FI842142A7 - Foerfarande foer framstaellning av farmakologiskt aktiva substituerade acylpiperazinokinazoliner. - Google Patents

Foerfarande foer framstaellning av farmakologiskt aktiva substituerade acylpiperazinokinazoliner. Download PDF

Info

Publication number
FI842142A7
FI842142A7 FI842142A FI842142A FI842142A7 FI 842142 A7 FI842142 A7 FI 842142A7 FI 842142 A FI842142 A FI 842142A FI 842142 A FI842142 A FI 842142A FI 842142 A7 FI842142 A7 FI 842142A7
Authority
FI
Finland
Prior art keywords
farmakologiskt
acylpiperazinokinazoliner
aktiva
substituerade
foerfarande foer
Prior art date
Application number
FI842142A
Other languages
English (en)
Finnish (fi)
Other versions
FI842142A0 (fi
Inventor
Jan Koenig
Miroslav Rajsner
Vaclav Trcka
Svetluse Macova
Original Assignee
Spofa Vereinigte Pharma Werke
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Spofa Vereinigte Pharma Werke filed Critical Spofa Vereinigte Pharma Werke
Publication of FI842142A0 publication Critical patent/FI842142A0/fi
Publication of FI842142A7 publication Critical patent/FI842142A7/fi
Priority to SU864028548A priority Critical patent/SU1572409A3/ru

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI842142A 1983-06-01 1984-05-29 Foerfarande foer framstaellning av farmakologiskt aktiva substituerade acylpiperazinokinazoliner. FI842142A7 (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
SU864028548A SU1572409A3 (ru) 1984-05-29 1986-11-25 Подающее устройство лесоуборочных машин дл поперечной подачи бревна и его обрубки

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CS833905A CS236097B1 (en) 1983-06-01 1983-06-01 Acylderivatives of 2-piperazinochinazoline and method of their preparation

Publications (2)

Publication Number Publication Date
FI842142A0 FI842142A0 (fi) 1984-05-29
FI842142A7 true FI842142A7 (fi) 1984-12-02

Family

ID=5380483

Family Applications (1)

Application Number Title Priority Date Filing Date
FI842142A FI842142A7 (fi) 1983-06-01 1984-05-29 Foerfarande foer framstaellning av farmakologiskt aktiva substituerade acylpiperazinokinazoliner.

Country Status (8)

Country Link
US (1) US4775673A (cs)
JP (1) JPS606668A (cs)
CH (1) CH661726A5 (cs)
CS (1) CS236097B1 (cs)
DE (1) DE3419223C2 (cs)
FI (1) FI842142A7 (cs)
FR (1) FR2547822B1 (cs)
GB (1) GB2142625B (cs)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CS236097B1 (en) * 1983-06-01 1985-05-15 Jan Koenig Acylderivatives of 2-piperazinochinazoline and method of their preparation
US4775223A (en) * 1984-09-20 1988-10-04 Canon Kabushiki Kaisha Lactic acid derivative, liquid crystal composition containing same and liquid crystal device
AT384218B (de) * 1985-12-04 1987-10-12 Gerot Pharmazeutika Verfahren zur herstellung von neuen chinazolin-derivaten
RU2124511C1 (ru) * 1993-05-14 1999-01-10 Фармасьютикал Ко., Лтд Производные пиперазина
IT1270993B (it) * 1994-03-18 1997-05-26 Recordati Chem Pharm Derivati chinzolilamminici attivi come alfa-antagonisti
US6248888B1 (en) 1997-11-14 2001-06-19 Teva Pharmaceutical Industries Ltd. Process for the preparation of terazosin hydrochloride dihydrate
US6313294B1 (en) 1998-02-04 2001-11-06 Development Center For Biotechnology Process for preparing amides
FR2951447B1 (fr) 2009-10-19 2012-10-19 Rhodia Operations Composes de type ether-amide et utilisattions

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1156973A (en) * 1965-07-06 1969-07-02 Quinazoline Derivatives
US3511836A (en) * 1967-12-13 1970-05-12 Pfizer & Co C 2,4,6,7-tetra substituted quinazolines
US3574212A (en) * 1968-02-02 1971-04-06 Pfizer Quinazolinylureas
US4189484A (en) * 1977-11-08 1980-02-19 Mitsubishi Yuka Pharmaceutical Co., Ltd. Antihypertensive quinazoline derivatives
US4309541A (en) * 1978-09-20 1982-01-05 Ciba-Geigy Corporation Piperidinyl-lactams
US4287341A (en) * 1979-11-01 1981-09-01 Pfizer Inc. Alkoxy-substituted-6-chloro-quinazoline-2,4-diones
GB2068961B (en) * 1980-02-13 1983-11-30 Sankyo Co Quinazoline derivatives
US4377581A (en) * 1980-03-03 1983-03-22 Pfizer Inc. Chloro- and alkoxy-substituted-2,4-diaminoquinazolines
JPS5793977A (en) * 1980-11-26 1982-06-11 Sankyo Co Ltd Acylaminoquinazoline derivative and its preparation
EP0060081B1 (en) * 1981-03-05 1985-07-17 Pfizer Inc. Piperazinoquinazoline antihypertensives, processes for preparing them, pharmaceutical compositions containing them, and immunogenic protein conjugates formed from them
US4440769A (en) * 1983-02-11 1984-04-03 Abbott Laboratories 2-(4-Phenylalkanoylpiperazin-1-yl) quinazoline compounds, pharmaceutical compositions and method of producing α1 antagonistic activity
CS236097B1 (en) * 1983-06-01 1985-05-15 Jan Koenig Acylderivatives of 2-piperazinochinazoline and method of their preparation

Also Published As

Publication number Publication date
FR2547822B1 (fr) 1986-12-26
DE3419223C2 (de) 1995-09-07
CS236097B1 (en) 1985-05-15
FR2547822A1 (fr) 1984-12-28
FI842142A0 (fi) 1984-05-29
GB8413741D0 (en) 1984-07-04
GB2142625B (en) 1987-04-15
JPS606668A (ja) 1985-01-14
DE3419223A1 (de) 1984-12-06
GB2142625A (en) 1985-01-23
CH661726A5 (de) 1987-08-14
US4775673A (en) 1988-10-04

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Legal Events

Date Code Title Description
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Owner name: SPOFA SPOJENE PODNIKU PRO ZDRAVOTNICKOU