FR1334957A - Procédé de préparation de nouveaux amino-pyrazoles - Google Patents

Procédé de préparation de nouveaux amino-pyrazoles

Info

Publication number
FR1334957A
FR1334957A FR885434A FR885434A FR1334957A FR 1334957 A FR1334957 A FR 1334957A FR 885434 A FR885434 A FR 885434A FR 885434 A FR885434 A FR 885434A FR 1334957 A FR1334957 A FR 1334957A
Authority
FR
France
Prior art keywords
pyrazoles
preparation
novel amino
amino
novel
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR885434A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
BASF Schweiz AG
Original Assignee
Ciba Geigy AG
Ciba AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH77061A external-priority patent/CH401071A/de
Priority claimed from CH824061A external-priority patent/CH426844A/de
Priority claimed from CH1059861A external-priority patent/CH448104A/de
Application filed by Ciba Geigy AG, Ciba AG filed Critical Ciba Geigy AG
Priority to FR890056A priority Critical patent/FR1856M/fr
Application granted granted Critical
Publication of FR1334957A publication Critical patent/FR1334957A/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/57—Nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D215/14—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR885434A 1961-01-24 1962-01-22 Procédé de préparation de nouveaux amino-pyrazoles Expired FR1334957A (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR890056A FR1856M (fr) 1961-01-24 1962-03-06 Nouvel amino-pyrazole utilisable en thérapeutique, notamment comme médicament pour le traitement des affections inflammatoires.

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
CH77061A CH401071A (de) 1961-01-24 1961-01-24 Verfahren zur Herstellung neuer Aminopyrazole
CH430561 1961-04-12
CH824061A CH426844A (de) 1961-01-24 1961-07-13 Verfahren zur Herstellung neuer Aminopyrazole
CH1059861A CH448104A (de) 1963-01-11 1961-09-13 Verfahren zur Herstellung neuer Aminopyrazole
CH1327461 1961-11-15

Publications (1)

Publication Number Publication Date
FR1334957A true FR1334957A (fr) 1963-08-16

Family

ID=27508888

Family Applications (1)

Application Number Title Priority Date Filing Date
FR885434A Expired FR1334957A (fr) 1961-01-24 1962-01-22 Procédé de préparation de nouveaux amino-pyrazoles

Country Status (5)

Country Link
US (1) US3169966A (fr)
DE (3) DE1223394B (fr)
DK (1) DK108725C (fr)
FR (1) FR1334957A (fr)
GB (1) GB937732A (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1994029300A1 (fr) * 1993-06-07 1994-12-22 Rhone Poulenc Agrochimie Fongicides pyrazoles substitues en position 3 par un heterocycle

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1252435A (fr) * 1968-02-02 1971-11-03
EP0070376A1 (fr) * 1981-07-13 1983-01-26 American Cyanamid Company Aminopyrazolines substituées par des hétérocycles
US4347251A (en) * 1981-07-13 1982-08-31 American Cyanamid Company Novel 3-substituted amino-1-substituted heteroaryl-2-pyrazolines
US4407803A (en) * 1981-08-17 1983-10-04 Abbott Laboratories Antiinflammatory 1-(quinolinyl)-2-pyrazoline derivatives
DE3132915A1 (de) * 1981-08-20 1983-03-03 Kali-Chemie Pharma Gmbh, 3000 Hannover 1,5-diphenylpyrazolin-3-on-verbindungen sowie verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3442860A1 (de) * 1984-11-24 1986-05-28 Kali-Chemie Pharma Gmbh, 3000 Hannover 5-alkyl-1-phenyl-2-piperazinoalkylpyrazolin-3- on-verbindungen sowie verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
EP1273580B1 (fr) * 2001-07-05 2005-06-15 Pfizer Products Inc. Sulfonyl heteroaryl triazoles comme agent anti-inflammatoire et analgetique
RU2005119173A (ru) * 2002-12-20 2006-02-27 Фармация Корпорейшн (Us) Ациклические пиразольные соединения
US7842810B2 (en) * 2005-03-31 2010-11-30 Janssen Pharmaceutica, Nv Bicyclic pyrazole compounds as antibacterial agents
BR112012033341B1 (pt) 2010-06-30 2022-08-23 Cyclerion Therapeutics, Inc Estimulantes de sgc
US9061030B2 (en) 2010-11-09 2015-06-23 Ironwood Pharmaceuticals, Inc. sGC stimulators
EP2797915B1 (fr) 2011-12-27 2016-07-13 Ironwood Pharmaceuticals, Inc. Dérivés de 2-bénzyl-3-(oxazole/thiazole)-5-(pyrimidin-2-yl)-1(H)-pyrazole en tant que stimulateurs de la cyclase de guanylate soluble (sGC) pour le traitement de la hypertension ou de l'insuffisance cardiaque
WO2014060381A1 (fr) * 2012-10-18 2014-04-24 Bayer Cropscience Ag Composés hétérocycliques pour la lutte contre les nuisibles

