FI863353A - Gem-dihalogen- och gem-tetrahalogen-1,2-diamino-4,9-diazadodekaner. - Google Patents

Gem-dihalogen- och gem-tetrahalogen-1,2-diamino-4,9-diazadodekaner. Download PDF

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Publication number
FI863353A
FI863353A FI863353A FI863353A FI863353A FI 863353 A FI863353 A FI 863353A FI 863353 A FI863353 A FI 863353A FI 863353 A FI863353 A FI 863353A FI 863353 A FI863353 A FI 863353A
Authority
FI
Finland
Prior art keywords
gem
diazadodecaner
tetrahalogen
dihalogen
diamino
Prior art date
Application number
FI863353A
Other languages
English (en)
Other versions
FI84817B (fi
FI84817C (fi
FI863353A0 (fi
Inventor
Fritz Gerhart
Pierre Mamont
Original Assignee
Merrell Dow Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma
Publication of FI863353A0 publication Critical patent/FI863353A0/fi
Publication of FI863353A publication Critical patent/FI863353A/fi
Publication of FI84817B publication Critical patent/FI84817B/fi
Application granted granted Critical
Publication of FI84817C publication Critical patent/FI84817C/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/02Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C211/15Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
FI863353A 1985-08-21 1986-08-19 Foerfarande foer framstaellning av en terapeutiskt aktiv gem-6,6-difluor-1,12-diamino-4,9-diazadodekan. FI84817C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76793485A 1985-08-21 1985-08-21
US76793485 1985-08-21

Publications (4)

Publication Number Publication Date
FI863353A0 FI863353A0 (fi) 1986-08-19
FI863353A true FI863353A (fi) 1987-02-22
FI84817B FI84817B (fi) 1991-10-15
FI84817C FI84817C (fi) 1992-01-27

Family

ID=25081013

Family Applications (1)

Application Number Title Priority Date Filing Date
FI863353A FI84817C (fi) 1985-08-21 1986-08-19 Foerfarande foer framstaellning av en terapeutiskt aktiv gem-6,6-difluor-1,12-diamino-4,9-diazadodekan.

Country Status (19)

Country Link
EP (1) EP0220409B1 (fi)
JP (2) JPH0660131B2 (fi)
KR (1) KR900006124B1 (fi)
CN (1) CN1012815B (fi)
AR (1) AR242554A1 (fi)
AT (1) ATE69801T1 (fi)
AU (1) AU585052B2 (fi)
CA (1) CA1274547C (fi)
DE (1) DE3682652D1 (fi)
DK (1) DK396786A (fi)
ES (1) ES2001247A6 (fi)
FI (1) FI84817C (fi)
GR (1) GR862148B (fi)
HU (1) HUT44754A (fi)
IL (1) IL79753A0 (fi)
NO (1) NO164973C (fi)
NZ (1) NZ217247A (fi)
PT (1) PT83232B (fi)
ZA (1) ZA866180B (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4695654A (en) * 1985-08-21 1987-09-22 Merrell Dow Pharmaceuticals Inc. Gem-dihalo-1,8-diamino-4-aza-octanes
JPH06181890A (ja) * 1992-10-06 1994-07-05 Terumo Corp Mri造影剤
KR101286158B1 (ko) * 2011-08-24 2013-07-15 씨제이제일제당 (주) 발효액에서 1,4-디아미노부탄의 분리 및 정제하는 방법
CN109456198A (zh) * 2018-11-14 2019-03-12 上海阿拉丁生化科技股份有限公司 一种2,2`-二氨基-n-甲基二乙胺的合成方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4004996A (en) * 1974-12-23 1977-01-25 Merck & Co., Inc. Fluorination of organic compounds
GB2082579B (en) * 1980-08-23 1984-02-08 Merrell Toraude & Co Fluorinated diaminobutane derivatives
US4695654A (en) * 1985-08-21 1987-09-22 Merrell Dow Pharmaceuticals Inc. Gem-dihalo-1,8-diamino-4-aza-octanes

Also Published As

Publication number Publication date
CN1012815B (zh) 1991-06-12
KR900006124B1 (ko) 1990-08-24
NO863344L (no) 1987-02-23
DE3682652D1 (de) 1992-01-09
GR862148B (en) 1986-12-23
JPH072741A (ja) 1995-01-06
CA1274547A (en) 1990-09-25
CN86105088A (zh) 1987-04-29
JPH0660131B2 (ja) 1994-08-10
ATE69801T1 (de) 1991-12-15
JPS6245565A (ja) 1987-02-27
JPH0798777B2 (ja) 1995-10-25
AU6155786A (en) 1987-02-26
NZ217247A (en) 1989-10-27
EP0220409B1 (en) 1991-11-27
AR242554A1 (es) 1993-04-30
NO863344D0 (no) 1986-08-20
HUT44754A (en) 1988-04-28
PT83232A (en) 1986-09-01
CA1274547C (en) 1990-09-25
ES2001247A6 (es) 1988-05-01
DK396786D0 (da) 1986-08-20
ZA866180B (en) 1987-04-29
FI84817B (fi) 1991-10-15
PT83232B (pt) 1988-07-01
DK396786A (da) 1987-02-22
IL79753A0 (en) 1986-11-30
NO164973C (no) 1990-12-05
AU585052B2 (en) 1989-06-08
EP0220409A2 (en) 1987-05-06
FI84817C (fi) 1992-01-27
FI863353A0 (fi) 1986-08-19
EP0220409A3 (en) 1988-12-14
NO164973B (no) 1990-08-27
KR870002046A (ko) 1987-03-28

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Legal Events

Date Code Title Description
MM Patent lapsed
MM Patent lapsed

Owner name: MERRELL DOW PHARMACEUTICALS INC.