FI940186A - 9H-imidatso/1,2-a/bentsimidatsoli-3-asetamidijohdannaisia, niiden valmistus ja niiden käyttö terapiassa - Google Patents

9H-imidatso/1,2-a/bentsimidatsoli-3-asetamidijohdannaisia, niiden valmistus ja niiden käyttö terapiassa Download PDF

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Publication number
FI940186A
FI940186A FI940186A FI940186A FI940186A FI 940186 A FI940186 A FI 940186A FI 940186 A FI940186 A FI 940186A FI 940186 A FI940186 A FI 940186A FI 940186 A FI940186 A FI 940186A
Authority
FI
Finland
Prior art keywords
imidazo
benzimidazole
therapy
preparation
acetamide derivatives
Prior art date
Application number
FI940186A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI940186A0 (fi
Inventor
Pascal George
Peretti Danielle De
Jocelyne Roy
Jean-Paul Schmitt
Mireille Sevrin
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9300337A external-priority patent/FR2700544B1/fr
Priority claimed from FR9309013A external-priority patent/FR2707987B1/fr
Application filed by Synthelabo filed Critical Synthelabo
Publication of FI940186A0 publication Critical patent/FI940186A0/fi
Publication of FI940186A publication Critical patent/FI940186A/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI940186A 1993-01-15 1994-01-14 9H-imidatso/1,2-a/bentsimidatsoli-3-asetamidijohdannaisia, niiden valmistus ja niiden käyttö terapiassa FI940186A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9300337A FR2700544B1 (fr) 1993-01-15 1993-01-15 Dérivés de 9H-imidazo[1,2-a]benzimidazole-3-acétamide, leur préparation et leur application en thérapeutique.
FR9309013A FR2707987B1 (fr) 1993-07-22 1993-07-22 Dérivés de 9H-imidazo[1,2-a]benzimidazole-3-acétamide, leur préparation et leur application en thérapeutique .

Publications (2)

Publication Number Publication Date
FI940186A0 FI940186A0 (fi) 1994-01-14
FI940186A true FI940186A (fi) 1994-07-16

Family

ID=26230029

Family Applications (1)

Application Number Title Priority Date Filing Date
FI940186A FI940186A (fi) 1993-01-15 1994-01-14 9H-imidatso/1,2-a/bentsimidatsoli-3-asetamidijohdannaisia, niiden valmistus ja niiden käyttö terapiassa

Country Status (16)

Country Link
US (1) US5466706A (zh)
EP (1) EP0607076A1 (zh)
JP (1) JPH06271575A (zh)
CN (1) CN1097743A (zh)
AU (1) AU665137B2 (zh)
CA (1) CA2113490A1 (zh)
CZ (1) CZ9394A3 (zh)
FI (1) FI940186A (zh)
HU (1) HUT70407A (zh)
IL (1) IL108343A0 (zh)
NO (1) NO940130L (zh)
NZ (1) NZ250679A (zh)
PL (1) PL301901A1 (zh)
RU (1) RU94000725A (zh)
SK (1) SK4694A3 (zh)
TW (1) TW253886B (zh)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2719843B1 (fr) * 1994-05-10 1996-06-07 Synthelabo Dérivés de 5,6-dihydro-4h-imidazo [2',1':2,3] imidazo-[4,5,1-ij] quinoléine et de 4,5-dihydroimidazo [1,2-a] pyrrolo-[1,2,3-cd] benzimidazole, leur préparation et leur application en thérapeutique.
FR2741073B1 (fr) * 1995-11-09 1997-12-12 Synthelabo Derives de 4,5-dihydroimidazo(1,2-a)pyrrolo(1,2,3-cd) benzimidazole, leur preparation et leur application en therapeutique
GB9702524D0 (en) * 1997-02-07 1997-03-26 Merck Sharp & Dohme Therapeutic agents
FR2759698B1 (fr) * 1997-02-20 1999-03-19 Synthelabo Derives de 1,4-diphenylimidazole-5-acetamide, leur preparation et leur application en therapeutique
JP2004509103A (ja) * 2000-09-11 2004-03-25 セプレイコー　インコーポレイテッド モノアミン受容体及び輸送体のリガンドならびにその使用方法
KR20040034594A (ko) * 2001-01-26 2004-04-28 브리스톨-마이어스스퀴브컴파니 코르티코트로핀 방출 인자 억제제로서의 이미다졸릴 유도체
MXPA05006438A (es) * 2002-12-18 2005-09-08 Mallinckrodt Inc Derivados de acetamidas de heteroarilo.
FR2870239B1 (fr) 2004-05-11 2006-06-16 Sanofi Synthelabo Derives de carbamate de 2h- ou 3h-benzo[e]indazol-1-yle, leur preparation et leur application en therapeutique.
US7498439B2 (en) * 2004-06-22 2009-03-03 Mallinckrodt Inc. Synthesis of heteroaryl acetamides from reaction mixtures having reduced water content
DK2001892T3 (da) 2006-03-17 2013-07-01 Ambit Biosciences Corp Imidazolthiazolforbindelser til behandling af proliferative sygdomme
CN101868465B (zh) 2007-09-19 2013-12-25 埃姆比特生物科学公司 包含N-(5-叔丁基-异噁唑-3-基)-N’-{4-[7-(2-吗啉-4-基-乙氧基)咪唑并[2，1-b][1，3]苯并噻唑-2-基]苯基}脲的固体形式、其组合物及其应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3732243A (en) * 1970-06-23 1973-05-08 Sankyo Co 2-(p-bromophenyl)-9-dimethyl-amino-propyl-9h-imidazo(1,2-a)benzimidazole
GB1484615A (en) * 1974-11-23 1977-09-01 Lepetit Spa Tricyclic n-containing derivatives
FR2568879B1 (fr) * 1984-08-07 1986-12-12 Synthelabo Imidazo(1,2-a)quinolines, leur preparation et leur application en therapeutique
US4675323A (en) * 1985-08-06 1987-06-23 Synthelabo Imidazo(1,2-a)quinoline derivatives useful as anxiolytic agents
US5240944A (en) * 1988-12-28 1993-08-31 Kotobuki Seiyaku Co. Ltd. Cyclic guanidine derivatives, anti-ulceratives and method of manufacturing the same

Also Published As

Publication number Publication date
AU5317794A (en) 1995-05-25
PL301901A1 (en) 1994-07-25
NO940130D0 (no) 1994-01-14
SK4694A3 (en) 1995-02-08
NO940130L (no) 1994-07-18
US5466706A (en) 1995-11-14
IL108343A0 (en) 1994-04-12
CZ9394A3 (en) 1994-08-17
JPH06271575A (ja) 1994-09-27
CA2113490A1 (en) 1994-07-16
TW253886B (zh) 1995-08-11
HU9400109D0 (en) 1994-05-30
AU665137B2 (en) 1995-12-14
RU94000725A (ru) 1997-05-27
CN1097743A (zh) 1995-01-25
NZ250679A (en) 1995-07-26
HUT70407A (en) 1995-10-30
FI940186A0 (fi) 1994-01-14
EP0607076A1 (fr) 1994-07-20

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