FI924230A7 - Substituoituja pyridinyyliamino-1H-indoleja, -1H-indatsoleja,-2H-indatsoleja, -bentso(b)tiofeeneja ja -1,2-bentsoisotiatsoleja, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä - Google Patents
Substituoituja pyridinyyliamino-1H-indoleja, -1H-indatsoleja,-2H-indatsoleja, -bentso(b)tiofeeneja ja -1,2-bentsoisotiatsoleja, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä Download PDFInfo
- Publication number
- FI924230A7 FI924230A7 FI924230A FI924230A FI924230A7 FI 924230 A7 FI924230 A7 FI 924230A7 FI 924230 A FI924230 A FI 924230A FI 924230 A FI924230 A FI 924230A FI 924230 A7 FI924230 A7 FI 924230A7
- Authority
- FI
- Finland
- Prior art keywords
- indazoles
- benzoisothiazoles
- thiophenes
- indoles
- medicaments
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/764,031 US5185350A (en) | 1991-09-23 | 1991-09-23 | Substituted pyridinylamino-1h-indoles,1h-indazoles,2h-indazoles, benzo (b)thiophenes and 1,2-benzisothiazoles |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI924230A0 FI924230A0 (fi) | 1992-09-21 |
| FI924230L FI924230L (fi) | 1993-03-24 |
| FI924230A7 true FI924230A7 (fi) | 1993-03-24 |
Family
ID=25069502
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI924230A FI924230A7 (fi) | 1991-09-23 | 1992-09-21 | Substituoituja pyridinyyliamino-1H-indoleja, -1H-indatsoleja,-2H-indatsoleja, -bentso(b)tiofeeneja ja -1,2-bentsoisotiatsoleja, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä |
Country Status (18)
| Country | Link |
|---|---|
| US (2) | US5185350A (enExample) |
| EP (1) | EP0534343B1 (enExample) |
| JP (1) | JP2961023B2 (enExample) |
| KR (1) | KR930006006A (enExample) |
| AT (1) | ATE160346T1 (enExample) |
| AU (1) | AU653263B2 (enExample) |
| CA (1) | CA2078814C (enExample) |
| CZ (1) | CZ290692A3 (enExample) |
| DE (1) | DE69223205T2 (enExample) |
| DK (1) | DK0534343T3 (enExample) |
| ES (1) | ES2111025T3 (enExample) |
| FI (1) | FI924230A7 (enExample) |
| GR (1) | GR3025774T3 (enExample) |
| HU (1) | HUT64055A (enExample) |
| IL (1) | IL103232A0 (enExample) |
| MX (1) | MX9205374A (enExample) |
| NO (1) | NO923686L (enExample) |
| TW (1) | TW207539B (enExample) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0550507A1 (en) * | 1990-09-13 | 1993-07-14 | Beecham Group p.l.c. | Indole ureas as 5 ht receptor antagonist |
| US5356910A (en) | 1993-07-19 | 1994-10-18 | Hoechst-Roussel Pharmaceuticals Inc. | Use of N-(pyridinyl)-1H-indol-1-amines for the treatment of obsessive-compulsive disorder |
| CA2176127A1 (en) * | 1993-12-21 | 1995-06-29 | William Henry Walker Lunn | Methods for the treatment or prevention of conditions associated with amyloidogenic reptides |
| DE19626373A1 (de) * | 1996-07-02 | 1998-01-08 | Boehringer Ingelheim Kg | Neuartige Verwendung von Wirkstoffen, welche die Funktion von nichtneuronalem Acetylcholin beeinflussen |
| TW200302722A (en) * | 2002-02-13 | 2003-08-16 | Astrazeneca Ab | Therapeutic agents |
| US20050222123A1 (en) | 2004-01-27 | 2005-10-06 | North Shore-Long Island Jewish Research Institute | Cholinesterase inhibitors for treating inflammation |
| EP1718638A4 (en) | 2004-02-20 | 2009-04-22 | Smithkline Beecham Corp | NEW COMPOUNDS |
| JP4787471B2 (ja) * | 2004-05-21 | 2011-10-05 | 株式会社ポッカコーポレーション | 脳機能亢進剤 |
| JP4698671B2 (ja) | 2004-06-01 | 2011-06-08 | エフ.ホフマン−ラ ロシュ アーゲー | モノアミン再取り込み阻害剤としての3−アミノ−1−アリールプロピルインドール |
| EP2351737A1 (en) * | 2005-11-30 | 2011-08-03 | F. Hoffmann-La Roche AG | 3-Amino-1-arylpropyl indoles and aza-substituted indoles |
