FI955523A0 - 1-(2-bentsimidatsolyyli)-1,5-diatsasyklo-oksataaniyhdisteet - Google Patents
1-(2-bentsimidatsolyyli)-1,5-diatsasyklo-oksataaniyhdisteetInfo
- Publication number
- FI955523A0 FI955523A0 FI955523A FI955523A FI955523A0 FI 955523 A0 FI955523 A0 FI 955523A0 FI 955523 A FI955523 A FI 955523A FI 955523 A FI955523 A FI 955523A FI 955523 A0 FI955523 A0 FI 955523A0
- Authority
- FI
- Finland
- Prior art keywords
- diazacyklo
- benzimidazolyl
- octane compounds
- octane
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP15599593 | 1993-05-20 | ||
PCT/JP1994/000787 WO1994027973A1 (fr) | 1993-05-20 | 1994-05-16 | Derive 1-(2-benzimidazolyl)-1,5-diazacyclooctane |
Publications (2)
Publication Number | Publication Date |
---|---|
FI955523A FI955523A (fi) | 1995-11-16 |
FI955523A0 true FI955523A0 (fi) | 1995-11-16 |
Family
ID=15618048
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI955523A FI955523A0 (fi) | 1993-05-20 | 1995-11-16 | 1-(2-bentsimidatsolyyli)-1,5-diatsasyklo-oksataaniyhdisteet |
Country Status (7)
Country | Link |
---|---|
US (1) | US5624948A (fi) |
EP (1) | EP0699668A4 (fi) |
KR (1) | KR960702445A (fi) |
CA (1) | CA2161876A1 (fi) |
FI (1) | FI955523A0 (fi) |
NO (1) | NO954654L (fi) |
WO (1) | WO1994027973A1 (fi) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6423704B2 (en) | 1995-12-20 | 2002-07-23 | Aventis Pharmaceuticals Inc. | Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic diseases |
ATE221883T1 (de) * | 1995-12-20 | 2002-08-15 | Aventis Pharma Inc | Substituierte 4-(1h-benzimidazol-2-yl)(1, 4)diazepane für die behandlung von allergischen krankheiten |
US6194406B1 (en) | 1995-12-20 | 2001-02-27 | Aventis Pharmaceuticals Inc. | Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic disease |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1140119A (en) * | 1978-04-03 | 1983-01-25 | Joseph Torremans | N-heterocyclyl-4-piperidinamines |
JPS5879983A (ja) * | 1981-11-06 | 1983-05-13 | Kanebo Ltd | 新規なベンズイミダゾ−ル誘導体、その製造法およびその医薬組成物 |
US4588722A (en) * | 1984-01-09 | 1986-05-13 | Janssen Pharmaceutica N.V. | N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives |
US4835161A (en) * | 1986-02-03 | 1989-05-30 | Janssen Pharmaceutica N.V. | Anti-histaminic compositions containing n-heterocyclyl-4-piperidinamines |
EP0232937B1 (en) * | 1986-02-03 | 1992-08-19 | Janssen Pharmaceutica N.V. | Anti-histaminic compositions containing n-heterocyclyl-4-piperidinamines |
US4943580A (en) * | 1987-03-09 | 1990-07-24 | Janssen Pharmaceutica N.V. | Anti-histaminic benzimidazole, imidazopyridine and purine derivatives |
US4988689A (en) * | 1987-07-01 | 1991-01-29 | Janssen Pharmaceutica N.V. | ((Pharmacologically active bicyclic heterocyclic)methyl and -heteroatom) substituted hexahydro-1H-azepines and pyrrolidines |
FR2668150B1 (fr) * | 1990-10-17 | 1994-11-18 | Theramex | Nouveaux derives du terbutylphenyl 1-amino 4-hydroxybutane, leurs procedes de preparation et les compositions pharmaceutiques en renfermant. |
-
1994
- 1994-05-16 US US08/537,747 patent/US5624948A/en not_active Expired - Fee Related
- 1994-05-16 EP EP94914624A patent/EP0699668A4/en not_active Withdrawn
- 1994-05-16 KR KR1019950704962A patent/KR960702445A/ko not_active Application Discontinuation
- 1994-05-16 WO PCT/JP1994/000787 patent/WO1994027973A1/ja not_active Application Discontinuation
- 1994-05-16 CA CA002161876A patent/CA2161876A1/en not_active Abandoned
-
1995
- 1995-11-16 FI FI955523A patent/FI955523A0/fi unknown
- 1995-11-17 NO NO954654A patent/NO954654L/no unknown
Also Published As
Publication number | Publication date |
---|---|
KR960702445A (ko) | 1996-04-27 |
CA2161876A1 (en) | 1994-12-08 |
EP0699668A1 (en) | 1996-03-06 |
FI955523A (fi) | 1995-11-16 |
US5624948A (en) | 1997-04-29 |
NO954654D0 (no) | 1995-11-17 |
WO1994027973A1 (fr) | 1994-12-08 |
EP0699668A4 (en) | 1996-09-18 |
NO954654L (no) | 1996-01-22 |
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