FI972795L - Pyrimidiinijohdannaisia - Google Patents

Pyrimidiinijohdannaisia Download PDF

Info

Publication number
FI972795L
FI972795L FI972795A FI972795A FI972795L FI 972795 L FI972795 L FI 972795L FI 972795 A FI972795 A FI 972795A FI 972795 A FI972795 A FI 972795A FI 972795 L FI972795 L FI 972795L
Authority
FI
Finland
Prior art keywords
pyrimidine derivatives
pyrimidine
derivatives
Prior art date
Application number
FI972795A
Other languages
English (en)
Swedish (sv)
Other versions
FI972795A7 (fi
FI972795A0 (fi
Inventor
Mitsuteru Hirata
Takeo Deushi
Yoshio Takahashi
Masahiro Tamura
Takeshi Ohshima
Toshiaki Oda
Hiroyuki Sonoki
Masami Shiratsuchi
Original Assignee
Kowa Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kowa Co filed Critical Kowa Co
Publication of FI972795A7 publication Critical patent/FI972795A7/fi
Publication of FI972795A0 publication Critical patent/FI972795A0/fi
Publication of FI972795L publication Critical patent/FI972795L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/69Benzenesulfonamido-pyrimidines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI972795A 1994-12-28 1995-12-19 Pyrimidiinijohdannaisia FI972795L (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP32732994 1994-12-28
JP16945495 1995-07-05
PCT/JP1995/002605 WO1996020177A1 (en) 1994-12-28 1995-12-19 Pyrimidine derivatives

Publications (3)

Publication Number Publication Date
FI972795A7 FI972795A7 (fi) 1997-06-27
FI972795A0 FI972795A0 (fi) 1997-06-27
FI972795L true FI972795L (fi) 1997-06-27

Family

ID=26492784

Family Applications (1)

Application Number Title Priority Date Filing Date
FI972795A FI972795L (fi) 1994-12-28 1995-12-19 Pyrimidiinijohdannaisia

Country Status (12)

Country Link
US (2) US6008224A (fi)
EP (1) EP0801062B1 (fi)
CN (1) CN1171785A (fi)
AT (1) ATE238285T1 (fi)
CA (1) CA2207100C (fi)
DE (1) DE69530516T2 (fi)
ES (1) ES2196090T3 (fi)
FI (1) FI972795L (fi)
HU (1) HUT77534A (fi)
NO (1) NO973001L (fi)
PT (1) PT801062E (fi)
WO (1) WO1996020177A1 (fi)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5883092A (en) * 1995-09-06 1999-03-16 Kowa Co., Ltd. Pyrimidine derivatives as endothelin antagonists
US7566452B1 (en) 1999-05-04 2009-07-28 New York University Cancer treatment with endothelin receptor antagonists
CA2315614C (en) * 1999-07-29 2004-11-02 Pfizer Inc. Pyrazoles
DE60025803T2 (de) * 2000-01-25 2006-11-02 F. Hoffmann-La Roche Ag Herstellung von sulfonamiden
US6387915B2 (en) 2000-05-31 2002-05-14 Pfizer Inc. Isoxazole-sulfonamide endothelin antagonists
US6670362B2 (en) 2000-09-20 2003-12-30 Pfizer Inc. Pyridazine endothelin antagonists
EP3836941A4 (en) 2018-08-14 2022-05-18 Tosk, Inc. METHODS AND COMPOSITIONS FOR THE TREATMENT OF MUCOSITIS
WO2020036975A1 (en) 2018-08-14 2020-02-20 Tosk, Inc. Methods and compositions for reducing fluorouracil induced toxicity
WO2020036974A1 (en) 2018-08-14 2020-02-20 Tosk, Inc. Methods and compositions for reducing radiation induced toxicity
US11446303B2 (en) 2019-06-21 2022-09-20 Tosk, Inc. Uridine phosphorylase (UPase) inhibitors for treatment of liver conditions
IL299703A (en) 2020-07-07 2023-03-01 Tosk Inc Uridine phosphorylase inhibitors for the treatment or prevention of lung disease

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2086544C1 (ru) * 1991-06-13 1997-08-10 Хоффманн-Ля Рош АГ Бензолсульфонамидные производные пиримидина или их соли, фармацевтическая композиция для лечения заболеваний, связанных с активностью эндотелина
TW394761B (en) * 1993-06-28 2000-06-21 Hoffmann La Roche Novel Sulfonylamino Pyrimidines
IL111959A (en) * 1993-12-17 2000-07-16 Tanabe Seiyaku Co N-(polysubstituted pyrimidin-4-yl) benzenesulfonamide derivatives their preparation and pharmaceutical compositions containing them
US5883092A (en) * 1995-09-06 1999-03-16 Kowa Co., Ltd. Pyrimidine derivatives as endothelin antagonists

Also Published As

Publication number Publication date
NO973001L (no) 1997-08-27
US6337334B1 (en) 2002-01-08
AU4190096A (en) 1996-07-19
DE69530516D1 (de) 2003-05-28
HUT77534A (hu) 1998-05-28
EP0801062A4 (en) 1998-04-29
EP0801062B1 (en) 2003-04-23
PT801062E (pt) 2003-08-29
WO1996020177A1 (en) 1996-07-04
CA2207100C (en) 2008-02-19
FI972795A7 (fi) 1997-06-27
ATE238285T1 (de) 2003-05-15
ES2196090T3 (es) 2003-12-16
CN1171785A (zh) 1998-01-28
CA2207100A1 (en) 1996-07-04
DE69530516T2 (de) 2003-12-24
FI972795A0 (fi) 1997-06-27
AU696216B2 (en) 1998-09-03
US6008224A (en) 1999-12-28
NO973001D0 (no) 1997-06-27
EP0801062A1 (en) 1997-10-15

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