FI914611L - 2-aminopyrimidin-4 -karboxamidderivat, framstaellning och terapeutisk anvaendning av dem. - Google Patents

2-aminopyrimidin-4 -karboxamidderivat, framstaellning och terapeutisk anvaendning av dem. Download PDF

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Publication number
FI914611L
FI914611L FI914611A FI914611A FI914611L FI 914611 L FI914611 L FI 914611L FI 914611 A FI914611 A FI 914611A FI 914611 A FI914611 A FI 914611A FI 914611 L FI914611 L FI 914611L
Authority
FI
Finland
Prior art keywords
carboxamider
anvaendning
aminopyrimidin
dem
therapeutic
Prior art date
Application number
FI914611A
Other languages
English (en)
Finnish (fi)
Other versions
FI914611A7 (fi
FI914611A0 (fi
Inventor
Pascal George
Christian Maloizel
Benoit Marabout
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of FI914611A0 publication Critical patent/FI914611A0/fi
Publication of FI914611A7 publication Critical patent/FI914611A7/fi
Publication of FI914611L publication Critical patent/FI914611L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
FI914611A 1990-10-02 1991-10-01 2-aminopyrimidin-4 -karboxamidderivat, framstaellning och terapeutisk anvaendning av dem. FI914611L (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9012094A FR2667317B1 (fr) 1990-10-02 1990-10-02 Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.

Publications (3)

Publication Number Publication Date
FI914611A0 FI914611A0 (fi) 1991-10-01
FI914611A7 FI914611A7 (fi) 1992-04-03
FI914611L true FI914611L (fi) 1992-04-03

Family

ID=9400824

Family Applications (1)

Application Number Title Priority Date Filing Date
FI914611A FI914611L (fi) 1990-10-02 1991-10-01 2-aminopyrimidin-4 -karboxamidderivat, framstaellning och terapeutisk anvaendning av dem.

Country Status (18)

Country Link
US (1) US5210086A (cs)
EP (1) EP0480794A1 (cs)
JP (1) JPH04273870A (cs)
KR (1) KR920008033A (cs)
AU (1) AU637261B2 (cs)
CA (1) CA2052609A1 (cs)
CS (1) CS299991A3 (cs)
FI (1) FI914611L (cs)
FR (1) FR2667317B1 (cs)
HU (1) HUT59392A (cs)
IE (1) IE913459A1 (cs)
IL (1) IL99612A0 (cs)
MX (1) MX9101341A (cs)
NO (1) NO913843L (cs)
NZ (1) NZ240055A (cs)
PL (1) PL291886A1 (cs)
PT (1) PT99138A (cs)
ZA (1) ZA917853B (cs)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0522914A1 (fr) * 1991-06-27 1993-01-13 Synthelabo Dérivés de 2-pipéridinylpyrimidine-4-carboxamide, leur préparation et leur application en thérapeutique
DK0520882T3 (da) * 1991-06-27 1995-12-11 Synthelabo Derivater af 2-aminopyrimidin-4-carboxamid, deres fremstilling og deres terapeutiske anvendelse
FR2691148B1 (fr) * 1992-05-18 1994-07-01 Synthelabo Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.
FR2691147B1 (fr) * 1992-05-18 1994-07-01 Synthelabo Derives de 2-piperidinylpyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.
FR2713225B1 (fr) * 1993-12-02 1996-03-01 Sanofi Sa N-pipéridino-3-pyrazolecarboxamide substitué.
FR2699171B1 (fr) * 1992-12-14 1995-02-03 Synthelabo Dérivés de 2-amino-N[[[4-aminocarbonyl) pyrimidin-2-yl]amino]alkyl]pyrimidine-4-carboxamide, leur préparation et leur application en thérapeutique.
FR2693195B1 (fr) * 1992-07-03 1994-09-23 Synthelabo Dérivés de 2-amino-N-[[[(4-aminocarbonyl)pyrimidin-2-yl]amino]alkyl] pyrimidine-4-carboxamide, leur préparation et leur application en thérapeutique.
ES2073951T3 (es) * 1992-07-03 1995-08-16 Synthelabo Derivados de 2-amino-n-(((4-(aminocarbonil)pirimidin-2-il)amino)alquil)pirimidina-4-carboxamida, su preparacion y su aplicacion en terapeutica.
FR2697253B1 (fr) * 1992-10-22 1994-12-02 Synthelabo Dérivés de 2-aminopyrimidine-4-carboxamide, leur préparation et leur application en thérapeutique.
WO1995002419A1 (fr) * 1993-07-14 1995-01-26 Yamanouchi Pharmaceutical Co., Ltd. Remede agissant contre le dysfonctionnement urinaire associe a l'hypertrophie de la prostate
FR2724382B1 (fr) * 1994-09-13 1996-10-18 Synthelabo Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique
FR2724383B1 (fr) * 1994-09-13 1996-10-18 Synthelabo Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique
CA2232147A1 (en) * 1997-04-03 1998-10-03 F. Hoffmann-La Roche Ag Phenoxymethyl piperidine derivatives
US6110937A (en) 1997-04-03 2000-08-29 Syntex Usa, Inc. Phenoxymethyl piperidine derivatives for the treatment of neuropathic pain
TR200102800T2 (tr) 1999-03-26 2002-01-21 Astrazeneca Ab Yeni bileşikler.
GB0013060D0 (en) * 2000-05-31 2000-07-19 Astrazeneca Ab Chemical compounds
GB0021670D0 (en) * 2000-09-04 2000-10-18 Astrazeneca Ab Chemical compounds
EP1318988A2 (en) * 2000-09-11 2003-06-18 Sepracor, Inc. Ligands for monoamine receptors and transporters, and methods of use thereof (neurotransmission)
GB0117899D0 (en) * 2001-07-23 2001-09-12 Astrazeneca Ab Chemical compounds
SE0102809D0 (sv) * 2001-08-22 2001-08-22 Astrazeneca Ab Novel compounds

