FI853198A0 - PHARMACEUTICAL COMPOSITION INNEHAOLLANDE I VATTEN INSTABILA ELLER BEGRAENSAT LOESLIGA LAEKEMEDEL OCH FOERFARANDE FOER FRAMSTAELLNING AV DEM. - Google Patents

PHARMACEUTICAL COMPOSITION INNEHAOLLANDE I VATTEN INSTABILA ELLER BEGRAENSAT LOESLIGA LAEKEMEDEL OCH FOERFARANDE FOER FRAMSTAELLNING AV DEM.

Info

Publication number
FI853198A0
FI853198A0 FI853198A FI853198A FI853198A0 FI 853198 A0 FI853198 A0 FI 853198A0 FI 853198 A FI853198 A FI 853198A FI 853198 A FI853198 A FI 853198A FI 853198 A0 FI853198 A0 FI 853198A0
Authority
FI
Finland
Prior art keywords
loesliga
instabila
begraensat
vatten
eller
Prior art date
Application number
FI853198A
Other languages
Finnish (fi)
Other versions
FI86140C (en
FI853198L (en
FI86140B (en
Inventor
Bernhard Willi Werner Mueller
Ulrich Brauns
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6217510&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI853198(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of FI853198A0 publication Critical patent/FI853198A0/en
Publication of FI853198L publication Critical patent/FI853198L/en
Application granted granted Critical
Publication of FI86140B publication Critical patent/FI86140B/en
Publication of FI86140C publication Critical patent/FI86140C/en

Links

Classifications

    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B82—NANOTECHNOLOGY
    • B82Y—SPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00—Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/69—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
    • A61K47/6949—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes
    • A61K47/6951—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes using cyclodextrin
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08B—POLYSACCHARIDES; DERIVATIVES THEREOF
    • C08B37/00—Preparation of polysaccharides not provided for in groups C08B1/00 - C08B35/00; Derivatives thereof
    • C08B37/0006—Homoglycans, i.e. polysaccharides having a main chain consisting of one single sugar, e.g. colominic acid
    • C08B37/0009—Homoglycans, i.e. polysaccharides having a main chain consisting of one single sugar, e.g. colominic acid alpha-D-Glucans, e.g. polydextrose, alternan, glycogen; (alpha-1,4)(alpha-1,6)-D-Glucans; (alpha-1,3)(alpha-1,4)-D-Glucans, e.g. isolichenan or nigeran; (alpha-1,4)-D-Glucans; (alpha-1,3)-D-Glucans, e.g. pseudonigeran; Derivatives thereof
    • C08B37/0012—Cyclodextrin [CD], e.g. cycle with 6 units (alpha), with 7 units (beta) and with 8 units (gamma), large-ring cyclodextrin or cycloamylose with 9 units or more; Derivatives thereof
    • C08B37/0015—Inclusion compounds, i.e. host-guest compounds, e.g. polyrotaxanes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nanotechnology (AREA)
  • Materials Engineering (AREA)
  • Biotechnology (AREA)
  • Public Health (AREA)
  • Biochemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Polymers & Plastics (AREA)
  • Organic Chemistry (AREA)
  • Biophysics (AREA)
  • Veterinary Medicine (AREA)
  • General Engineering & Computer Science (AREA)
  • Medical Informatics (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Epidemiology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Novel pharmaceutical compositions comprise inclusion compounds of drugs, which are instable or only sparingly soluble in water, with partially etherified beta -cyclodextrin derivatives having hydroxyalkyl and optionally additional alkyl groups.
FI853198A 1983-12-21 1985-08-20 Process for the preparation of a pharmaceutical preparation containing a water-insoluble or water-unstable drug FI86140C (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE19833346123 DE3346123A1 (en) 1983-12-21 1983-12-21 PHARMACEUTICAL PREPARATIONS OF SUBSTANCES MEDICAL OR UNSTABLE IN WATER AND METHOD FOR THE PRODUCTION THEREOF
DE3346123 1983-12-21
PCT/EP1984/000417 WO1985002767A1 (en) 1983-12-21 1984-12-20 Pharmaceutical compositions containing drugs which are instable or sparingly soluble in water and methods for their preparation
EP8400417 1984-12-20

Publications (4)

Publication Number Publication Date
FI853198A0 true FI853198A0 (en) 1985-08-20
FI853198L FI853198L (en) 1985-08-20
FI86140B FI86140B (en) 1992-04-15
FI86140C FI86140C (en) 1992-07-27

Family

ID=6217510

Family Applications (1)

Application Number Title Priority Date Filing Date
FI853198A FI86140C (en) 1983-12-21 1985-08-20 Process for the preparation of a pharmaceutical preparation containing a water-insoluble or water-unstable drug

Country Status (17)

Country Link
EP (1) EP0149197B2 (en)
JP (1) JPS61500788A (en)
AT (1) ATE51145T1 (en)
AU (1) AU565966B2 (en)
CA (1) CA1222697A (en)
CY (1) CY1689A (en)
DE (2) DE3346123A1 (en)
DK (1) DK175288B1 (en)
FI (1) FI86140C (en)
HK (1) HK131293A (en)
HU (1) HU200943B (en)
LU (1) LU90283I2 (en)
NL (1) NL980009I1 (en)
NO (1) NO2000007I1 (en)
SG (1) SG24893G (en)
WO (1) WO1985002767A1 (en)
ZA (1) ZA8410042B (en)

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AU565966B2 (en) 1987-10-01
SG24893G (en) 1993-08-06
EP0149197B1 (en) 1990-03-21
CA1222697A (en) 1987-06-09
HUT40561A (en) 1987-01-28
AU3835285A (en) 1985-07-12
DK359585A (en) 1985-08-07
EP0149197A3 (en) 1985-08-14
DK175288B1 (en) 2004-08-09
JPH0570612B2 (en) 1993-10-05
NL980009I1 (en) 1998-05-06
HK131293A (en) 1993-12-03
NO2000007I1 (en) 2000-09-21
DK359585D0 (en) 1985-08-07
LU90283I2 (en) 1998-11-03
DE3346123A1 (en) 1985-06-27
CY1689A (en) 1994-01-14
ZA8410042B (en) 1985-09-25
FI86140C (en) 1992-07-27
WO1985002767A1 (en) 1985-07-04
DE3481680D1 (en) 1990-04-26
ATE51145T1 (en) 1990-04-15
JPS61500788A (en) 1986-04-24
FI853198L (en) 1985-08-20
EP0149197B2 (en) 1997-01-08
FI86140B (en) 1992-04-15
EP0149197A2 (en) 1985-07-24
HU200943B (en) 1990-09-28

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