| JP2009517432A (ja) | 2005-11-30 | 2009-04-30 | エフ.ホフマン−ラ ロシュ アーゲー | 3−アミノ−2−アリールプロピルアザインドールおよびその使用 |
| RU2008120138A (ru) * | 2005-11-30 | 2010-01-10 | Ф. Хоффманн-Ля Рош Аг (Ch) | 3-амино-1-арилпропилиндолы и аза-замещенные индолы |
| KR102534969B1 (ko) * | 2021-08-20 | 2023-05-26 | 김수영 | 포켓 인슐레이터 및 이를 포함하는 단열체 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE115143T1 (de) * | 1987-04-24 | 1994-12-15 | Hoechst Roussel Pharma | N-(pyridinyl)-1h-indol-1-amine, verfahren zu deren herstellung und ihre verwendung als arzneimittel. |
| US4970219A (en) * | 1989-06-28 | 1990-11-13 | Hoechst-Roussel Pharmaceuticals Inc. | Heteroarylamino- and heteroaryloxypyridinamine compounds which have useful utility in treating skin disorders |
| US4983615A (en) * | 1989-06-28 | 1991-01-08 | Hoechst-Roussel Pharmaceuticals Inc. | Heteroarylamino- and heteroaryloxypyridinamine compounds which are useful in treating skin disorders |
| US5006537A (en) * | 1989-08-02 | 1991-04-09 | Hoechst-Roussel Pharmaceuticals, Inc. | 1,3-dihydro-1-(pyridinylamino)-2H-indol-2-ones |
| US5177088A (en) * | 1991-04-17 | 1993-01-05 | Hoechst-Roussel Pharmaceuticals Incorporated | Substituted 3-(pyridinylamino)-indoles |
-
1991
- 1991-09-23 US US07/764,031 patent/US5185350A/en not_active Expired - Fee Related
-
1992
- 1992-09-10 TW TW081107145A patent/TW207539B/zh active
- 1992-09-21 DK DK92116110T patent/DK0534343T3/da active
- 1992-09-21 ES ES92116110T patent/ES2111025T3/es not_active Expired - Lifetime
- 1992-09-21 FI FI924230A patent/FI924230A7/fi unknown
- 1992-09-21 DE DE69223205T patent/DE69223205T2/de not_active Expired - Fee Related
- 1992-09-21 EP EP92116110A patent/EP0534343B1/en not_active Expired - Lifetime
- 1992-09-21 AT AT92116110T patent/ATE160346T1/de not_active IP Right Cessation
- 1992-09-21 IL IL103232A patent/IL103232A0/xx unknown
- 1992-09-22 AU AU25297/92A patent/AU653263B2/en not_active Expired - Fee Related
- 1992-09-22 MX MX9205374A patent/MX9205374A/es not_active IP Right Cessation
- 1992-09-22 KR KR1019920017238A patent/KR930006006A/ko not_active Withdrawn
- 1992-09-22 CZ CS922906A patent/CZ290692A3/cs unknown
- 1992-09-22 CA CA002078814A patent/CA2078814C/en not_active Expired - Lifetime
- 1992-09-22 HU HU9203023A patent/HUT64055A/hu unknown
- 1992-09-22 JP JP4251779A patent/JP2961023B2/ja not_active Expired - Fee Related
- 1992-09-22 NO NO92923686A patent/NO923686L/no unknown
-
1993
- 1993-03-25 US US08/038,317 patent/US5328918A/en not_active Expired - Lifetime
-
1997
- 1997-12-23 GR GR970403425T patent/GR3025774T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI924230A0 (fi) | 1992-09-21 |
| US5185350A (en) | 1993-02-09 |
| EP0534343A1 (en) | 1993-03-31 |
| DE69223205T2 (de) | 1998-05-14 |
| AU653263B2 (en) | 1994-09-22 |
| DK0534343T3 (da) | 1998-07-27 |
| US5328918A (en) | 1994-07-12 |
| JP2961023B2 (ja) | 1999-10-12 |
| CA2078814C (en) | 2003-09-09 |
| NO923686L (no) | 1993-03-24 |
| JPH061787A (ja) | 1994-01-11 |
| IL103232A0 (en) | 1993-02-21 |
| CZ290692A3 (en) | 1993-04-14 |
| TW207539B (enExample) | 1993-06-11 |
| ES2111025T3 (es) | 1998-03-01 |
| FI924230L (fi) | 1993-03-24 |
| HU9203023D0 (en) | 1993-11-29 |
| EP0534343B1 (en) | 1997-11-19 |
| ATE160346T1 (de) | 1997-12-15 |
| CA2078814A1 (en) | 1993-03-24 |
| DE69223205D1 (de) | 1998-01-02 |
| GR3025774T3 (en) | 1998-03-31 |
| AU2529792A (en) | 1993-03-25 |
| KR930006006A (ko) | 1993-04-20 |
| HUT64055A (en) | 1993-11-29 |
| MX9205374A (es) | 1993-03-01 |
| NO923686D0 (no) | 1992-09-22 |
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