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3290317A (en) * 1960-03-07 1966-12-06 Sterling Drug Inc 1-(nu-aryl-nu-alkanoylaminoalkyl)-4-aryl-4-piperidinols and their esters
GB1203149A (en) * 1968-06-10 1970-08-26 Ici Ltd Piperidine derivatives
GB1280699A (en) * 1968-12-23 1972-07-05 Robins Co Inc A H 0-substituted-4-phenoxypiperidines
DE2143730A1 (de) * 1971-09-01 1973-03-08 Byk Gulden Lomberg Chem Fab Substituierte pyridine, verfahren zu deren herstellung und sie enthaltende arzneimittel
US4031221A (en) * 1974-06-17 1977-06-21 American Hoechst Corporation Method of treating pain and hypertension
DE2549999A1 (de) * 1975-11-07 1977-05-12 Boehringer Mannheim Gmbh Piperidin-derivate und verfahren zu ihrer herstellung
DE2737630A1 (de) * 1977-08-20 1979-03-01 Boehringer Mannheim Gmbh Neue aminopropanolderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
FR2618436B1 (fr) * 1987-07-23 1989-10-27 Synthelabo Derives de piperidine, leur preparation et leur application en therapeutique
FR2644786B1 (fr) * 1989-03-21 1993-12-31 Adir Cie Nouveaux derives fluoro-4 benzoiques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent
FR2656609B1 (fr) * 1989-12-28 1992-03-27 Synthelabo Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.

Also Published As

Publication number Publication date
NO913843D0 (no) 1991-10-01
US5210086A (en) 1993-05-11
FI914611A7 (fi) 1992-04-03
FI914611A0 (fi) 1991-10-01
FR2667317B1 (fr) 1992-12-04
FR2667317A1 (fr) 1992-04-03
HU913137D0 (en) 1992-01-28
EP0480794A1 (fr) 1992-04-15
AU8487191A (en) 1992-04-09
ZA917853B (en) 1992-07-29
IL99612A0 (en) 1992-08-18
NZ240055A (en) 1992-09-25
KR920008033A (ko) 1992-05-27
NO913843L (no) 1992-04-03
IE913459A1 (en) 1992-04-08
CA2052609A1 (en) 1992-04-03
CS299991A3 (en) 1992-04-15
MX9101341A (es) 1992-06-05
PL291886A1 (en) 1992-07-27
HUT59392A (en) 1992-05-28
JPH04273870A (ja) 1992-09-30
PT99138A (pt) 1993-12-31
AU637261B2 (en) 1993-05-20

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