FR2143295A1 - Thiolincosaminide derivs - useful eg as inters for lincomycin analogues - Google Patents
Thiolincosaminide derivs - useful eg as inters for lincomycin analoguesInfo
- Publication number
- FR2143295A1 FR2143295A1 FR7222565A FR7222565A FR2143295A1 FR 2143295 A1 FR2143295 A1 FR 2143295A1 FR 7222565 A FR7222565 A FR 7222565A FR 7222565 A FR7222565 A FR 7222565A FR 2143295 A1 FR2143295 A1 FR 2143295A1
- Authority
- FR
- France
- Prior art keywords
- useful
- alkyl
- lincomycin
- analogues
- residue
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
- C07H15/16—Lincomycin; Derivatives thereof
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Crystallography & Structural Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Title cpds of formula (I) and when AC is H, their acid addn salts: (where n is 1-4; Alk is not >4C alkyl or -CH2CH2OAC1; Ac and Ac1 are both H or both carboxylic acyl; R1 is not >18C satd or is not >10C unsatd aliphatic hydrocarbon, >11C aromatic hydrocarbyl or is not >8C oxa or thiacarbocyclic aromatic hydrocarbyl; and XR3 is H or residue in which X is O or S and R3 is H, carboxylic acyl, lower alkyl, alkenyl, cycloalkyl, cycloalkenyl, alkoxyalkyl or alkylthioalkyl, or Ph, Bz, furyl, furfuryl, thienyl or thenyl; when X is O and R3 is alkyl, R1 and R3 can be joined together so as to form a is not >5C oxacycloalkyl residue with 3-6 ring atoms) may be N-acylated with an L-2-pyrrolidinecarboxylic acid to give antibacterially active lincomycin analogues. The free bases of (I; Ac=Ac1-H) can be used as buffers or antacids; they may be used for modifying polyurethane resins, and their thiocyanates form corlrosion-inhibiting condensation prods with HCHO. The fluolsilicate salts are useful as mothproofing agents, and the fluoroarsenates and hexafluorophosphates are useful as pesticides.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US15610071A | 1971-06-23 | 1971-06-23 | |
| US16190971A | 1971-07-12 | 1971-07-12 | |
| US19899071A | 1971-11-15 | 1971-11-15 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2143295A1 true FR2143295A1 (en) | 1973-02-02 |
| FR2143295B1 FR2143295B1 (en) | 1977-12-23 |
Family
ID=27387802
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7222565A Granted FR2143295A1 (en) | 1971-06-23 | 1972-06-22 | Thiolincosaminide derivs - useful eg as inters for lincomycin analogues |
Country Status (14)
| Country | Link |
|---|---|
| JP (1) | JPS5724359B1 (en) |
| AR (1) | AR192797A1 (en) |
| BE (1) | BE785375A (en) |
| CA (1) | CA971956A (en) |
| CH (1) | CH587286A5 (en) |
| DE (1) | DE2229950C2 (en) |
| FI (1) | FI56688C (en) |
| FR (1) | FR2143295A1 (en) |
| IL (1) | IL39658A (en) |
| NL (1) | NL176678C (en) |
| NO (1) | NO138949C (en) |
| PH (2) | PH11975A (en) |
| SE (2) | SE384685B (en) |
| YU (1) | YU36743B (en) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE977645C (en) * | 1954-03-12 | 1967-11-30 | Brown | Return magnetic amplifier in two-way switching |
| JPS5859309A (en) * | 1981-10-02 | 1983-04-08 | Toyota Motor Corp | Structure holding monolithic catalyst |
| JPS60107313U (en) * | 1983-12-21 | 1985-07-22 | マツダ株式会社 | catalytic converter |
| JPS60159815U (en) * | 1984-04-02 | 1985-10-24 | トヨタ自動車株式会社 | Vehicle exhaust gas purification converter |
| JPS63117U (en) * | 1986-06-19 | 1988-01-05 | ||
| US7871982B2 (en) | 2005-12-09 | 2011-01-18 | Meiji Seika Kaisha, Ltd. | Lincomycin derivatives and antimicrobial agents comprising the same as active ingredient |
| JP5356223B2 (en) | 2007-05-31 | 2013-12-04 | Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 | Lincomycin derivatives and antibacterial agents containing the same as active ingredients |
| WO2008146919A1 (en) | 2007-05-31 | 2008-12-04 | Meiji Seika Kaisha, Ltd. | Lincosamide derivative, and antibacterial agent comprising the same as active ingredient |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS4839417A (en) * | 1971-06-23 | 1973-06-09 |
-
1969
- 1969-12-19 SE SE6917642A patent/SE384685B/en unknown
-
1972
- 1972-06-02 CA CA143,734A patent/CA971956A/en not_active Expired
- 1972-06-09 IL IL39658A patent/IL39658A/en unknown
- 1972-06-14 CH CH884172A patent/CH587286A5/xx not_active IP Right Cessation
- 1972-06-14 FI FI1700/72A patent/FI56688C/en active
- 1972-06-19 NL NLAANVRAGE7208333,A patent/NL176678C/en not_active IP Right Cessation
- 1972-06-20 DE DE2229950A patent/DE2229950C2/en not_active Expired
- 1972-06-22 YU YU1660/72A patent/YU36743B/en unknown
- 1972-06-22 NO NO2230/72A patent/NO138949C/en unknown
- 1972-06-22 AR AR242688A patent/AR192797A1/en active
- 1972-06-22 JP JP6190172A patent/JPS5724359B1/ja active Pending
- 1972-06-22 FR FR7222565A patent/FR2143295A1/en active Granted
- 1972-06-22 SE SE6917642A patent/SE384686B/en unknown
- 1972-06-23 PH PH13637A patent/PH11975A/en unknown
- 1972-06-23 BE BE785375A patent/BE785375A/en not_active IP Right Cessation
-
1976
- 1976-07-22 PH PH18720A patent/PH13663A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| YU36743B (en) | 1984-08-31 |
| PH11975A (en) | 1978-09-28 |
| SE384686B (en) | 1976-05-17 |
| JPS5724359B1 (en) | 1982-05-24 |
| CA971956A (en) | 1975-07-29 |
| BE785375A (en) | 1972-12-27 |
| NO138949B (en) | 1978-09-04 |
| IL39658A (en) | 1977-04-29 |
| FI56688B (en) | 1979-11-30 |
| IL39658A0 (en) | 1972-08-30 |
| FR2143295B1 (en) | 1977-12-23 |
| DE2229950A1 (en) | 1972-12-28 |
| DE2229950C2 (en) | 1983-09-15 |
| NL176678C (en) | 1985-05-17 |
| NO138949C (en) | 1978-12-13 |
| FI56688C (en) | 1980-03-10 |
| CH587286A5 (en) | 1977-04-29 |
| NL7208333A (en) | 1972-12-28 |
| PH13663A (en) | 1980-08-26 |
| SE384685B (en) | 1976-05-17 |
| AR192797A1 (en) | 1973-03-14 |
| YU166072A (en) | 1982-06-18 |
| NL176678B (en) | 1984-12-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |