzae Drugs 0.000 abstract 1
- 230000007935 neutral effect Effects 0.000 abstract 1
- 102000004196 processed proteins & peptides Human genes 0.000 abstract 1
- 102000004169 proteins and genes Human genes 0.000 abstract 1
- 108090000623 proteins and genes Proteins 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
- C07F9/301—Acyclic saturated acids which can have further substituents on alkyl
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
- C07F9/3808—Acyclic saturated acids which can have further substituents on alkyl
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB2910176 | 1976-07-13 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2358414A1 true FR2358414A1 (fr) | 1978-02-10 |
| FR2358414B1 FR2358414B1 (enExample) | 1979-06-01 |
Family
ID=10286172
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7721280A Granted FR2358414A1 (fr) | 1976-07-13 | 1977-07-11 | Derives peptidiques, leur preparation et leur application comme agents antibacteriens |
Country Status (13)
| Country | Link |
|---|---|
| JP (1) | JPS539720A (enExample) |
| AU (1) | AU2684777A (enExample) |
| BE (1) | BE856724A (enExample) |
| DE (1) | DE2730524A1 (enExample) |
| DK (1) | DK317177A (enExample) |
| FR (1) | FR2358414A1 (enExample) |
| IL (1) | IL52469A0 (enExample) |
| IT (1) | IT1081511B (enExample) |
| LU (1) | LU77725A1 (enExample) |
| NL (1) | NL7707736A (enExample) |
| NZ (1) | NZ184603A (enExample) |
| SE (1) | SE7708120L (enExample) |
| ZA (1) | ZA774073B (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0014834A1 (de) * | 1979-01-18 | 1980-09-03 | Hoechst Aktiengesellschaft | Verfahren zur Herstellung von Carbonsäureamiden und Peptiden |
| EP1585751A4 (en) * | 2002-11-14 | 2008-08-13 | Celmed Oncology Usa Inc | PEPTIDE DEFORMYLASE-ACTIVATED PRODRUGS |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GR73085B (enExample) * | 1977-12-20 | 1984-01-31 | Hoffmann La Roche | |
| CA1108125A (en) * | 1977-12-23 | 1981-09-01 | Frank R. Atherton | Olgiopeptide derivatives of phosphonic acid |
| EP0103867B1 (en) * | 1982-09-17 | 1986-12-17 | Kyowa Hakko Kogyo Co., Ltd. | Phosphorus-containing peptide derivative |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2298335A1 (fr) * | 1975-01-27 | 1976-08-20 | Hoffmann La Roche | Nouveaux derives de peptides d'acides phosphonique et phosphinique |
-
1977
- 1977-06-29 IT IT25208/77A patent/IT1081511B/it active
- 1977-07-06 DE DE19772730524 patent/DE2730524A1/de active Pending
- 1977-07-06 ZA ZA00774073A patent/ZA774073B/xx unknown
- 1977-07-06 IL IL52469A patent/IL52469A0/xx unknown
- 1977-07-07 AU AU26847/77A patent/AU2684777A/en active Pending
- 1977-07-08 NZ NZ184603A patent/NZ184603A/xx unknown
- 1977-07-11 FR FR7721280A patent/FR2358414A1/fr active Granted
- 1977-07-11 LU LU77725A patent/LU77725A1/xx unknown
- 1977-07-11 JP JP8209977A patent/JPS539720A/ja active Pending
- 1977-07-12 SE SE7708120A patent/SE7708120L/xx unknown
- 1977-07-12 DK DK317177A patent/DK317177A/da unknown
- 1977-07-12 NL NL7707736A patent/NL7707736A/xx not_active Application Discontinuation
- 1977-07-12 BE BE179267A patent/BE856724A/xx unknown
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2298335A1 (fr) * | 1975-01-27 | 1976-08-20 | Hoffmann La Roche | Nouveaux derives de peptides d'acides phosphonique et phosphinique |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0014834A1 (de) * | 1979-01-18 | 1980-09-03 | Hoechst Aktiengesellschaft | Verfahren zur Herstellung von Carbonsäureamiden und Peptiden |
| EP1585751A4 (en) * | 2002-11-14 | 2008-08-13 | Celmed Oncology Usa Inc | PEPTIDE DEFORMYLASE-ACTIVATED PRODRUGS |
Also Published As
| Publication number | Publication date |
|---|---|
| FR2358414B1 (enExample) | 1979-06-01 |
| SE7708120L (sv) | 1978-01-14 |
| NZ184603A (en) | 1980-03-05 |
| DK317177A (da) | 1978-01-14 |
| DE2730524A1 (de) | 1978-01-19 |
| IT1081511B (it) | 1985-05-21 |
| AU2684777A (en) | 1979-01-11 |
| JPS539720A (en) | 1978-01-28 |
| NL7707736A (nl) | 1978-01-17 |
| LU77725A1 (enExample) | 1978-09-14 |
| IL52469A0 (en) | 1977-10-31 |
| BE856724A (fr) | 1978-01-12 |
| ZA774073B (en) | 1978-05-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |