DK359585D0 - PHARMACEUTICAL CONDITIONS CONTAINING USTABLE OR SPARELY SOLUBLE IN WATER AND PROCEDURES FOR THEIR PREPARATION - Google Patents

PHARMACEUTICAL CONDITIONS CONTAINING USTABLE OR SPARELY SOLUBLE IN WATER AND PROCEDURES FOR THEIR PREPARATION

Info

Publication number
DK359585D0
DK359585D0 DK359585A DK359585A DK359585D0 DK 359585 D0 DK359585 D0 DK 359585D0 DK 359585 A DK359585 A DK 359585A DK 359585 A DK359585 A DK 359585A DK 359585 D0 DK359585 D0 DK 359585D0
Authority
DK
Denmark
Prior art keywords
water
ustable
procedures
preparation
conditions containing
Prior art date
Application number
DK359585A
Other languages
Danish (da)
Other versions
DK359585A (en
DK175288B1 (en
Inventor
Bernhard Willi Werner Mueller
Ulrich Brauns
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6217510&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK359585(D0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of DK359585A publication Critical patent/DK359585A/en
Publication of DK359585D0 publication Critical patent/DK359585D0/en
Application granted granted Critical
Publication of DK175288B1 publication Critical patent/DK175288B1/en

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Classifications

    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B82—NANOTECHNOLOGY
    • B82Y—SPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00—Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/69—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
    • A61K47/6949—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes
    • A61K47/6951—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes using cyclodextrin
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08B—POLYSACCHARIDES; DERIVATIVES THEREOF
    • C08B37/00—Preparation of polysaccharides not provided for in groups C08B1/00 - C08B35/00; Derivatives thereof
    • C08B37/0006—Homoglycans, i.e. polysaccharides having a main chain consisting of one single sugar, e.g. colominic acid
    • C08B37/0009—Homoglycans, i.e. polysaccharides having a main chain consisting of one single sugar, e.g. colominic acid alpha-D-Glucans, e.g. polydextrose, alternan, glycogen; (alpha-1,4)(alpha-1,6)-D-Glucans; (alpha-1,3)(alpha-1,4)-D-Glucans, e.g. isolichenan or nigeran; (alpha-1,4)-D-Glucans; (alpha-1,3)-D-Glucans, e.g. pseudonigeran; Derivatives thereof
    • C08B37/0012—Cyclodextrin [CD], e.g. cycle with 6 units (alpha), with 7 units (beta) and with 8 units (gamma), large-ring cyclodextrin or cycloamylose with 9 units or more; Derivatives thereof
    • C08B37/0015—Inclusion compounds, i.e. host-guest compounds, e.g. polyrotaxanes

Abstract

Novel pharmaceutical compositions comprise inclusion compounds of drugs, which are instable or only sparingly soluble in water, with partially etherified beta -cyclodextrin derivatives having hydroxyalkyl and optionally additional alkyl groups.
DK198503595A 1983-12-21 1985-08-07 Pharmaceutical agents containing drugs which are unstable or sparingly soluble in water, and methods for their preparation DK175288B1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE19833346123 DE3346123A1 (en) 1983-12-21 1983-12-21 PHARMACEUTICAL PREPARATIONS OF SUBSTANCES MEDICAL OR UNSTABLE IN WATER AND METHOD FOR THE PRODUCTION THEREOF
DE3346123 1983-12-21
EP8400417 1984-12-20
PCT/EP1984/000417 WO1985002767A1 (en) 1983-12-21 1984-12-20 Pharmaceutical compositions containing drugs which are instable or sparingly soluble in water and methods for their preparation

Publications (3)

Publication Number Publication Date
DK359585A DK359585A (en) 1985-08-07
DK359585D0 true DK359585D0 (en) 1985-08-07
DK175288B1 DK175288B1 (en) 2004-08-09

Family

ID=6217510

Family Applications (1)

Application Number Title Priority Date Filing Date
DK198503595A DK175288B1 (en) 1983-12-21 1985-08-07 Pharmaceutical agents containing drugs which are unstable or sparingly soluble in water, and methods for their preparation

Country Status (17)

Country Link
EP (1) EP0149197B2 (en)
JP (1) JPS61500788A (en)
AT (1) ATE51145T1 (en)
AU (1) AU565966B2 (en)
CA (1) CA1222697A (en)
CY (1) CY1689A (en)
DE (2) DE3346123A1 (en)
DK (1) DK175288B1 (en)
FI (1) FI86140C (en)
HK (1) HK131293A (en)
HU (1) HU200943B (en)
LU (1) LU90283I2 (en)
NL (1) NL980009I1 (en)
NO (1) NO2000007I1 (en)
SG (1) SG24893G (en)
WO (1) WO1985002767A1 (en)
ZA (1) ZA8410042B (en)

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HU181703B (en) * 1980-05-09 1983-11-28 Chinoin Gyogyszer Es Vegyeszet Process for producing aqueus solutuins of water insoluble or hardly soluble vitamines, steroides, localanesthetics, prostanoides and non-steroid and antiphlogistic agents
US4371673A (en) * 1980-07-21 1983-02-01 The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services Water soluble forms of retinoids

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DE3346123A1 (en) 1985-06-27
LU90283I2 (en) 1998-11-03
NL980009I1 (en) 1998-05-06
CY1689A (en) 1994-01-14
FI86140C (en) 1992-07-27
SG24893G (en) 1993-08-06
JPS61500788A (en) 1986-04-24
JPH0570612B2 (en) 1993-10-05
DK359585A (en) 1985-08-07
NO2000007I1 (en) 2000-09-21
EP0149197A2 (en) 1985-07-24
DK175288B1 (en) 2004-08-09
FI853198L (en) 1985-08-20
DE3481680D1 (en) 1990-04-26
HU200943B (en) 1990-09-28
AU3835285A (en) 1985-07-12
FI853198A0 (en) 1985-08-20
ATE51145T1 (en) 1990-04-15
FI86140B (en) 1992-04-15
CA1222697A (en) 1987-06-09
ZA8410042B (en) 1985-09-25
HUT40561A (en) 1987-01-28
EP0149197A3 (en) 1985-08-14
HK131293A (en) 1993-12-03
AU565966B2 (en) 1987-10-01
EP0149197B2 (en) 1997-01-08
WO1985002767A1 (en) 1985-07-04
EP0149197B1 (en) 1990-03-21

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