FR2358414A1 - Derives peptidiques, leur preparation et leur application comme agents antibacteriens - Google Patents
Derives peptidiques, leur preparation et leur application comme agents antibacteriensInfo
- Publication number
- FR2358414A1 FR2358414A1 FR7721280A FR7721280A FR2358414A1 FR 2358414 A1 FR2358414 A1 FR 2358414A1 FR 7721280 A FR7721280 A FR 7721280A FR 7721280 A FR7721280 A FR 7721280A FR 2358414 A1 FR2358414 A1 FR 2358414A1
- Authority
- FR
- France
- Prior art keywords
- phosphonic acid
- antibacterial
- activity against
- gram positive
- against gram
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 108090000765 processed proteins & peptides Proteins 0.000 title abstract 3
- ABLZXFCXXLZCGV-UHFFFAOYSA-N Phosphorous acid Chemical compound OP(O)=O ABLZXFCXXLZCGV-UHFFFAOYSA-N 0.000 title 1
- 230000000844 anti-bacterial effect Effects 0.000 title 1
- 230000000694 effects Effects 0.000 title 1
- 241000147019 Enterobacter sp. Species 0.000 abstract 1
- 241000588724 Escherichia coli Species 0.000 abstract 1
- 241000606768 Haemophilus influenzae Species 0.000 abstract 1
- 241000588915 Klebsiella aerogenes Species 0.000 abstract 1
- 241000293869 Salmonella enterica subsp. enterica serovar Typhimurium Species 0.000 abstract 1
- 241000607715 Serratia marcescens Species 0.000 abstract 1
- 230000002378 acidificating effect Effects 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 150000001413 amino acids Chemical class 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- GRKSQRAVWODMGW-UHFFFAOYSA-N ethylphosphonic acid Chemical compound [CH2]CP(O)(O)=O GRKSQRAVWODMGW-UHFFFAOYSA-N 0.000 abstract 1
- 229940047650 haemophilus influenzae Drugs 0.000 abstract 1
- 230000007935 neutral effect Effects 0.000 abstract 1
- 102000004196 processed proteins & peptides Human genes 0.000 abstract 1
- 102000004169 proteins and genes Human genes 0.000 abstract 1
- 108090000623 proteins and genes Proteins 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
- C07F9/301—Acyclic saturated acids which can have further substituents on alkyl
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
- C07F9/3808—Acyclic saturated acids which can have further substituents on alkyl
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
L'invention concerne des composés chimiques nouveaux, un procédé pour leur préparation, et des préparations pharmaceutiques les contenant. Les nouveaux composés sont des dérivés peptidiques de formule générale :
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB2910176 | 1976-07-13 |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2358414A1 true FR2358414A1 (fr) | 1978-02-10 |
FR2358414B1 FR2358414B1 (fr) | 1979-06-01 |
Family
ID=10286172
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7721280A Granted FR2358414A1 (fr) | 1976-07-13 | 1977-07-11 | Derives peptidiques, leur preparation et leur application comme agents antibacteriens |
Country Status (13)
Country | Link |
---|---|
JP (1) | JPS539720A (fr) |
AU (1) | AU2684777A (fr) |
BE (1) | BE856724A (fr) |
DE (1) | DE2730524A1 (fr) |
DK (1) | DK317177A (fr) |
FR (1) | FR2358414A1 (fr) |
IL (1) | IL52469A0 (fr) |
IT (1) | IT1081511B (fr) |
LU (1) | LU77725A1 (fr) |
NL (1) | NL7707736A (fr) |
NZ (1) | NZ184603A (fr) |
SE (1) | SE7708120L (fr) |
ZA (1) | ZA774073B (fr) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0014834A1 (fr) * | 1979-01-18 | 1980-09-03 | Hoechst Aktiengesellschaft | Procédé de préparation d'amides d'acides carboxyliques et de peptides |
EP1585751A2 (fr) * | 2002-11-14 | 2005-10-19 | Celmed Oncology (USA), Inc. | Promedicaments actives par peptide deformylase |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GR73085B (fr) * | 1977-12-20 | 1984-01-31 | Hoffmann La Roche | |
CA1108125A (fr) * | 1977-12-23 | 1981-09-01 | Frank R. Atherton | Derives oligopeptides de l'acide phosphonique |
DE3368418D1 (en) * | 1982-09-17 | 1987-01-29 | Kyowa Hakko Kogyo Kk | Phosphorus-containing peptide derivative |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2298335A1 (fr) * | 1975-01-27 | 1976-08-20 | Hoffmann La Roche | Nouveaux derives de peptides d'acides phosphonique et phosphinique |
-
1977
- 1977-06-29 IT IT25208/77A patent/IT1081511B/it active
- 1977-07-06 IL IL52469A patent/IL52469A0/xx unknown
- 1977-07-06 DE DE19772730524 patent/DE2730524A1/de active Pending
- 1977-07-06 ZA ZA00774073A patent/ZA774073B/xx unknown
- 1977-07-07 AU AU26847/77A patent/AU2684777A/en active Pending
- 1977-07-08 NZ NZ184603A patent/NZ184603A/xx unknown
- 1977-07-11 JP JP8209977A patent/JPS539720A/ja active Pending
- 1977-07-11 LU LU77725A patent/LU77725A1/xx unknown
- 1977-07-11 FR FR7721280A patent/FR2358414A1/fr active Granted
- 1977-07-12 DK DK317177A patent/DK317177A/da unknown
- 1977-07-12 NL NL7707736A patent/NL7707736A/xx not_active Application Discontinuation
- 1977-07-12 SE SE7708120A patent/SE7708120L/xx unknown
- 1977-07-12 BE BE179267A patent/BE856724A/fr unknown
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2298335A1 (fr) * | 1975-01-27 | 1976-08-20 | Hoffmann La Roche | Nouveaux derives de peptides d'acides phosphonique et phosphinique |
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0014834A1 (fr) * | 1979-01-18 | 1980-09-03 | Hoechst Aktiengesellschaft | Procédé de préparation d'amides d'acides carboxyliques et de peptides |
EP1585751A2 (fr) * | 2002-11-14 | 2005-10-19 | Celmed Oncology (USA), Inc. | Promedicaments actives par peptide deformylase |
EP1585751A4 (fr) * | 2002-11-14 | 2008-08-13 | Celmed Oncology Usa Inc | Promedicaments actives par peptide deformylase |
Also Published As
Publication number | Publication date |
---|---|
NZ184603A (en) | 1980-03-05 |
IT1081511B (it) | 1985-05-21 |
ZA774073B (en) | 1978-05-30 |
FR2358414B1 (fr) | 1979-06-01 |
IL52469A0 (en) | 1977-10-31 |
LU77725A1 (fr) | 1978-09-14 |
BE856724A (fr) | 1978-01-12 |
AU2684777A (en) | 1979-01-11 |
DK317177A (da) | 1978-01-14 |
DE2730524A1 (de) | 1978-01-19 |
SE7708120L (sv) | 1978-01-14 |
JPS539720A (en) | 1978-01-28 |
NL7707736A (nl) | 1978-01-17 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |