FR1453246A - Benzazoles substitués en position 5 et leurs procédés de fabrication - Google Patents

Benzazoles substitués en position 5 et leurs procédés de fabrication

Info

Publication number
FR1453246A
FR1453246A FR995446A FR995446A FR1453246A FR 1453246 A FR1453246 A FR 1453246A FR 995446 A FR995446 A FR 995446A FR 995446 A FR995446 A FR 995446A FR 1453246 A FR1453246 A FR 1453246A
Authority
FR
France
Prior art keywords
benzazoles
substituted
manufacturing processes
processes
manufacturing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR995446A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Application granted granted Critical
Publication of FR1453246A publication Critical patent/FR1453246A/fr
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FR995446A 1963-11-19 1964-11-18 Benzazoles substitués en position 5 et leurs procédés de fabrication Expired FR1453246A (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US32484563A 1963-11-19 1963-11-19
US33284463A 1963-12-23 1963-12-23
US575955A US3336192A (en) 1963-11-19 1966-08-30 Anthelmintic substituted benzimidazole compositions

Publications (1)

Publication Number Publication Date
FR1453246A true FR1453246A (fr) 1966-06-03

Family

ID=27406361

Family Applications (2)

Application Number Title Priority Date Filing Date
FR995446A Expired FR1453246A (fr) 1963-11-19 1964-11-18 Benzazoles substitués en position 5 et leurs procédés de fabrication
FR5974A Expired FR4233M (fr) 1963-11-19 1965-02-17

Family Applications After (1)

Application Number Title Priority Date Filing Date
FR5974A Expired FR4233M (fr) 1963-11-19 1965-02-17

Country Status (9)

Country Link
US (1) US3336192A (fr)
BE (1) BE655924A (fr)
BR (1) BR6464278D0 (fr)
DE (1) DE1470104A1 (fr)
FR (2) FR1453246A (fr)
GB (1) GB1085634A (fr)
IL (1) IL22368A (fr)
NL (1) NL6413474A (fr)
SE (1) SE322780B (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0510235A1 (fr) * 1991-04-26 1992-10-28 Dong-A Pharm. Co., Ltd. Dérivés de benzoxazine ou de benzothiazine et leur procédé de préparation

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3471620A (en) * 1965-12-16 1969-10-07 Monsanto Chem Australia Ltd Anthelmintic compositions and methods employing 2 - (2' - thiazolin - 2' - yl)-benzimidazoles
US3625954A (en) * 1968-03-20 1971-12-07 Pfizer 1-aroylbenzimidazoles
US3864351A (en) * 1971-10-04 1975-02-04 Pfizer 1-({60 -Carboxymethoxybenzoyl-2-(2{40 -pyridyl)benzimidazoles
DE3611343A1 (de) * 1986-04-04 1987-10-08 Boehringer Mannheim Gmbh Heterocyclisch substituierte benzimidazole, verfahren zu ihrer herstellung, arzneimittel sowie zwischenprodukte
JPS6480941A (en) * 1987-09-22 1989-03-27 Fuji Photo Film Co Ltd Silver halide photographic sensitive material
FR2643903A1 (fr) * 1989-03-03 1990-09-07 Union Pharma Scient Appl Nouveaux derives de benzimidazole, leurs procedes de preparation, intermediaires de synthese, compositions pharmaceutiques les contenant, utiles notamment pour le traitement des maladies cardiovasculaires, et des ulceres duodenaux
JP2832028B2 (ja) * 1989-04-20 1998-12-02 キヤノン株式会社 化合物およびこれを含む液晶組成物およびこれを使用した液晶素子
SE9301489D0 (sv) * 1993-04-30 1993-04-30 Ab Astra Veterinary composition
KR100314351B1 (ko) * 1998-10-01 2002-03-21 민경윤 벤즈이미다졸유도체의장용성제제및그제조방법
US8501957B2 (en) * 2008-12-10 2013-08-06 China Medical University Benzimidazole compounds and their use as anticancer agents

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL264338A (fr) * 1960-05-04
US3192108A (en) * 1961-07-27 1965-06-29 Merck & Co Inc Anthelmintic compositions and method of using same

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0510235A1 (fr) * 1991-04-26 1992-10-28 Dong-A Pharm. Co., Ltd. Dérivés de benzoxazine ou de benzothiazine et leur procédé de préparation

Also Published As

Publication number Publication date
BR6464278D0 (pt) 1973-08-09
IL22368A (en) 1969-01-29
FR4233M (fr) 1966-06-20
GB1085634A (en) 1967-10-04
SE322780B (fr) 1970-04-20
NL6413474A (fr) 1965-05-20
BE655924A (fr) 1965-05-18
US3336192A (en) 1967-08-15
DE1470104A1 (de) 1969-11-13

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