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2903460A (en) * 1956-04-07 1959-09-08 Sandoz Ag Pyrazolone derivatives
US2833779A (en) * 1956-10-29 1958-05-06 American Cyanamid Co Substituted pyrazoles
US3041343A (en) * 1959-10-14 1962-06-26 Sandoz Ltd 4-(thienyl-2'')-and 4-(pyridyl-3'')-5-aminopyrazoles

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1994029300A1 (fr) * 1993-06-07 1994-12-22 Rhone Poulenc Agrochimie Fongicides pyrazoles substitues en position 3 par un heterocycle
FR2707295A1 (fr) * 1993-06-07 1995-01-13 Rhone Poulenc Agrochimie Fongicides pyrazoles substitués en position 3 par un hétérocycle.

Also Published As

Publication number Publication date
DE1224746B (de) 1966-09-15
US3169966A (en) 1965-02-16
DK108725C (da) 1968-02-05
DE1231248B (de) 1966-12-29
DE1223394B (de) 1966-08-25
GB937732A (en) 1963-09-25

Similar Documents

Publication Publication Date Title
FR1334957A (fr) Procédé de préparation de nouveaux amino-pyrazoles
FR1503559A (fr) Procédé de préparation de nouveaux gonahexaènes
FR1318335A (fr) Procédé de préparation des permonosulfates
BE612971A (fr) Procédé de préparation de nouveaux aminopyrazoles
CH410933A (fr) Procédé de préparation de nouveaux A-nor-B-homo-6-oxo-stéroïdes
FR1250191A (fr) Procédé de préparation de tricyclodécanes nouveaux
FR1337786A (fr) Procédé de préparation de 3-(alpha-arylalcoyl)-sydnonimines
FR1295713A (fr) Procédé de préparation de nouveaux aminoacétylènes
FR1339223A (fr) Procédé de préparation de 1-oxo-2-nitratocycloalcanes
FR1310522A (fr) Procédé de préparation de 2-cyano-3-oxo-stéroïdes
FR1294974A (fr) Procédé de préparation de gallium-alkyles
FR1300297A (fr) Procédé de préparation de la méthyl-3-chromone
FR1352123A (fr) Procédé de préparation de nouveaux nitrofurfurannes
CH433273A (fr) Procédé de préparation de nouveaux A-nor-B-homo-3-oxo-stéroïdes
FR1374331A (fr) Procédé de préparation de diphénylalkylamines substituées
FR1337954A (fr) Procédé de préparation de nouveaux hydrazides
FR1291963A (fr) Procédé de préparation de polycarbodiimides
FR1339152A (fr) Procédé de préparation de nouveaux benzènesulfonyl-semicarbazides
FR1344980A (fr) Procédé de préparation de nouveaux cyclo-stéroïdes
FR1341686A (fr) Procédé de préparation de nouveaux oxydo-stéroïdes
FR1459885A (fr) Procédé de préparation de nouveaux diaza-cyclo-alcanes
FR1367071A (fr) Procédé de préparation de nouveaux 2beta-aminostéroïdes
FR1473807A (fr) Procédé de préparation de 6alpha-méthyl-16-méthylène-stéroïdes
FR1307151A (fr) Procédé de préparation de formamidochloroformamidines
FR1292112A (fr) Procédé de préparation de déhydro-stéroïdes